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Cat. No.	Product Name	Form
C0048	Deacetylase Inhibitor Cocktail (100× in 70% DMSO) 去乙酰化酶抑制剂 Cocktail（100× in 70% DMSO）	Solution (100× <em>in</em> 70% DMSO)
C0001	Protease Inhibitor Cocktail (EDTA-Free, 100× in DMSO) 蛋白酶抑制剂 Cocktail (EDTA-Free, 100× in DMSO)	Solution (EDTA-Free,100× <em>in</em> DMSO)
C0005	Cell Counting Kit-8 (CCK-8) Cell Counting Kit-8 (CCK-8)	Solution <em>in</em> bottle
C0003	Phosphatase Inhibitor Cocktail II (100× DMSO) 磷酸酶抑制剂 Cocktail II (100× DMSO)	Solution (100× <em>in</em> DMSO)
C0002	Phosphatase Inhibitor Cocktail I (100× ddH2O) 磷酸酶抑制剂 Cocktail I (100× ddH2O)	Solution (100× <em>in</em> ddH2O)
C0004	Phosphatase Inhibitor Cocktail III (2 Tubes, 100x) 磷酸酶抑制剂 Cocktail III (2 Tubes, 100x)	2 Tube Solution (100×)
C0051	Penicillin-Streptomycin Solution (100×), Sterile 青霉素-链霉素双抗溶液（100×），灭菌	Solution <em>in</em> bottle
C0090	Mag Beads Streptavidin (1 μm) 链霉亲和素磁珠 (1 μm)
C0050	BCA Protein Quantification Kit BCA蛋白浓度测定试剂盒	Solution <em>in</em> bottle
C0052	Penicillin-Streptomycin-Amphotericin B Solution (100×), Sterile 青霉素-链霉素-两性霉素B三抗溶液（100×），灭菌	Solution <em>in</em> bottle
C0105	Protein A Immunoprecipitation Kit Protein A 免疫沉淀试剂盒
CL0060	Estrogen Receptor inhibitor kit Estrogen Receptor inhibitor kit
CL0079	Adenosine Receptor inhibitor kit Adenosine Receptor inhibitor kit
CL0120	Bcr-Abl inhibitor/degrader kit Bcr-Abl inhibitor/degrader kit
CL0123	AMPK inhibitor/activator kit AMPK inhibitor/activator kit
CL0078	Glucocorticoid Receptor inhibitor/activator kit Glucocorticoid Receptor inhibitor/activator kit
CL0083	Dehydrogenase inhibitor kit Dehydrogenase inhibitor kit
CL0118	p38 inhibitor kit p38 inhibitor kit
CL0143	PKA/cAMP inhibitor/activator kit PKA/cAMP inhibitor/activator kit
CL0119	Histone Demethylase inhibitor kit Histone Demethylase inhibitor kit
CL0061	Histone Methyltransferase inhibitor kit Histone Methyltransferase inhibitor kit
CL0067	Sodium Channel inhibitor kit Sodium Channel inhibitor kit
CL0141	Notch pathway inhibitor kit Notch pathway inhibitor kit
CL0070	GABA Receptor inhibitor kit GABA Receptor inhibitor kit
CL0122	ACE inhibitor kit ACE inhibitor kit
CL0147	c-FMS inhibitor kit c-FMS inhibitor kit
CL0058	EGFR inhibitor kit EGFR inhibitor kit
CL0135	ROCK inhibitor kit ROCK inhibitor kit
CL0112	PKC inhibitor kit PKC inhibitor kit
CL0101	STAT inhibitor kit STAT inhibitor kit
CL0093	PARP inhibitor kit PARP inhibitor kit
CL0117	DPP4 inhibitor kit DPP4 inhibitor kit
CL0125	AChE inhibitor kit AChE inhibitor kit
CL0146	JNK inhibitor kit JNK inhibitor kit
CL0068	VEGFR inhibitor kit VEGFR inhibitor kit
C0113	Magrose Beads Heparin 肝素磁珠
C0104B	Protein A/G Immunomagnetic Beads Protein A/G 免疫沉淀磁珠
C0116B	Protein G Immunomagnetic Beads Protein G 免疫沉淀磁珠
C0117	Protein L Immunoprecipitation Kit Protein L 免疫沉淀试剂盒
CL0071	PDGFR inhibitor kit PDGFR inhibitor kit
C0092	Mag Beads Streptavidin (2.8 μm) 链霉亲和素磁珠 (2.8 μm)
CL0113	ER stress pathway inhibitor/inducer kit ER stress pathway inhibitor/inducer kit
CL0056	CDK inhibitor kit CDK inhibitor kit
CL0130	DUB inhibitor kit DUB inhibitor kit
CL0084	FGFR inhibitor kit FGFR inhibitor kit
CL0094	FLT3 inhibitor kit FLT3 inhibitor kit
CL0114	ERK inhibitor kit ERK inhibitor kit
CL0091	MEK inhibitor kit MEK inhibitor kit
CL0116	MAO inhibitor kit MAO inhibitor kit
CL0109	Ras inhibitor kit Ras inhibitor kit
CL0105	Sirtuin inhibitor/activator kit Sirtuin inhibitor/activator kit
CL0150	DNA Methyltransferase/Demethylase inhibitor kit DNA Methyltransferase/Demethylase inhibitor kit
CL0144	Endothelin Receptor antagonist kit Endothelin Receptor antagonist kit
CL0074	Microtubule/Tubulin inhibitor kit Microtubule/Tubulin inhibitor kit
CL0107	Src inhibitor/activator kit Src inhibitor/activator kit
CL0142	MMP inhibitor kit MMP inhibitor kit
CL0089	c-Met/HGFR inhibitor kit c-Met/HGFR inhibitor kit
CL0057	PI3K inhibitor kit PI3K inhibitor kit
CL0134	p53 inhibitor/reactivator kit p53 inhibitor/reactivator kit
CL0090	RNA Synthesis inhibitor/activator kit RNA Synthesis inhibitor/activator kit
CL0115	Proton Pump inhibitor kit Proton Pump inhibitor kit
C0105	Protein A Immunoprecipitation Kit Protein A 免疫沉淀试剂盒
CL0060	Estrogen Receptor inhibitor kit Estrogen Receptor inhibitor kit
CL0079	Adenosine Receptor inhibitor kit Adenosine Receptor inhibitor kit
CL0120	Bcr-Abl inhibitor/degrader kit Bcr-Abl inhibitor/degrader kit
CL0123	AMPK inhibitor/activator kit AMPK inhibitor/activator kit
CL0078	Glucocorticoid Receptor inhibitor/activator kit Glucocorticoid Receptor inhibitor/activator kit
CL0083	Dehydrogenase inhibitor kit Dehydrogenase inhibitor kit
CL0118	p38 inhibitor kit p38 inhibitor kit
CL0143	PKA/cAMP inhibitor/activator kit PKA/cAMP inhibitor/activator kit
CL0119	Histone Demethylase inhibitor kit Histone Demethylase inhibitor kit
CL0061	Histone Methyltransferase inhibitor kit Histone Methyltransferase inhibitor kit
CL0067	Sodium Channel inhibitor kit Sodium Channel inhibitor kit
CL0141	Notch pathway inhibitor kit Notch pathway inhibitor kit
CL0070	GABA Receptor inhibitor kit GABA Receptor inhibitor kit
CL0122	ACE inhibitor kit ACE inhibitor kit
CL0147	c-FMS inhibitor kit c-FMS inhibitor kit
CL0058	EGFR inhibitor kit EGFR inhibitor kit
CL0135	ROCK inhibitor kit ROCK inhibitor kit
CL0112	PKC inhibitor kit PKC inhibitor kit
CL0101	STAT inhibitor kit STAT inhibitor kit
CL0093	PARP inhibitor kit PARP inhibitor kit
CL0117	DPP4 inhibitor kit DPP4 inhibitor kit
CL0125	AChE inhibitor kit AChE inhibitor kit
CL0146	JNK inhibitor kit JNK inhibitor kit
CL0068	VEGFR inhibitor kit VEGFR inhibitor kit
C0113	Magrose Beads Heparin 肝素磁珠
C0104B	Protein A/G Immunomagnetic Beads Protein A/G 免疫沉淀磁珠
C0116B	Protein G Immunomagnetic Beads Protein G 免疫沉淀磁珠
C0117	Protein L Immunoprecipitation Kit Protein L 免疫沉淀试剂盒
CL0071	PDGFR inhibitor kit PDGFR inhibitor kit
C0092	Mag Beads Streptavidin (2.8 μm) 链霉亲和素磁珠 (2.8 μm)
CL0113	ER stress pathway inhibitor/inducer kit ER stress pathway inhibitor/inducer kit
CL0056	CDK inhibitor kit CDK inhibitor kit
CL0130	DUB inhibitor kit DUB inhibitor kit
CL0084	FGFR inhibitor kit FGFR inhibitor kit
CL0094	FLT3 inhibitor kit FLT3 inhibitor kit
CL0114	ERK inhibitor kit ERK inhibitor kit
CL0091	MEK inhibitor kit MEK inhibitor kit
CL0116	MAO inhibitor kit MAO inhibitor kit
CL0109	Ras inhibitor kit Ras inhibitor kit
CL0069	JAK inhibitor kit JAK inhibitor kit
CL0096	Wnt/β-catenin/PORCN inhibitor/activator kit Wnt/β-catenin/PORCN inhibitor/activator kit
CL0045	COX inhibitor kit COX inhibitor kit
CL0139	ROS inhibitor kit ROS inhibitor kit
C0089	Mag Beads Streptavidin (300 nm) 链霉亲和素磁珠 (300 nm)
C0093	Mag Beads Streptavidin (3 μm) 链霉亲和素磁珠 (3 μm)
C0108	Magrose Beads Protein G Protein G 琼脂糖磁珠
C0094	Mag Beads Streptavidin (5 μm) 链霉亲和素磁珠 (5 μm)
C0095	Magrose Beads Streptavidin (Ultra-suspension) 琼脂糖链霉亲和素磁珠
C0105B	Protein A Immunomagnetic Beads Protein A 免疫沉淀磁珠
C0117B	Protein L Immunomagnetic Beads Protein L 免疫沉淀磁珠
CEPY-0006	Human Cystatin SN/CST1 ELISA Pair Set Human Cystatin SN/CST1 ELISA 抗体对
CEPY-0003	Human Cystatin C/CST3 ELISA Pair Set Human Cystatin C/CST3 ELISA 抗体对
CL0137	E1/E2/E3 Enzyme inhibitor kit E1/E2/E3 Enzyme inhibitor kit
CL0131	SGLT inhibitor kit SGLT inhibitor kit
CL0128	HMGCR inhibitor kit HMGCR inhibitor kit
CL0075	c-Kit inhibitor kit c-Kit inhibitor kit
CL0138	Carbonic Anhydrase inhibitor kit Carbonic Anhydrase inhibitor kit
CL0077	Reverse Transcriptase inhibitor kit Reverse Transcriptase inhibitor kit
CL0102	Akt inhibitor/activator kit Akt inhibitor/activator kit
CL0080	TGFβ signaling pathway inhibitor/activator kit TGFβ signaling pathway inhibitor/activator kit
CL0129	Aurora Kinase inhibitor kit Aurora Kinase inhibitor kit
CL0098	HER2 inhibitor kit HER2 inhibitor kit
CL0076	PPAR inhibitor/activator kit PPAR inhibitor/activator kit
CL0064	PDE inhibitor kit PDE inhibitor kit
CL0092	GSK-3 inhibitor kit GSK-3 inhibitor kit
CL0140	BTK inhibitor kit BTK inhibitor kit
C0046	RIPA Lysis Buffer (Middle) RIPA裂解液(中)	Solution <em>in</em> bottle
C0045	RIPA Lysis Buffer (Strong) RIPA裂解液(强)	Solution <em>in</em> bottle
C0006	SYBR Green qPCR Master Mix (No ROX) SYBR Green qPCR Master Mix (No ROX)	Solution <em>in</em> bottle
C0008	SYBR Green qPCR Master Mix (Low ROX) SYBR Green qPCR Master Mix (Low ROX)	Solution <em>in</em> bottle
C0047	RIPA Lysis Buffer (Weak) RIPA裂解液(弱)	Solution <em>in</em> bottle
C0007	SYBR Green qPCR Master Mix (High ROX) SYBR Green qPCR Master Mix (High ROX)	Solution <em>in</em> bottle

Cat. No.	Product Name	Target	Signaling Pathways
T10682L	CARM1-IN-1 CARM1-IN-7G	Histone Methyltransferase	Chromatin/Epigenetic
	CARM1-IN-1 (CARM1-IN-7G) 是 CARM1 的选择性抑制剂，IC50 为 8.6 μM。 CARM1-IN-1 对 PRMT1 和 SET7 的活性较弱，IC50 > 600 μM。
T11332	FUBP1-IN-1 FUBP1–IN-1	Others	Others
	FUBP1 - in-1, with an IC50 value of 11.0 M, is an effective FUSE binding protein 1 (FUBP1) inhibitor that can interfere with the binding of FUBP1 to its SINGLE-strand target DNA FUSE sequence.
T11025	hDHODH-IN-3 DHODH-IN-2	Dehydrogenase	Metabolism
	hDHODH-IN-3 是人二氢乳清酸脱氢酶的抑制剂，pMIC50 值为 8.6。 hDHODH-IN-3 可以抑制麻疹病毒的复制。
T11029	hDHODH-IN-5 DHODH-IN-7	Dehydrogenase	Metabolism
	hDHODH-IN-5 是人源二氢乳清酸脱氢酶的抑制剂 (hDHODH, IC50 = 0.91 μM)。
T40290	CDK12-IN-5 CDK12-IN-5
	CDK12-IN-5 is a pyrazolotriazine compound that effectively inhibits CDK12, with an IC50 value of 23.9 nM at a high ATP concentration of 2 mM. However, CDK12-IN-5 does not exhibit inhibitory effects on CDK2/Cyclin E (IC50 = 173 μM) and CDK9/Cyclin T1 (IC50 = 127 μM) at the same high ATP concentration of 2 mM, as stated in WO2021116178A1.
T39705	ATG7-IN-1 ATG7-IN-1	Autophagy	Autophagy
	ATG7-IN-1 是一种选择性 ATG7 抑制剂，IC50 为 62 nM。
T8763	PTGR2-IN-1 PTGR2-IN-22	Others	Others
	PTGR2-IN-1 是有效的 PTGR2抑制剂，IC50为 ~0.7 μM。它能够提高转染 PTGR2 的 HEK293T 细胞 15-keto-PGE2 依赖的 PPARγ 转录活性。
T40443	JAK2-IN-6 JAK2-IN-6	JAK	Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
	JAK2-IN-6是一种有效的、有选择性的 JAK2抑制剂(ic50为22.86 μg/mL),是一种多取代氨基噻唑衍生物。JAK2-IN-6抑制 JAK2酶的活性，通过干扰与 JAK2相关的信号通路，从而对 JAK2失调的特定疾病产生治疗作用，对 JAK1和JAK3不显示出活性。JAK2是一种参与调节细胞生长和分裂的信号通路的蛋白质。JAK2的异常激活与多种疾病有关，包括某些类型的癌症和炎症性疾病。JAK2-IN-6对癌细胞具有抗增殖活性。
T11028	hDHODH-IN-4 DHODH-IN-5	Dehydrogenase	Metabolism
	hDHODH-IN-4 (DHODH-IN-5) 是一种有效的人二氢硼酸脱氢酶 (DHODH) 抑制剂，对人重组 DHODH 的 pIC50 为 7.8。hDHODH-IN-4 抑制麻疹病毒复制，pMIC50 为 8.8。
T40109	APOL1-IN-1 APOL1-IN-1	Others	Others
	APOL1-IN-1是一种有效的载脂蛋白 L1(APOL1) 的抑制剂，可用于研究局灶节段性肾小球硬化 (FSGS) 和非糖尿病肾病 (NDKD) 的发病原理，促进对此类疾病的研究。
T9863	PKCiota-IN-2 PKCiota-IN-49	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKCiota-IN-2 (PKCiota-IN-49) 是一种有效的 PKCiota (PKC-ι) 抑制剂，IC50 为 2.8 nM。PKCiota-IN-2 还抑制 PKC-α 和 PKC-ε，IC50 分别为 71 nM 和 350 nM。
T38684	AKR1C3-IN-4 AKR1C3-IN-4	NADPH	Metabolism
	AKR1C3-IN-4 是醛酮还原酶 1C3 (AKR1C3) 选择性抑制剂，IC50为 0.56 μM。它在去势抵抗性前列腺癌中有研究的价值。
T40146	Sec61-IN-1 Sec61-IN-1	Others	Others
	Sec61-IN-1是一种有效的Sec61抑制剂。
T39764	ALK2-IN-4 ALK2-IN-4
	ALK2-IN-4, a highly effective ALK2 inhibitor.
T35899	JAK1-IN-8 JAK1-IN-8	JAK	Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
	JAK1-IN-8，Janus 激酶 1 (JAK1)的特异性抑制剂（IC50<500 nM）。
T38905	FATP1-IN-1 FATP1-IN-1	Others	Others
	FATP1-IN-1 是一种强效的脂肪酸转运蛋白1（FATP1）抑制剂。它能有效抑制对FATP1功能至关重要的重组人类或小鼠的酰辅酶A合成酶活性。其抑制特征通过IC50值体现，分别为人类FATP1的0.046 μM 和小鼠FATP1的0.60 μM。
T2043	Mutant IDH1-IN-1 IDH1-IN-1	Dehydrogenase; Isocitrate Dehydrogenase (IDH)	Metabolism
	Mutant IDH1-IN-1 是 IDH1突变体的选择性抑制剂，能够作用于突变体 IDH1 R132C/R132C (IC50:4 nM) ，IDH1 R132H/R132H (IC50:42 nM) ，IDH1 R132H/WT (IC50:80 nM) 和野生型 IDH1 (IC50:143 nM)。
T11031	hDHODH-IN-7 DHODH-IN-9	Dehydrogenase	Metabolism
	hDHODH-IN-7 (DHODH-IN-9) 是一种含嗪的类似物，是一种人二氢乳清酸酯脱氢酶抑制剂。hDHODH-IN-7 具有抗病毒作用，pMIC50 为 7.4。
T40350	HPK1-IN-4 HPK1-IN-4	MAPK	MAPK
	HPK1-IN-4是一种HPK1（MAPK41）抑制剂，IC 50为0.061 nM。HPK1-IN-4常被作为临床前免疫治疗工具化合物。
T39389	KDM2B-IN-2 KDM2B-IN-2	Histone Demethylase	Chromatin/Epigenetic
	KDM2B-IN-2是一种有效的组蛋白去甲基化酶 (KDM2B) 抑制剂。
T35900	JAK2-IN-7 JAK2-IN-7	JAK	Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
	JAK2-IN-7 是一种选择性 JAK2抑制剂，对 JAK2，SET-2 和 Ba/F3V617F 细胞的IC50为 3、11.7 和 41 nM。 JAK2-IN-7 的选择性是 JAK1, JAK3，FLT3 的 14 倍以上。JAK2-IN-7 刺激细胞周期停滞在 G0/G1 期，并诱导肿瘤细胞凋亡 (apoptosis)，具有抗肿瘤活性。
T4438	Porcn-IN-1 Porcupine-IN-1	Porcupine	Stem Cells
	Porcn-IN-1 (Porcupine-IN-1) 是一种有效的porcupine 抑制剂(IC50:0.5±0.2 nM)。
T8336	OGG1-IN-08 OGG1-IN-O8	Others	Others
	OGG1-IN-08 (OGG1-IN-O8) 是 8-氧鸟嘌呤 DNA 糖基酶-1 抑制剂(IC50:0.22 μM)。它能够减少 OGG1 的糖基化酶和裂解酶活性。
T38078	TLR7/8-IN-1 TLR7/8-IN-1	TLR	Immunology/Inflammation
	TLR7/8-IN-1，是一种结晶态TLR7/TLR8抑制剂，对于自身免疫性疾病研究具有重要价值[1]。
T15660	KHK-IN-1 KHK-IN-8,Ketohexokinase inhibitor 8	Others	Others
	KHK-IN-1 (KHK-IN-8) 是一种选择性的、细胞膜渗透性的己酮糖激酶 (KHK) 抑制剂 (IC50=12 nM; F=34%)。KHK-IN-1 抑制 HepG2 细胞裂解液中 F1P 生成，IC50为400 nM。KHK-IN-1 可用于研究糖尿病和肥胖症。
T12345	CBP/p300-IN-3 P300/CBP-IN-3	Histone Acetyltransferase	Chromatin/Epigenetic
	CBP/p300-IN-3 (P300/CBP-IN-3) 是一种组蛋白乙酰转移酶抑制剂。
T28865	STAT3-IN-B9 STAT3 IN B9,B9	STAT	JAK/STAT signaling; Stem Cells
	STAT3-IN-B9 (B9) 是异常 STAT3 激活的抑制剂，可抑制 MDA-MB-468、MDA-MB-231 和 DU145 等肿瘤细胞的增殖。
T39752	CDK12-IN-2 CDK12 inhibitor 2,CDK12-IN-2	CDK	Cell Cycle/Checkpoint
	CDK12-IN-2 (CDK12 inhibitor 2) 是一种有效的选择性 CDK12 抑制剂，对 CDK12、CDK2、CDK7 和 CDK9 的 IC50 为 52 nM、>100 μM、>10 μM 和 16 μM。 CDK12-IN-2可用于研究CDK12的功能。
T78823	Quorum Sensing-IN-3 QS-IN-1	Antibacterial	Microbiology/Virology
	Quorum Sensing-IN-3 (QS-IN-1)是一种对细菌群体感应有抑制作用的化合物，可抑制细菌之间的信息交流，抑制生物膜的形成。
T79607	h-NTPDase-IN-2 hNTPDase-IN-2	Phosphatase	Metabolism
	h-NTPDase-IN-2 是一种广谱 NTPDase 抑制剂，对多种 h-NTPDas 亚型都具有抑制作用。
T39669	TLR7/8/9-IN-1 TLR7/8/9-IN-1	TLR	Immunology/Inflammation
	TLR7/8/9-IN-1 是具有口服活性的Toll 样受体7/8/9小分子拮抗剂，IC50为43 nM。
T24133	HDAC8-IN-20a HDAC8 IN 20a,HDAC8IN20a,HDAC8 inhibitor-20a,HDAC8 inhibitor 20a	HDAC	Chromatin/Epigenetic; DNA Damage/DNA Repair
	HDAC8-IN-20a (HDAC8 inhibitor-20a) 是一种有效的、具有选择性的HDAC8抑制剂，IC50为27 nM。HDAC8-IN-20a 可阻断生长受体存活信号的激活。
T11580	Heme Oxygenase-1-IN-1 HO-1-IN-1	Reactive Oxygen Species	Immunology/Inflammation; Metabolism; NF-κB
	Heme Oxygenase-1-IN-1 (HO-1-IN-1) 是一种血红素加氧酶 1 (HO-1) 抑制剂，IC50=250 nM。
T29017	TrxR1-IN-B19 TrxR1INB19,Go Y015,TrxR1 IN B19,Go-Y015	Others	Others
	TrxR1-IN-B19 (TrxR1 IN B19) 是一种 TrxR1 抑制剂，通过靶向 TrxR1 和 ROS 介导的 ER 应激激活，通过小分子选择性杀死胃癌细胞。
T24131	HDAC3-IN-T247 HDAC3 inhibitor T247,HDAC3 inhibitor-T247,HDAC3 IN T247,T247	Histone Demethylase; Antiviral	Chromatin/Epigenetic; Immunology/Inflammation
	HDAC3-IN-T247 (HDAC3 inhibitor T247) 是一种具有选择性和有效性的组蛋白去乙酰化酶 3（HDAC3）抑制剂，具有抗癌和抗病毒活性。HDAC3-IN-T247 以剂量依赖的方式诱导人结肠癌 HCT116 细胞中 NF-κB 乙酰化。HDAC3-IN-T247 抑制癌细胞增殖。
T24410	LIMK-IN-22j LIMK IN 22j,LIMK inhibitor-22j,LIMK inhibitor 22j	LIM Kinase	Cell Cycle/Checkpoint
	LIMK-IN-22j (LIMK inhibitor 22j) 是一种有效的选择性 LIMK 抑制剂。
T24793	SIRT6-IN-5 SIRT6 inhibitor5,SIRT6 IN 5,SIRT6 inhibitor-5,SIRT6 inhibitor 5	Sirtuin	Chromatin/Epigenetic; DNA Damage/DNA Repair
	SIRT6-IN-5（SIRT6 inhibitor 5）是一种具有有效性和选择性的 SIRT6 抑制剂，IC50 值为 34 μM。SIRT6-IN-5 具有免疫抑制和化疗增敏作用，可增加 H3K9 的乙酰化并增加培养细胞中的葡萄糖摄取，减少 T 细胞增殖。
T23709	alphaSYN-IN-NAB2 alphaSYN inhibitor NAB2,alphaSYNINNAB2,alphaSYN-IN-NAB2,NAB2,alphaSYN inhibitor-NAB2
	alphaSYN-IN-NAB2 是一种神经元保护剂，是一种由 NAB2基因编码的蛋白质。NAB2 高效且具有选择性地保护多种细胞免受 α-syn 毒性。NAB2 对依赖于 E3 泛素连接酶 Rsp5/Nedd4 的内体转运具有促进作用。NAB2 确定 α-syn 生物学中的一个可活性分子节点，该节点可以纠正其潜在病理学的多个方面，包括功能失调的内体和内质网到高尔基体囊泡的运输。NAB2参与细胞分化、凋亡和应激反应等细胞过程，可用来研究癌症、神经发育和神经元活动。
T23867	Cdc7-IN-7c Cdc7 inhibitor-7c,Cdc7 inhibitor 7c,Cdc7 IN 7c	CDK	Cell Cycle/Checkpoint
	Cdc7-IN-7c (Cdc7 inhibitor-7c) 具有抗肿瘤活性，对肝癌，肺癌，肾癌，脑癌，宫颈癌有抑制作用。
T9017	HPK1-IN-2 Thieno[2,3-b]pyridin-6(7H)-one, 4-amino-5-[6-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]-HPK1-IN-2,HPK1-IN-2	Others; FLT; Src	Angiogenesis; Others; Tyrosine Kinase/Adaptors
	HPK1-IN-2 (Thieno[2,3-b]pyridin-6(7H)-one, 4-amino-5-[6-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]-HPK1-IN-2) 是一种有效且具有口服活性的造血祖细胞激酶-1 抑制剂(HPK1；IC50<0.05 µM)。它还抑制 Lck (0.05 µM<IC50<0.5 µM) 和 Flt3 (IC50<0.05 µM) 激酶活性，具有抗肿瘤活性。
T15782	Lp-PLA2-IN-1 Lp-PLA2 inhibitor 1,Lp-PLA2 -IN-1	Phospholipase	Metabolism
	Lp-PLA2-IN-1 (Lp-PLA2 inhibitor 1) 是脂蛋白相关磷脂酶 A2(Lp-PLA2) 抑制剂。它有潜力用于动脉粥样硬化、阿尔茨海默氏病的研究。
T63208L	Aβ-IN-1 TFA Aβ-IN-1 TFA（2766509-32-2 Free base）
	Aβ-IN-1 TFA 能够抑制和逆转不同类型的蛋白质聚集。
T3161L	BACE-IN-1 acetate BACE-IN-1 acetate (350228-37-4，Free base)	BACE	Neuroscience
	BACE-IN-1 acetate (BACE-IN-1 acetate (350228-37-4，Free base)) 已被用作 BACE1 抑制剂测定中的 β 位淀粉样前体蛋白 (APP) 裂解酶-1 (BACE1) 抑制剂。 β-位点淀粉样前体蛋白 (APP) 切割酶-1 (BACE1)是一种天冬氨酸蛋白酶，属于蛋白酶家族，由六个腔内半胱氨酸残基组成。这些残基有助于形成三个分子间二硫键和 N-连接的糖基化位点。
T10792L	CHK1-IN-4 hydrochloride CHK1-IN-4 hydrochloride（2120398-41-4 Free base）	Chk	Cell Cycle/Checkpoint
	CHK1-IN-4 hydrochloride 是有效的checkpoint kinase 1 (chk1) 抑制剂，对肿瘤细胞中 chk1 磷酸化具有有效的抑制作用。CHK1-IN-4 hydrochloride 显示出抗肿瘤活性。
T19206	β-Lactamase-IN-1 4-(1,3-dihydroxypropan-2-yl)-6-methoxypyrido[2,3-b]pyrazin-3-one,beta-lactamase-IN-1	Antibacterial	Microbiology/Virology
	β-Lactamase-IN-1 (4-(1,3-dihydroxypropan-2-yl)-6-methoxypyrido[2,3-b]pyrazin-3-one) 是一种 β-Lactamase 抑制剂，针对淋病奈瑟菌的感染。
T28652	S6K1-IN-DG2 S6K1 Inhibitor DG2,S6K1-Inhibitor-DG2,S6K1 IN DG2,S6K1INDG2,S6K1InhibitorDG2	mTOR	PI3K/Akt/mTOR signaling
	S6K1-IN-DG2(S6K1InhibitorDG2) 是一种有效的 p70S6K 抑制剂，IC50 值小于 100 nM。
TP2160L1	YAP-TEAD-IN-1 acetate YAP-TEAD-IN-1 acetate (1659305-78-8 Free base)	YAP	Stem Cells
	YAP-TEAD-IN-1 acetate 是一种有效的、竞争性的 YAP-TEAD 相互作用抑制剂，IC50 为 25 nM。
T23897	CLK1/2-IN-3 CLK1/2 inhibitor 3,CLK1/2-inhibitor-3,CLK1/2 IN 3,CLK1/2IN3	CDK	Cell Cycle/Checkpoint
	CLK1/2-IN-3(Cpd-3) 是一种具有高效性和选择性的 CLK1 和 CLK2 抑制剂，抗增殖活性，抑制 CLK1、CLK2、SRPK1、SRPK2、SRPK3 的的活性。CLK1/2-IN-3 可诱导核斑点扩大，可诱导S6K pre-mRNA选择性剪接和随后抑制多种癌细胞类型细胞生长。
T15572	IN-1130	ALK	Angiogenesis; Tyrosine Kinase/Adaptors
	IN-1130 是一种选择性的 ALK5 抑制剂，对 ALK5 介导的 Smad3 磷酸化、酪蛋白和 p38α 丝裂原活化蛋白激酶的 ALK5 磷酸化，IC50 值为 5.3 nM、36 nM 和 4.3 μM。
T63399L	mTOR/HDAC-IN-1 HCl mTOR/HDAC-IN-1 HCl（2815286-02-1 Free base)	HDAC; mTOR	Chromatin/Epigenetic; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
	mTOR/HDAC-IN-1 HCl 是一种有效的 mTOR 和 HDAC 双重抑制剂，具有潜在的抗炎、抗增殖、自噬和诱导凋亡作用，可用于研究癌症。mTOR/HDAC-IN-1 HCl 是一种有效的 mTOR 和 HDAC 双重抑制剂，具有潜在的抗炎、抗增殖、自噬和凋亡诱导作用，可用于研究癌症。

Cat. No.	Product Name	Target	Signaling Pathways
T5070	LC3-mHTT-IN-AN2 5,7-二羟基-4-苯基香豆素,5,7-Dihydroxy-4-phenylcoumarin	Antibacterial; Autophagy; ATTECs	Autophagy; Microbiology/Virology; PROTAC
	LC3-mHTT-IN-AN2 (5,7-Dihydroxy-4-phenylcoumarin) 是一种 mHTT-LC3 接头化合物，可与突变亨廷顿蛋白(mHTT) 和 LC3B 相互作用。它将 mHTT 靶向自噬体以等位基因选择性方式降低培养的亨廷顿病小鼠神经元中的 mHTT 水平。它存在于西番莲植物中，具有抗菌活性。
T19289	DL-Glyceric Acid Glyceric Acid (20% in Water,ca.2 mol/L)	Others	Others
	DL-glyceric acid is a compound that is excessively secreted in the urine of patients with D-glyceric aciduria.
T73070	STAT3-IN-14
	STAT3-IN-14是一种STAT3抑制剂，具有STAT3磷酸化抑制活性，可直接与 STAT3的铰链区结合。
T75511	BChE-IN-10
	BChE-IN-10 (compound 6)，一种从白芨 (Bletilla striata) 分离提取的丁酰胆碱酯酶 (BChE) 混合型抑制剂，具有 6.4 μM 的IC50，适用于阿尔兹海默症 (AD) 研究。
T81684	Neuroinflammatory-IN-1
	Neuroinflammatory-IN-1 (Compound 5)，作为一种抗神经炎剂，对NO生成表现出显著的抑制效果，其IC50为65.4 μM。
T73073	PTP1B-IN-21
	PTP1B-IN-21 是蛋白酪氨酸磷酸酶 1B (PTP1B) 的选择性抑制剂 (IC50=1.56 μM)，抑制力超出高度同源 T 细胞蛋白酪氨酸磷酸酶 (TCPTP；IC50>100 μM)，PTP1B 是抑制 2 型糖尿病的重要靶点。
T73202	BChE-IN-11
	BChE-IN-11 是一种有效的、选择性的、非竞争性BChE(丁基胆碱酯酶)抑制剂，其IC50为 2.1 μM。BChE-IN-11 可用于阿尔茨海默病 (AD) 的研究。
T75545	PCSK9-IN-9
	PCSK9-IN-9 是一种天然来源的异香豆素。PCSK9-IN-9 可抑制原蛋白转化酶枯草菌素 kexin 型 9 (PCSK9)、IDOL 和 SREBP2的 mRNA 表达水平。PCSK9-IN-9 抑制 PCSK9的 IC50为 11.9 μM。
T75513	BChE-IN-12
	BChE-IN-12 (compound 12) 为一种高效BChE非竞争性抑制剂，其IC50值为2.3 μM。该化合物可从白芨(Bletilla striata)中分离提取，适用于阿尔兹海默症(AD)的研究。
T73072	PTP1B-IN-20
	PTP1B-IN-20 是蛋白酪氨酸磷酸酶 1B (PTP1B) 的选择性抑制剂 (IC50=1.05 μM)，抑制力超出高度同源 T 细胞蛋白酪氨酸磷酸酶 (TCPTP；IC50=78.0 μM)，PTP1B 是抑制 2 型糖尿病的重要靶点。
T81629	OAT1/3-IN-2
	OAT1/3-IN-2（化合物8）是一种针对OAT1和OAT3的双重抑制剂。该化合物能够以10 μM的浓度逆转Cys-Hg对HEK-OAT1细胞的毒害作用，并可能对肾脏具有保护效应。OAT1/3-IN-2适用于研究汞导致的肾脏损伤。
T80713	α-Glucosidase-IN-37
	α-Glucosidase-IN-37（Compound 11）展示出中等水平的抑制作用，能够抑制LPS诱导的NO产生，并在巨噬细胞中表现出23.7 μM的IC50值。该化合物对α-Glucosidase的抑制活性相对较弱。
T75612	α-Glucosidase-IN-24
	α-Glucosidase-IN-24 (Compound 13) 是一种α-Glucosidase 抑制剂，IC50为 451 μM，可以从Swertia kouitchensis 中分离得到。
T75544	AChE/BChE-IN-11
	AChE/BChE-IN-11 (compound 1) 是一种有效的 AChE 和 BChE 双重抑制剂，AChE 和BChE 的IC50值为分别为 70 和 71 μM。AChE/BChE-IN-11 是一种天然产物，可以从朝鲜蓟叶中分离得到。AChE/BChE-IN-11 可用于阿尔茨海默病 (AD) 研究。
T75504	Xanthine oxidase-IN-8
	Xanthine oxidase-IN-8 (Icarisids J) (Compound 7) 是一种 XOD 抑制剂，IC50值为 29.71 μM。
T75505	Xanthine oxidase-IN-9
	Xanthine oxidase-IN-9 (Icarisids E) (Compound 2)，一种黄嘌呤氧化酶 (XOD) 高效抑制剂，具有31.81 μM 的 IC50 值。
T81630	OAT1/3-IN-1
	OAT1/3-IN-1（化合物7）是针对OAT1和OAT3的双重抑制剂。该化合物能逆转Cys-Hg（10 μM）对HEK-OAT1细胞引起的毒害，表明其对肾脏有潜在的保护效应。OAT1/3-IN-1适合用于探究汞引起的肾脏损伤机制研究。
T72581	SARS-CoV MPro-IN-2
	SARS-CoVMPro-IN-2 是一种有效的SARS-CoV-2 Mpro 抑制剂，IC50sub>值为 72.07 nM。病毒的主要蛋白酶 Mpro 作为加工病毒多蛋白的主要酶，有助于 SARS-CoV-2 在宿主细胞中的复制和转录，并已被定性为药物发现的有吸引力的靶点。SARS-CoVMPro-IN-2 具有研究 COVID-19 的潜力。
TN3270	(R)-3β-Hydroxy steroid sulfotransferase-IN-11	Others	Others
	(R)-3β-Hydroxy steroid sulfotransferase-IN-11 在生命科学相关研究中具有广泛的应用。
TJS1779	Protosappanin A 原苏木素A,PTA	NADPH-oxidase; IL Receptor; IκB/IKK; TNF; NF-κB; TLR; ROS; COX; HIV Protease; JAK; NO Synthase; STAT	Angiogenesis; Apoptosis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Microbiology/Virology; Neuroscience; NF-κB; Proteases/Proteasome; Stem Cells
	Protosappanin A (PTA) 是从苏木中分离得到的免疫抑制成分和主要联苯化合物，通过下调 JAK2和 STAT3的磷酸化，抑制 JAK2/STAT3依赖的炎症通路。
T1879	3-Methyladenine 3-MA,3-甲基腺嘌呤,NSC 66389	Mitophagy; PI3K; Endogenous Metabolite; Autophagy	Autophagy; Metabolism; PI3K/Akt/mTOR signaling
	3-Methyladenine (3-MA) 是一种 PI3K 抑制剂，选择性抑制 IB 类 PI3Kγ (IC50=60 μM) 和 III 类 VPS34 (IC50=25 μM)。3-Methyladenine 具有自噬抑制活性。
T19146	5,6-Dihydrouridine	Endogenous Metabolite	Metabolism
	5,6-Dihydrouridine 是一种修饰碱基，存在于真核生物、细菌和某些古细菌tRNA D 环的保守位置。
T4898	Potassium 1-carboxyvinyl hydrogenphosphate PEP-K,磷酸烯醇丙酮酸单钾盐,Phospho(enol)pyruvic acid monopotassium	Others; Endogenous Metabolite	Metabolism; Others
	Potassium 1-carboxyvinyl hydrogenphosphate (PEP-K) 是内源性代谢产物的一种。
T15157	Dodecanoylcarnitine Lauroylcarnitine	Endogenous Metabolite	Metabolism
	Dodecanoylcarnitine（(-)-Lauroylcarnitine）和脂肪酸氧化紊乱有关，使用 Dodecanoylcarnitine 可使鲑鱼降钙素的通透性增加。
T20225	Dicentrine, (-)- L-Dicentrine,荷包牡丹碱,NSC 251699,NSC251699,NSC-251699	Others	Others
	Dicentrine, (-)- (NSC-251699) 是一种在几种植物物种中发现的非卟啉生物碱，在小鼠内脏痛的急性模型中显示出显著的镇痛活性。
T4722	O-Acetyl-L-serine hydrochloride	Others; Endogenous Metabolite	Metabolism; Others
	O-Acetyl-L-serine hydrochloride 是内源性代谢产物的一种。
TN1698	Glucotropaeolin potassium 金莲葡糖硫苷钾盐,Glucotropaeolin,Benzylglucosinolate potassium,Glucotropaeolin Potassium Salt	Others	Others
	Glucotropaeolin potassium (Benzylglucosinolate potassium) 存在于十字花科蔬菜中，并且可适度减少动物的自发性DNA 损伤。
T4809	Pyrimidine 嘧啶,Metadiazine	Others; Endogenous Metabolite	Metabolism; Others
	Pyrimidine (Metadiazine) 是内源性代谢产物的一种。
T5282	5-Methyluridine Ribothymidine,5-甲基尿甙,Thymine riboside	Others; Endogenous Metabolite	Metabolism; Others
	5-Methyluridine (Thymine riboside) 是发现于人体液中的内源性甲基化核苷。
T5076	L-Allothreonine L-别苏氨酸,L-allo-Threonine	Others; Endogenous Metabolite	Metabolism; Others
	L-Allothreonine (L-allo-Threonine) 是内源性代谢产物的一种。
T4969	Guanosine 5'-triphosphate trisodium salt 鸟苷-5'-三磷酸三钠盐,GTP Trisodium salt,5'-GTP trisodium salt	Endogenous Metabolite	Metabolism
	Guanosine 5'-triphosphate trisodium salt (5'-GTP trisodium salt) 为G蛋白(G proteins)信号转导过程中的活化剂。
TJS0387	Desoxyrhaponticin 去氧土大黄苷,Deoxyrhapontin,脱氧土大黄苷,Deoxyrhaponticin	Apoptosis; Fatty Acid Synthase	Apoptosis; Metabolism
	Desoxyrhaponticin (Deoxyrhaponticin) 是来自西藏营养食品唐古特大黄中的一种二苯乙烯苷。它是脂肪酸合成酶抑制剂，抑制细胞内 FAS 活性，下调人乳腺癌 MCF-7细胞中 FAS 的表达。它是控制糖尿病餐后高血糖的潜在药物。
T4713	Phosphorylcholine chloride calcium salt tetrahydrate Phosphocholine chloride calcium salt tet,胆碱磷酸氯化钙四水,CalciuM Phosphorylcholine Tetrahydrate	Others; Endogenous Metabolite	Metabolism; Others
	Phosphorylcholine chloride calcium salt tetrahydrate (Phosphocholine chloride calcium salt tet) 是内源性代谢产物的一种。
T0710	L-Cycloserine Levcycloserine,Levcicloserina,(-)-Cycloserine,(S)-Cycloserine,Levcycloserinum,环丝氨酸,(S)-4-Amino-3-isoxazolidone	HIV Protease; GABA Receptor	Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Proteases/Proteasome
	L-Cycloserine ((-)-Cycloserine) 不可逆地抑制大肠杆菌以及各种动物大脑中的 GABA 吡哆醛 5'-磷酸依赖性转氨酶，导致体内抑制性神经递质 γ-氨基丁酸水平升高。
T5875	4-Methoxycinnamic acid	Endogenous Metabolite	Metabolism
	4-Methoxycinnamic acid 是天然苯丙烷类化合物。
T13509	4-Vinylphenol	Apoptosis; Endogenous Metabolite	Apoptosis; Metabolism
	4-Vinylphenol 是酒中乳酸菌对香豆酸和阿魏酸的代谢产物，在白花蛇舌草中发现。 4-Vinylphenol 在体内诱导细胞凋亡。
T3O2784	Vitamin B6 维生素B6	Others	Others
	Vitamin B6 是人体某些辅酶的成分，参与多种代谢反应，特别是与氨基酸代谢有关。维生素B6在防治妊娠和放射病呕吐中的临床应用。
TQ0273	Neopterin D-(+)-Neopterin,2-Amino-6-((1S,2R)-1,2,3-trihydroxypropyl)pteridin-4(3H)-one,新蝶呤	Endogenous Metabolite	Metabolism
	Neopterin (D-(+)-Neopterin) 是三磷酸腺苷的一种分解产物，是细胞免疫系统激活的标志物。
T4104	Ophiopojaponin C 麦冬皂苷C,Ophiopogonin C	Others	Others
	Ophiopogonin C' pharmacological activities may be related to the substances in nucleus mainly.
T5647	6-Methylcoumarin Toncarine,6-甲基香豆素	Others	Others
	6-Methylcoumarin (Toncarine) 是一种合成香料，广泛用于化妆品中。
T3S0693	Blinin	Others	Others
	Blinin 是一种二萜，分离自植物 Conyza blinii 中。
T5812	Zinc Phytate	Others	Others
	Zinc Phytate 存在于食物中，对人类吸收营养有重要意义。
T4814	(R)-5-Oxopyrrolidine-2-carboxylic acid D-Pyroglutamic acid,(R)-(+)-2-Pyrrolidone-5-carboxylic acid,D-焦谷氨酸	Others; Endogenous Metabolite	Metabolism; Others
	(R)-5-Oxopyrrolidine-2-carboxylic acid (D-Pyroglutamic acid) 是内源性代谢产物的一种。
T3912	Saikosaponin B1 柴胡皂苷B1,柴胡皂苷 B1	Others	Others
	Saikosaponin B1 是柴胡的生物活性成分，具有抗癌作用。它能够靶向SMO 抑制 Hedgehog 通路，显著抑制髓母细胞瘤模型中的肿瘤生长。
T5309	Dimethylamine hydrochloride N,N-Dimethylamine,二甲胺盐酸盐	Others	Others
	Dimethylamine hydrochloride (N,N-Dimethylamine) 大量存在于人类尿液中。
TN5086	Syringetin	Others	Others
	Syringetin 是一种存在于葡萄和葡萄酒中的类黄酮衍生物，可促进 B16F10 细胞的黑色素生成，抑制人肺腺癌中成骨细胞介导的破骨细胞生成。
T0925	Allantoin Glyoxyldiureide,尿囊素,5-Ureidohydantoin	Endogenous Metabolite; Imidazoline Receptor	Metabolism; Neuroscience
	Allantoin (Glyoxyldiureide) 是一种存在于尿液和植物中的尿素乙内酰脲，用于皮肤病制剂。
T24711	Ricinine 1,2-Dihydro-4-methoxy-1-methyl-2-oxonicotinonitrile,蓖麻碱,Ricinin,Ritsinin	Others	Others
	Ricinine (1,2-Dihydro-4-methoxy-1-methyl-2-oxonicotinonitrile) 是蓖麻植物中的一种主要生物碱，在 CCl4 诱导的肝损伤中具有保肝作用。
T5S0890	Oleandrin Neriostene,Folinerin,Foliandrin,欧夹竹桃苷	Apoptosis; ATPase; Potassium Channel; Sodium Channel	Apoptosis; Membrane transporter/Ion channel
	Oleandrin (Folinerin) 是夹竹桃属中的一种类固醇，可抑制Na+/K+-ATPase 活性，IC50为 620 nM。
T4852	Trimyristin Trimyristoylglycerol,Tritetradecanoin,三肉豆蔻酸甘油酯,Glyceryl trimyristate,甘油三肉豆蔻酸酯,1,2,3-Tritetradecanoylglycerol	Phosphatase; Endogenous Metabolite; AChE	Metabolism; Neuroscience
	Trimyristin (Tritetradecanoin) 是一种 Myristica fragransHoutt 的有效成分，能够显著抑制乙酰胆碱酯酶 (AChE)，酸性和碱性磷酸酶 (ACP/ALP) 特性。它对 AChE，ACP 和 ALP 的 IC50分别为 0.11、0.16 和 0.18 mM。
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	1016 种酪氨酸激酶抑制剂的独特集合，可用于高通量筛选和高内涵筛选；
L2550	谷氨酰胺代谢化合物库	565 compounds
	565 种谷氨酰胺代谢相关的分子，可以用于高通量和高内涵筛选；
L9411	半胱氨酸共价化合物库	70 compounds
	半胱氨酸共价库包含 70 个化合物。
L2300	离子通道库	931 compounds
	931 种与离子通道相关的生物活性小分子化合物的特有集合，用于离子通道相关的疾病和药物研究，可用于高通量筛选和高内涵筛选；
L3800	NF-κB 通路分子库	729 compounds
	729 个 NF-κB 信号通路相关的小分子化合物的特有集合，用于高通量、高内涵筛选；
L9900	药用辅料化合物库	182 compounds
	182 种 FDA 批准药品中的非活性成分集合
L1310	细胞骨架化合物库	759 compounds
	759 种细胞骨架相关的化合物，可以用于高通量和高内涵筛选；
L1400	MAPK 抑制剂库	365 compounds
	365 种与MAPK 信号通路相关的生物活性小分子化合物的特有集合，可用于高通量筛选和高内涵筛选；
L8600	泛素化化合物库	210 compounds
	210 种泛素化相关的小分子，用于高通量和高内涵筛选；
L3410	临床前化合物库	701 compounds
	701 种临床前小分子化合物的特有集合，用于高通量、高内涵筛选；
L1600	激酶抑制剂库	2720 compounds
	2720 种激酶抑制剂/调节剂的独特集合，用于特定靶向激酶，可用于高通量筛选和高内涵筛选；
L4700	免疫/炎症分子化合物库	4720 compounds
	4720 种具有抗炎症活性的化合物的特有集合，可用于高通量筛选和高内涵筛选；
L5510	肝脏毒性化合物库	1001 compounds
	1001 个肝脏毒性化合物的特有集合，可用于高通量、高内涵筛选，是毒理学研究的良好工具；

Cat. No.	Product Name	Species	Expression System
TMPY-01442	DMBT1 Protein, Human, Recombinant (His) GP340,deleted in malignant brain tumors 1,...	Human	HEK293 Cells
	Deleted in malignant brain tumors 1 protein, also known as glycoprotein 34, surfactant pulmonary-associated D-binding protein, DMBT1 and GP34, is a secreted protein which belongs to theDMBT1 family. DMBT1 contains 2CUB domains, 14SRCR domains and 1ZP domain. It is highly expressed in alveolar and macrophage tissues. In some macrophages, expression is detected on the membrane, and in other macrophages, it is strongly expressed in the phagosome/phagolysosome compartments. Defects in DMBT1 are invo...
TMPY-02033	CD44 Protein, Human, Recombinant (His) CD44 molecule (Indian blood group),IN,MC56...	Human	HEK293 Cells
	CD44 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 23.4 kDa and the accession number is P16070-1.
TMPY-01775	AIM2 Protein, Human, Recombinant (GST) absent in melanoma 2,PYHIN4	Human	Baculovirus Insect Cells
	AIM2, Absent In Melanoma 2 is a member of the interferon-inducible HIN-200 protein family that contains an amino-terminal pyrin domain and a carboxy-terminal oligonucleotide/oligosaccharide-binding domain, senses cytoplasmic DNA by means of its oligonucleotide/oligosaccharide-binding domain and interacts with ASC (apoptosis-associated speck-like protein containing a CARD) through its pyrin domain to activate caspase-1. In response to foreign cytoplasmic DNA, AIM2 forms an inflammasome, resulting...
TMPY-03430	RheB Protein, Human, Recombinant (His) Ras homolog enriched in brain,RHEB2	Human	Baculovirus Insect Cells
	RHEB is a recently discovered member of the Ras superfamily that may be involved in neural plasticity. This function is novel and not typically associated with the Ras proteins. RHEB gene is a member of the small GTPase superfamily and encodes a lipid-anchored, cell membrane protein with five repeats of the RAS-related GTP-binding region. RHEB is vital in regulation of growth and cell cycle progression due to its role in the insulin / TOR / S6K signaling pathway. The protein has GTPase activity ...
TMPJ-01125	PEA15 Protein, Human, Recombinant 15 kDa Phosphoprotein Enriched in Astrocyt...	Human	E. coli
	Astrocyticphosphoprotein PEA-15 (PEA15) is a death effector domain (DED)-containing protein. PEA15 is mainly expressed in the central nervous system, principally in astrocytes. Increased PEA15 levels affect tumorigenesis and cancer progression. PEA15 is overexpressed in breast cancers and gliomas as well as in type 2 diabetes. PEA15 blocks Ras-mediated inhibition of integrin activation and modulates the ERK MAP kinase cascade. PEA15 also inhibits RPS6KA3 activities by holding it in the cytoplasm...
TMPY-00580	DCUN1D2 Protein, Human, Recombinant (His) DCN1, defective in cullin neddylation 1, d...	Human	E. coli
	DCUN1D2 Protein, Human, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 32.4 kDa and the accession number is Q6PH85-1.
TMPJ-01126	RheB Protein, Human, Recombinant (GST) RHEB,Ras Homolog Enriched in Brain,GTP-B	Human	E. coli
	GTP-Binding Protein Rheb (RHEB) is a member of the small GTPase superfamily and encodes a lipid-anchored, cell membrane protein with five repeats of the RAS-related GTP-binding region. Highest levels of RHEB can be found in the skeletal and cardiac muscle, and it is vital in the regulation of growth and cell cycle progression due to its role in the Insulin/TOR/S6K signaling pathway. RHEB stimulates the phosphorylation of S6K1 and EIF4EBP1 through activation of mTORC1 signaling, and it activates...
TMPJ-01387	PACSIN2 Protein, Human, Recombinant (His) Protein Kinase C and Casein K...	Human	HEK293 Cells
	Protein Kinase C and Casein Kinase Substrate in Neurons Protein 2 (PACSIN2) is a member of the PACSIN family. PACSIN2 is localized to the plasma membrane via its coiled-coil domain. PACSIN2 is widely expressed and contains one FCH domain and one SH3 domain. PACSIN2 forms homo- and hetero-aggregates with other PACSINs. PACSIN2 may play a role in vesicle formation and transport. In addition, PACSIN2 is involved in linking the actin cytoskeleton with vesicle formation by regulating tubulin polymeri...
TMPJ-00272	RELT/TNFRSF19L Protein, Human, Recombinant (hFc) RELT,TNFRSF19L,Receptor expressed in lymphoid tissu...	Human	HEK293 Cells
	Tumor necrosis factor receptor superfamily member 19L (TNFRSF19L), also known as Receptor expressed in lymphoid tissues and RELT, is a member of the TNF-receptor superfamily. TNFRSF19L is a single-pass type membrane protein and contains one TNFR-Cys repeat. TNFRSF19L is highly expressed in spleen, lymph node, thymus, peripheral blood leukocytes, bone marrow and fetal liver. It has been shown TNFRSF19L activates the NF-kappaB pathway and selectively binds TNF receptor-associated factor 1 (TRAF1)....
TMPY-01710	IkB alpha/NFKBIA Protein, Human, Recombinant (His) IkB α,IKBA,nuclear factor of kappa light polypeptide gene en...	Human	E. coli
	Nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor, alpha (IkB alpha, NFKBIA, or IKBA), is a member of the NF-kappa-B inhibitor family that function to inhibit the NF-kB transcription factor. NFKBIA inhibits NF-kB by masking the nuclear localization signals (NLS) of NF-kB proteins and keeping them sequestered in an inactive state in the cytoplasm. Also, NFKBIA blocks the ability of NF-κB transcription factors to bind to DNA, which is required for NF-kB's proper function...
TMPJ-01307	PACSIN1 Protein, Human, Recombinant (His) Protein Kinase C and Casein K...	Human	HEK293 Cells
	Protein Kinase C and Casein Kinase Substrate in Neurons Protein 1 (PACSIN1) belongs to the PACSIN family. PACSIN1 contains one FCH domain and one SH3 domain. PACSIN1 is highly expressed in the brain and at lower leves in the heart, pancreas, and liver. PACSIN1 may play a role in vesicle formation and transport. PACSIN1 has been shown to interact with DNM1, PACSIN3, Huntingtin, and PACSIN2. In addition, PACSIN1 is phosphorylated by casein kinase 2 (CK2) and protein kinase C (PKC).
TMPH-03747	CCDC112 Protein, Human, Recombinant (His & Myc) Mutated in bladder cancer protein 1,Coiled...	Human	E. coli
	CCDC112 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 61.0 kDa and the accession number is Q8NEF3.
TMPH-01091	CHD1L Protein, Human, Recombinant (His & SUMO) Amplified in liver cancer protein 1,CHD1L,...	Human	E. coli
	DNA helicase which plays a role in chromatin-remodeling following DNA damage. Targeted to sites of DNA damage through interaction with poly(ADP-ribose) and functions to regulate chromatin during DNA repair. Able to catalyze nucleosome sliding in an ATP-dependent manner. Helicase activity is strongly stimulated upon poly(ADP-ribose)-binding. CHD1L Protein, Human, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 37.3 kDa an...
TMPY-03869	DCUN1D1 Protein, Human, Recombinant (His) DCNL1,SCCRO,Tes3,RP42,SCRO,DCUN1L1,DCN1, defective in	Human	E. coli
	DCUN1D1, also known as SCCRO, is part of an E3 ubiquitin ligase complex for neddylation. DCUN1D1 functions to recruit charged E2 and is involved in the release of inhibitory effects of CAND1 on cullin-RING ligase E3 complex assembly and activity. DCUN1D1 binds to the components of the neddylation pathway (Cullin-ROC1, Ubc12, and CAND1) and augments but is not required for cullin neddylation in reactions using purified recombinant proteins. DCUN1D1 also recruits Ubc12 approximately NEDD8 to the C...
TMPJ-00887	NFKB1 Protein, Human, Recombinant (His) Nuclear factor of κ light polypeptide gene enhancer in	Human	E. coli
	The 50 kD protein is a DNA binding subunit of the NF-kappa-B (NFKB) protein complex. NFKB is a transcription regulator that is activated by various intra- and extra-cellular stimuli such as cytokines, oxidant-free radicals, ultraviolet irradiation, and bacterial or viral products. Activated NFKB translocates into the nucleus and stimulates the expression of genes involved in a wide variety of biological functions. Inappropriate activation of NFKB has been associated with a number of inflammatory...
TMPH-00252	Bovine coronavirus (strain Mebus) Protein I (His) IORF,Protein in nucleocapsid ORF,N,I,Acces...	BCoV	E. coli
	Structural protein that is not essential for the viral replication either in tissue culture or in its natural host. Bovine coronavirus (strain Mebus) Protein I (His) is expressed in E. coli expression system with C-6xHis tag. The predicted molecular weight is 25.5 kDa and the accession number is P10525.
TMPH-00255	Bovine coronavirus (strain LSU-94LSS-051) Protein I (His) N internal ORF protein,Accessory prote...	BCoV	E. coli
	Structural protein that is not essential for the viral replication either in tissue culture or in its natural host. Bovine coronavirus (strain LSU-94LSS-051) Protein I (His) is expressed in E. coli expression system with C-6xHis tag. The predicted molecular weight is 24.4 kDa and the accession number is Q9QAR0.
TMPH-00253	Bovine coronavirus (strain 98TXSF-110-LUN) Protein I (His) IORF,N,Protein in nucleocapsid ORF,N i...	BCoV	E. coli
	Structural protein that is not essential for the viral replication either in tissue culture or in its natural host. Bovine coronavirus (strain 98TXSF-110-LUN) Protein I (His) is expressed in E. coli expression system with C-6xHis tag. The predicted molecular weight is 24.4 kDa and the accession number is Q8V431.
TMPH-00256	Bovine coronavirus (strain LY-138) Protein I (His) I,N internal ORF protein,N,Accessory prote...	BCoV	E. coli
	Structural protein that is not essential for the viral replication either in tissue culture or in its natural host. Bovine coronavirus (strain LY-138) Protein I (His) is expressed in E. coli expression system with C-6xHis tag. The predicted molecular weight is 25.4 kDa and the accession number is Q9QAR7.
TMPH-00254	Bovine coronavirus (strain 98TXSF-110-ENT) Protein I (His) Protein I,N internal ORF protein,...	BCoV	E. coli
	Structural protein that is not essential for the viral replication either in tissue culture or in its natural host. Bovine coronavirus (strain 98TXSF-110-ENT) Protein I (His) is expressed in E. coli expression system with C-6xHis tag. The predicted molecular weight is 24.0 kDa and the accession number is Q91A21.

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