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GPCR靶点分子库

GPCR靶点分子库

产品编号 L1500 GPCR Compound Library
  库化合物信息   Excel SDF

G 蛋白偶联受体(GPCR)的超家族是对真核细胞信号传导至关重要的多种跨膜蛋白。 GPCR 启动细胞对各种胞外介质的反应,参与几乎所有常见的人类疾病。近40%的上市药物通过调节 GPCR 功能起作用,70%的在研治疗新方法靶向 GPCR,此外,数百个“孤儿”GPCR(尚未鉴定出天然配体)是许多药物发现计划中研究的焦点。GPCR 靶向候选药物必须是对靶蛋白具有高亲和、特异性和合理的膜渗透性。TargetMol GPCR 靶向化合物库是由 1940 种与 G 蛋白及其耦联受体相关的生物活性小分子化合物的特有集合。用于GPCR 靶向的药物研发,GPCR 相关科学研究和药物筛选,可用于高通量、高内涵筛选。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 1940种与G蛋白及其耦联受体相关的生物活性小分子化合物,所有小分子都具有良好的生物和药理活性,部分是FDA批准的上市药物;
  • 是筛选GPCR 靶向药物的强大工具,也可用于用于制药公司和生物技术公司在各项研究和药物开发项目中GPCR的筛选;
  • 据估计大约200个孤儿GPCR功能是未知的,因此,使用我们的GPCR小分子化合物库来筛选功能未知的GPCR可能会产生潜在的新型GPCR候选药;
  • GPCR化合物库含有与受体相关的小分子,包括5-HT 受体、多巴胺受体、 阿片受体、肾上腺素受体、大麻素受体、mGluR和 ETA-受体等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

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包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L1500)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

5-HT Receptor (368)
Adrenergic Receptor (260)
Dopamine Receptor (228)
Histamine Receptor (175)
GPR (104)
Prostaglandin Receptor (98)
Adenosine Receptor (96)
Opioid Receptor (88)
Ras (72)
Apoptosis (67)
Cannabinoid Receptor (67)
Autophagy (65)
Endogenous Metabolite (61)
AChR (50)
CXCR (39)
S1P Receptor (37)
Hedgehog/Smoothened (34)
LPL Receptor (33)
Neurokinin receptor (32)
Sigma receptor (29)
Norepinephrine (26)
Serotonin Transporter (26)
Protease-activated Receptor (26)
Endothelin Receptor (24)
Antibacterial (24)
Glucagon Receptor (23)
SGLT (22)
Neuropeptide Y Receptor (21)
P2Y Receptor (21)
cAMP (21)
Calcium Channel (21)
Potassium Channel (20)
PDE (20)
Guanylate cyclase (19)
LPA Receptor (18)
OX Receptor (17)
Leukotriene Receptor (16)
GTPase (16)
Vasopressin Receptor (16)
P450 (15)
Bradykinin Receptor (14)
Rho (13)
Melanocortin Receptor (12)
Smo (12)
cholecystokinin (12)
Neurotensin Receptor (12)
GPCR19 (12)
NO Synthase (12)
Parasite (11)
Influenza Virus (11)
GHSR (11)
GRK (10)
Melatonin Receptor (10)
COX (10)
CaSR (10)
Sodium Channel (9)
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NF-κB (9)
Somatostatin (9)
Raf (9)
TRP/TRPV Channel (8)
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Bombesin Receptor (7)
Oxytocin Receptor (7)
PPAR (7)
Annexin A (7)
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CaMK (7)
HIV Protease (7)
Arrestin (7)
CDK (6)
Monoamine Oxidase (6)
TSH Receptor (6)
Glucocorticoid Receptor (6)
LTR (6)
PI3K (6)
Lipoxygenase (6)
IL Receptor (6)
PKA (6)
MT Receptor (6)
GNRH Receptor (6)
AChE (6)
P-gp (6)
Drug Metabolite (5)
NOS (5)
CGRP Receptor (5)
HCV Protease (5)
TNF (5)
GABA Receptor (5)
Transferase (5)
Mitophagy (5)
CRFR (5)
EGFR (4)
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ROS (4)
P2X Receptor (4)
Histone Methyltransferase (4)
Virus Protease (4)
PKC (4)
ERK (4)
MAO (4)
HER (4)
NMDAR (4)
Immunology/Inflammation related (3)
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STAT (3)
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transporter (2)
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lysosomal autophagy (1)
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GST (1)
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PTEN (1)
Angiotensin-converting Enzyme (ACE) (1)
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Motilin Receptor (1)
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Proteasome (1)
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Trk receptor (1)
LRRK2 (1)
Estrogen Receptor/ERR (1)
Wnt/beta-catenin (1)
Acyltransferase (1)
Serine Protease (1)
Casein Kinase (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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