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黄酮类天然产物库

黄酮类天然产物库

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产品编号 L6120 Flavonoid Natural Product Library
  库化合物信息   Excel SDF

黄酮,是指两个具有酚羟基的苯环(A-与 B-环)通过中央三碳原子相互连结而成的一系列化合物,其基本母核为2-苯基色原酮。黄酮类化合物是中草药中重要的活性物质之一。黄酮类化合物的主要药理作用有抗氧化、抗菌、抗肿瘤以及对心脑血管的保护作用等,其功能涉及清除自由基、炎症通路调控、能量感受通路调控、细胞周期调节等多种复杂机制。例如:黄芩、草豆蔻、红景天和淫羊藿等中药中含有的黄酮类可作为优良的 ROS 清除剂,在蠕虫中已证明黄酮类化合物可以降低氧化应激水平,银杏叶黄酮具有抗炎症、抗环腺苷酸乙酯酶活性、抗组胺活性等多种效用。

TargetMol 黄酮类天然产物库收集了 477 种黄酮类的天然产物,来源包括银杏、苦参、黄芪、忍冬、淫羊藿等多种传统中药材,库中化合物涉及多种生理功能,如芦丁、槲皮素具有扩张冠脉血管作用,橙皮苷具有抗炎作用,木犀草素、黄岑素、黄岑苷均具有一定程度抗菌作用,金雀异黄酮具有抗肿瘤作用等。该库可以为从事药物开发和药理研究的客户提供有力工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 477种黄酮类天然产物的独特集合,可用于高通量筛选和高内涵筛选;
  • 大部分化合物生物活性明确,具有抗肿瘤、抗炎、抗氧化、神经保护等多种功能;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L6120)
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客户使用化合物库发表的文献

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化合物库组成

Apoptosis (70)
Autophagy (50)
NF-κB (36)
Antibacterial (36)
Antioxidant (28)
Endogenous Metabolite (25)
COX (21)
Reactive Oxygen Species (19)
TNF (17)
Influenza Virus (15)
P450 (15)
PPAR (14)
Anti-infection (14)
Akt (12)
NO Synthase (12)
Tyrosinase (12)
Antifungal (11)
PI3K (11)
MMP (11)
HIV Protease (11)
p38 MAPK (10)
BCL (10)
GABA Receptor (10)
STAT (9)
Virus Protease (9)
Nrf2 (8)
Caspase (8)
IL Receptor (8)
ERK (8)
PKC (7)
AChE (7)
Mitochondrial Metabolism (7)
Estrogen Receptor/ERR (7)
ROS (6)
AMPK (6)
Lipoxygenase (6)
Estrogen/progestogen Receptor (6)
PARP (6)
JNK (5)
transporter (5)
Glucosidase (5)
EGFR (5)
Antifection (5)
DNA/RNA Synthesis (5)
Reductase (4)
PDE (4)
Parasite (4)
Interleukin (4)
Dehydrogenase (4)
ATPase (4)
Ferroptosis (4)
P-gp (3)
PKA (3)
Phosphatase (3)
Immunology/Inflammation related (3)
Beta Amyloid (3)
Prostaglandin Receptor (3)
Wnt/beta-catenin (3)
SARS-CoV (3)
Mitophagy (3)
TGF-beta/Smad (3)
Amylase (3)
CDK (3)
MAPK (3)
HSV (3)
TLR (3)
NOS (3)
5-HT Receptor (3)
UGT (3)
p53 (3)
Trk receptor (2)
Acyltransferase (2)
JAK (2)
MEK (2)
HDAC (2)
Xanthine Oxidase (2)
PTEN (2)
RAAS (2)
SGLT (2)
Free radical scavengers (2)
Opioid Receptor (2)
Aromatase (2)
LDL (2)
Sirtuin (2)
Pim (2)
S6 Kinase (2)
Integrin (2)
IGF-1R (2)
Bombesin Receptor (2)
AChR (2)
Antibiotic (2)
NOD (2)
IAP (2)
VEGFR (2)
MAO (2)
Progesterone Receptor (2)
Potassium Channel (2)
Leukotriene Receptor (1)
NMDAR (1)
CCR (1)
mTOR (1)
Thrombopoietin Receptor (1)
RSV (1)
cell cycle arrest (1)
ALK (1)
stilbene oxidase (1)
FGFR (1)
Proteasome (1)
FAAH (1)
Glucocorticoid Receptor (1)
CaSR (1)
Adenosine Receptor (1)
BACE (1)
Sodium Channel (1)
PAI-1 (1)
Histone Acetyltransferase (1)
Adrenergic Receptor (1)
Adenosine deaminase (1)
Drug Metabolite (1)
HCV Protease (1)
Beta-Secretase (1)
E1/E2/E3 Enzyme (1)
CXCR (1)
PERK (1)
CD38 (1)
Dynamin (1)
Serine/threonin kinase (1)
GSK-3 (1)
PGE Synthase (1)
NOD-like Receptor (NLR) (1)
Antiviral (1)
HIF/HIF Prolyl-Hydroxylase (1)
DPP-4 (1)
Phospholipase (1)
CaMK (1)
ROS Kinase (1)
ROR (1)
ABC (1)
c-Met/HGFR (1)
Calcium Channel (1)
Glucokinase (1)
GPR (1)
Norepinephrine (1)
Src (1)
Carbonic Anhydrase (1)
Gamma-secretase (1)
PAFR (1)
TRP/TRPV Channel (1)
HMG-CoA Reductase (1)
MyD88 (1)
Aryl Hydrocarbon Receptor (1)
IκB/IKK (1)
Fatty Acid Synthase (1)
Reverse Transcriptase (1)
hCE (1)
NMU2R (1)
Chloride channel (1)
Androgen Receptor (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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