- 全部删除
- 您的购物车当前为空
Epinastine(WAL801)是一种选择性和口服活性的histamine H1 receptor拮抗剂,主要用于治疗过敏性结膜炎。Epinastine还抑制人嗜酸性粒细胞释放 IL-8,也用作肥大细胞稳定剂,防止其释放组胺。
Epinastine(WAL801)是一种选择性和口服活性的histamine H1 receptor拮抗剂,主要用于治疗过敏性结膜炎。Epinastine还抑制人嗜酸性粒细胞释放 IL-8,也用作肥大细胞稳定剂,防止其释放组胺。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
2 mg | ¥ 128 | In stock | |
5 mg | ¥ 189 | In stock | |
10 mg | ¥ 266 | In stock | |
25 mg | ¥ 427 | In stock | |
50 mg | ¥ 619 | In stock | |
100 mg | ¥ 987 | In stock | |
500 mg | ¥ 2,580 | In stock | |
1 mL x 10 mM (in DMSO) | ¥ 252 | In stock |
Epinastine 相关产品
产品描述 | Epinastine (WAL801) is a selective and orally active histamine H1 receptor antagonist primarily used for treating allergic conjunctivitis. Epinastine also inhibits the release of IL-8 from human eosinophils and acts as a mast cell stabiliser to prevent the release of histamine. |
体外活性 | 方法:Epinastine(1nM-100μM)处理不同促分泌剂诱导的分离的人皮肤肥大细胞、嗜碱性粒细胞和嗜酸性粒细胞,研究其是否能影响这些细胞的体外激活作用。 |
体内活性 | In receptor binding studies, Epinastine shows a high affinity to H1-receptors in the guinea pig ileum. Epinastine inhibits histamine-induced reactions in the skin or the lung of rats, dogs and guinea pigs [1]. |
别名 | 依匹斯汀, WAL801, WAL 801 |
分子量 | 249.31 |
分子式 | C16H15N3 |
CAS No. | 80012-43-7 |
Smiles | N1=C(N)N2C=3C=CC=CC3CC=4C=CC=CC4C2C1 |
颜色 | White |
物理性状 | Solid |
存储 | keep away from direct sunlight,store under nitrogen | store at 4°C | Shipping with blue ice/Shipping at ambient temperature. |
溶解度信息 | DMSO: ≥ 40 mg/mL, Sonication is recommended. H2O: < 1 mg/mL (insoluble) |
评论内容