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抗生素库

抗生素库

产品编号 L4400 Antibiotics Library
  库化合物信息   Excel SDF

抗生素是对抗感染的强效药物,挽救了大量患者生命,抗生素的发现和使用使人类寿命至少延长了10年,因而被称为“20世纪伟大的医学发现”,然而由于抗生素滥用严重,耐药性的发展速度惊人。抗生素耐药性严重威胁公共健康、经济增长和全球经济稳定,因此在阻止抗生素滥用的同时,迫切需要推动研发新的和改造现有的抗生素。 TargetMol 抗生素库是有 708 个具有抗菌生物活性的化合物的集合,可用于抗生素类药物的筛选和其他相关医药研究。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 708个具有抗菌活性化合物的独特集合,是医药研究的优良工具库和药物筛选的有效载体;
  • 大部分产品属于上市药物,部分化合物已经得到FDA批准,是颇具研究潜力的抗生素活性化合物集合;
  • 生物活性和生物安全性已通过临床前研究和临床实验得到保障;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • 结构多样,药效显著,可渗透细胞;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L4400)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Antibacterial (544)
Antibiotic (521)
Antifungal (121)
Parasite (68)
Autophagy (67)
Topoisomerase (39)
ribosome (33)
Apoptosis (32)
DNA/RNA Synthesis (31)
Endogenous Metabolite (30)
Antifection (16)
DNA gyrase (13)
Influenza Virus (13)
HIV Protease (11)
Anti-infection (10)
Reactive Oxygen Species (9)
Mitophagy (9)
HSV (9)
Dehydrogenase (8)
P450 (8)
Phosphatase (8)
CAT (7)
ATPase (6)
COX (6)
NF-κB (6)
DHFR (5)
MMP (5)
Cell wall (5)
Nucleoside Antimetabolite/Analog (5)
PKC (5)
mTOR (4)
HIF/HIF Prolyl-Hydroxylase (4)
Microtubule Associated (4)
MAO (4)
STAT (4)
Glucosidase (3)
Glucocorticoid Receptor (3)
Ferroptosis (3)
Tyrosine Kinases (3)
Potassium Channel (3)
NADPH (3)
Estrogen/progestogen Receptor (3)
TLR (3)
SARS-CoV (3)
Virus Protease (3)
HSP (3)
Antiviral (3)
AChR (3)
Antioxidant (3)
Aminopeptidase (3)
ABC (2)
Lipoxygenase (2)
DNA Alkylation (2)
IL Receptor (2)
ROS (2)
Proton pump (2)
PPAR (2)
Proteasome (2)
DNA Alkylator/Crosslinker (2)
Complement System (2)
Antifolate (2)
MRP (2)
PI3K (2)
AChE (2)
p38 MAPK (2)
Sodium Channel (2)
TGF-beta/Smad (2)
DprE1 (2)
GABA Receptor (2)
Dopamine Receptor (2)
Glutathione Peroxidase (2)
Adrenergic Receptor (2)
TNF (2)
Hedgehog/Smoothened (2)
AhR (1)
Aryl Hydrocarbon Receptor (1)
UGT (1)
PD-1/PD-L1 (1)
Tyrosinase (1)
Phospholipase (1)
TRP/TRPV Channel (1)
PKA (1)
Src (1)
transporter (1)
PLK (1)
ATM/ATR (1)
Annexin A (1)
Adenosine deaminase (1)
Serine/threonin kinase (1)
Sirtuin (1)
Akt (1)
PTEN (1)
Pyroptosis (1)
Ras (1)
AMPK (1)
RSV (1)
Epigenetic Reader Domain (1)
ATTECs (1)
HBV (1)
iGluR (1)
Hydroxylase (1)
Hydrogenase (1)
HMG-CoA Reductase (1)
Histone Acetyltransferase (1)
DNA Methyltransferase (1)
HCV Protease (1)
Glutathione reductase (1)
Integrin (1)
DNA-PK (1)
GluCls (1)
Free radical scavengers (1)
Fatty Acid Synthase (1)
FAK (1)
FAAH (1)
Endothelin Receptor (1)
DNA (1)
Interleukin (1)
Nrf2 (1)
Carbonic Anhydrase (1)
NOS (1)
NOD-like Receptor (NLR) (1)
NOD (1)
Bombesin Receptor (1)
Estrogen Receptor/ERR (1)
NADPH-oxidase (1)
Calcium Channel (1)
c-Met/HGFR (1)
IRE1 (1)
CRISPR/Cas9 (1)
CRM1 (1)
LTR (1)
Liver X Receptor (1)
Lipid (1)
JNK (1)
IκB/IKK (1)
Neurokinin receptor (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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