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抗癌上市药物库

抗癌上市药物库

产品编号 L2110 Anti-Cancer Approved Drug Library
  库化合物信息   Excel SDF

尽管在过去的几十年中癌症的研究和治疗取得了巨大的成功,但癌症仍然是人类面临的巨大挑战,给患者身心健康带来巨大的痛苦。癌细胞具有许多显著不同的生物学特征,表现出无限的增殖潜能,维持自身生长信号的持续稳定,逃避应激信号诱导的细胞凋亡,刺激血管生长,为肿瘤提供营养,同时逃避免疫系统防御和诱导局部慢性炎症,发挥其侵袭和转移能力,表现出异常的代谢活动,并通过突变和表观遗传机制显著改变全基因组的稳定性。

根据文献报道和有关公开资料,我们挑选了1825 个具有抗癌活性或潜在抗癌活性的上市药物组成抗癌上市药物库,可用于具体癌症的阳性对照及不同癌症之间相关性研究。如果您对癌症相关适应症感兴趣,还可以关注我们其他三个库:抗癌分子库,癌细胞分化分子库,以及抗癌临床药物库。希望我们在抗癌研究的路上,助您一臂之力!

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 1825个具有抗癌活性小分子的独特集合,所有化合物都经过了严格的临床前研究和临床试验,由FDA、EMA或NMPA批准上市,可用于高通量、高内涵筛选。
  • 所有化合物都具有已知且良好的生物活性、安全性和生物利用度,这些特性可显着加速药物开发和优化,是进行癌症相关研究和药物重定位有效的筛选工具。
  • 作用靶点涉及PI3K、HDAC、mTOR、CDK、JAK 等癌症相关靶点,涉及的研究领域包括肺癌、乳腺癌、白血病、淋巴瘤等15种癌症;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2110)
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客户使用化合物库发表的文献

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化合物库组成

Autophagy (337)
Apoptosis (249)
Adrenergic Receptor (159)
5-HT Receptor (158)
Endogenous Metabolite (152)
Antibacterial (137)
COX (120)
Antibiotic (114)
Dopamine Receptor (108)
Histamine Receptor (104)
DNA/RNA Synthesis (80)
Sodium Channel (78)
Calcium Channel (75)
Potassium Channel (72)
AChR (67)
Parasite (53)
Glucocorticoid Receptor (52)
P450 (44)
HIV Protease (42)
Reactive Oxygen Species (38)
Ferroptosis (37)
Antifungal (36)
NF-κB (36)
EGFR (34)
Estrogen/progestogen Receptor (33)
GABA Receptor (33)
c-Kit (32)
VEGFR (32)
Mitophagy (31)
Topoisomerase (30)
PDGFR (29)
Nucleoside Antimetabolite/Analog (29)
PPAR (29)
SARS-CoV (28)
Influenza Virus (27)
Estrogen Receptor/ERR (27)
Dehydrogenase (27)
Prostaglandin Receptor (26)
PDE (25)
Serotonin Transporter (23)
Microtubule Associated (23)
Proton pump (22)
ATPase (20)
DNA Alkylator/Crosslinker (20)
Norepinephrine (20)
iGluR (19)
Androgen Receptor (19)
FLT (18)
HDAC (18)
JAK (17)
RAAS (17)
FGFR (17)
HSV (17)
Bcr-Abl (16)
Opioid Receptor (15)
c-Met/HGFR (15)
Virus Protease (15)
Adenosine Receptor (15)
Src (15)
TRP/TRPV Channel (14)
HBV (14)
Tyrosine Kinases (14)
Antifolate (13)
TNF (13)
Progesterone Receptor (13)
PKC (12)
CDK (12)
GNRH Receptor (12)
ROS (12)
Retinoid Receptor (12)
Raf (12)
SGLT (11)
ALK (11)
MAO (11)
DHFR (11)
NMDAR (11)
MRP (11)
P-gp (11)
Carbonic Anhydrase (10)
HMG-CoA Reductase (10)
Reverse Transcriptase (10)
AChE (10)
Proteasome (10)
Drug Metabolite (10)
PARP (10)
Antifection (9)
CaMK (9)
Phosphatase (9)
c-RET (9)
AMPK (9)
HCV Protease (9)
Lipoxygenase (8)
DNA Alkylation (8)
MMP (8)
mTOR (8)
PI3K (8)
BTK (8)
P2Y Receptor (8)
Monoamine Oxidase (8)
GluR (8)
HIF/HIF Prolyl-Hydroxylase (8)
Guanylate cyclase (7)
Monoamine Transporter (7)
Phospholipase (7)
TAM Receptor (7)
Trk receptor (7)
ABC (7)
Chloride channel (7)
HER (7)
STAT (7)
CFTR (7)
Thrombin (7)
GPR (7)
NADPH (7)
MEK (7)
Neurokinin receptor (7)
BCL (6)
DNA (6)
DNA Methyltransferase (6)
Interleukin (6)
Aromatase (6)
ribosome (6)
IL Receptor (6)
Vasopressin Receptor (6)
S1P Receptor (6)
Hedgehog/Smoothened (6)
P2X Receptor (6)
Mitochondrial Metabolism (6)
Transferase (6)
ERK (6)
LPL Receptor (5)
PKA (5)
Wnt/beta-catenin (5)
Nrf2 (5)
TLR (5)
ROCK (5)
Histone Methyltransferase (5)
Endothelin Receptor (5)
Caspase (5)
Ras (5)
FXR (5)
Akt (5)
CaSR (5)
ROS Kinase (5)
Glutathione Peroxidase (5)
HIF (5)
PGE Synthase (4)
HSP (4)
Fatty Acid Synthase (4)
NO Synthase (4)
Tyrosinase (4)
DPP-4 (4)
Annexin A (4)
GPCR19 (4)
NOD (4)
Leukotriene Receptor (4)
Oxytocin Receptor (4)
p38 MAPK (4)
IκB/IKK (4)
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Beta Amyloid (4)
Melatonin Receptor (4)
Smo (4)
GSK-3 (4)
Amino Acids and Derivatives (4)
Sigma receptor (4)
LTR (3)
Adenosine deaminase (3)
Serine/threonin kinase (3)
Syk (3)
Serine Protease (3)
Aminopeptidase (3)
Ligand for E3 Ligase (3)
Integrin (3)
Hydroxylase (3)
Melanocortin Receptor (3)
Cysteine Protease (3)
GST (3)
c-Fms (3)
Free radical scavengers (3)
Molecular Glues (3)
cholecystokinin (3)
IGF-1R (3)
AhR (3)
Isocitrate Dehydrogenase (IDH) (3)
Gamma-secretase (3)
Na-K-Cl cotransporter (3)
TGF-beta/Smad (3)
Xanthine Oxidase (3)
UGT (3)
FAK (3)
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MT Receptor (3)
CXCR (3)
MAPK (2)
LDL (2)
TOPK (2)
Gap Junction Protein (2)
Arginase (2)
Ligands for Target Protein for PROTAC (2)
NOS (2)
Cell wall (2)
GHSR (2)
Reductase (2)
IFNAR (2)
DNA gyrase (2)
PLK (2)
Cannabinoid Receptor (2)
CGRP Receptor (2)
CCR (2)
NOD-like Receptor (NLR) (2)
CAT (2)
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Beta-Secretase (2)
OAT (2)
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ROR (2)
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IRE1 (2)
Protease-activated Receptor (2)
YAP (2)
Ephrin Receptor (2)
Decarboxylase (2)
Aurora Kinase (2)
Somatostatin (2)
CRM1 (2)
Hexokinase (2)
RSV (2)
Glutathione reductase (2)
PD-1/PD-L1 (1)
Hydrogenase (1)
NPC1L1 (1)
NADPH-oxidase (1)
Platelet aggregation (1)
Complement System (1)
p53 (1)
Mdm2 (1)
Imidazoline Receptor (1)
S6 Kinase (1)
GluCls (1)
BACE (1)
PAFR (1)
Epigenetic Reader Domain (1)
Adiponectin receptor (1)
Thrombopoietin Receptor (1)
cAMP (1)
ACK (1)
PAD (1)
Chk (1)
Immunology/Inflammation related (1)
OX Receptor (1)
Bradykinin Receptor (1)
MTH1 (1)
FAAH (1)
GRK (1)
Glucagon Receptor (1)
PROTAC Linker (1)
CSF-1R (1)
DUB (1)
Na+/Ca2+ Exchanger (1)
Factor Xa (1)
RAR/RXR  (1)
Histone Demethylase (1)
PDK (1)
Lipase (1)
JNK (1)
VDA (1)
Neprilysin (1)
IAP (1)
Pyroptosis (1)
Histone Acetyltransferase (1)
Sirtuin (1)
Hck (1)
Liver X Receptor (1)
ATP Citrate Lyase (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Thyroid hormone receptor(THR) (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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