• TargetMol
    您的购物车当前为空
TargetMol | Compound Library

抗癌上市药物库现货

Anti-Cancer Approved Drug Library

Rating icon 很棒
产品编号 L2110

尽管在过去的几十年中癌症的研究和治疗取得了巨大的成功,但癌症仍然是人类面临的巨大挑战,给患者身心健康带来巨大的痛苦。癌细胞具有许多显著不同的生物学特征,表现出无限的增殖潜能,维持自身生长信号的持续稳定,逃避应激信号诱导的细胞凋亡,刺激血管生长,为肿瘤提供营养,同时逃避免疫系统防御和诱导局部慢性炎症,发挥其侵袭和转移能力,表现出异常的代谢活动,并通过突变和表观遗传机制显著改变全基因组的稳定性。

根据文献报道和有关公开资料,我们挑选了1800 个具有抗癌活性或潜在抗癌活性的上市药物组成抗癌上市药物库,可用于具体癌症的阳性对照及不同癌症之间相关性研究。如果您对癌症相关适应症感兴趣,还可以关注我们其他三个库:抗癌分子库,癌细胞分化分子库,以及抗癌临床药物库。希望我们在抗癌研究的路上,助您一臂之力!

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
资源下载
化合物库相关信息
Excel
SDF
联系我们获取更多批次信息

产品编号 L2110

抗癌上市药物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 1800个具有抗癌活性小分子的独特集合,所有化合物都经过了严格的临床前研究和临床试验,由FDA、EMA或NMPA批准上市,可用于高通量、高内涵筛选。
  • 所有化合物都具有已知且良好的生物活性、安全性和生物利用度,这些特性可显着加速药物开发和优化,是进行癌症相关研究和药物重定位有效的筛选工具。
  • 作用靶点涉及PI3K、HDAC、mTOR、CDK、JAK 等癌症相关靶点,涉及的研究领域包括肺癌、乳腺癌、白血病、淋巴瘤等癌症;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

使用TargetMol产品
发表顶级期刊文献

引用更多关于TargetMol产品的科学文献吧!

查看更多

Library Customization | TargetMol 化合物库定制

Compound Library | TargetMol
您可以通过点击按钮
定制您专属的化合物!
联系专属定制

Library Customization | TargetMol 化合物库组成

Autophagy
Apoptosis
Endogenous Metabolite
Antibacterial
Adrenergic Receptor
5-HT Receptor
Antibiotic
COX
Dopamine Receptor
Histamine Receptor
Potassium Channel
Sodium Channel
Parasite
DNA/RNA Synthesis
Calcium Channel
AChR
Cytochromes P450
NF-κB
Glucocorticoid Receptor
Reactive Oxygen Species
HIV Protease
EGFR
Antifungal
VEGFR
Estrogen/progestogen Receptor
Ferroptosis
Virus Protease
SARS-CoV
Mitophagy
GABA Receptor
Topoisomerase
c-Kit
PPAR
Estrogen Receptor/ERR
Nucleoside Antimetabolite/Analog
PDGFR
Dehydrogenase
Serotonin Transporter
Influenza Virus
Microtubule Associated
Prostaglandin Receptor
PDE
iGluR
JAK
ATPase
FGFR
TNF
HSV
HDAC
Norepinephrine
Proton pump
Interleukin
c-Met/HGFR
RAAS
Bcr-Abl
Androgen Receptor
Src
DNA Alkylator/Crosslinker
HBV
FLT
TRP/TRPV Channel
Adenosine Receptor
Tyrosine Kinases
Drug Metabolite
Opioid Receptor
Progesterone Receptor
MMP
Akt
Bcl-2 Family
CDK
AMPK
p38 MAPK
PI3K
PARP
PKC
Raf
ROS
Cholinesterase (ChE)
ALK
STAT
GNRH Receptor
Caspase
MAO
NMDAR
mTOR
SGLT
P-gp
Retinoid Receptor
HMG-CoA Reductase
HIF/HIF Prolyl-Hydroxylase
Carbonic Anhydrase
DHFR
HCV Protease
MRP
Antifolate
ERK
Reverse Transcriptase
c-RET
Ras
Proteasome
Phosphatase
DNA Alkylation
Lipoxygenase
CaMK
HSP
MEK
ROS Kinase
Monoamine Oxidase
ADC Cytotoxin
P2Y Receptor
ABC Transporter
Mitochondrial Metabolism
Antifection
Angiotensin-converting Enzyme (ACE)
Nrf2
Phospholipase
Anti-infection
NADPH
PKA
FXR
Guanylate cyclase
IL Receptor
GluR
TLR
Trk receptor
Beta Amyloid
DNA Methyltransferase
Thrombin
CFTR
HER
NO Synthase
S1P Receptor
Chloride channel
Transferase
Histone Methyltransferase
LPL Receptor
Glutathione Peroxidase
Wnt/beta-catenin
ROCK
P2X Receptor
Monoamine Transporter
Isocitrate Dehydrogenase (IDH)
Hedgehog/Smoothened
Endothelin Receptor
IκB/IKK
Kras
Aromatase
Neurokinin receptor
TAM Receptor
GPCR
JNK
Leukotriene Receptor
Gamma-secretase
Vasopressin Receptor
DNA
GPCR19
ribosome
HIF
Sigma receptor
Amino Acids and Derivatives
Antioxidant
GSK-3
Melatonin Receptor
CaSR
Serine Protease
Serine/threonin kinase
Annexin A
Molecular Glues
Smo
DPP-4
Fatty Acid Synthase
Xanthine Oxidase
IGF-1R
PGE Synthase
MAPK
Antiviral
Aminopeptidase
FKBP
Ligand for E3 Ligase
MDM-2/p53
NOD
Tyrosinase
MicroRNA
Integrin
Reductase
Cysteine Protease
UGT
MT Receptor
Na-K-Cl cotransporter
Glucosidase
PAK
Thrombopoietin Receptor
TGF-beta/Smad
Free radical scavengers
Decarboxylase
GST
c-Fms
Oxytocin Receptor
Hydroxylase
Adenosine Deaminase
Cuproptosis
Syk
FAK
AhR
NOD-like Receptor (NLR)
BTK
IKZF
NOS
Monocarboxylate transporter
ROR
CRM1
Ligands for Target Protein for PROTAC
YAP
Arginase
LTR
IFNAR
Cell wall
Tie-2
Cholecystokinin Receptor
Photosensitizer
Rho
Aryl Hydrocarbon Receptor
IRE1
LDL
DNA gyrase
Hexokinase
FAAH
CCR
CXCR
Aurora Kinase
Telomerase
ATP Citrate Lyase
Beta-Secretase
OAT
Sirtuin
Ephrin Receptor
RSV
Melanocortin Receptor
GHSR
PLK
CGRP Receptor
Cannabinoid Receptor
Complement System
Gap Junction Protein
Protease-activated Receptor
PD-1/PD-L1
Mdm2
NPC1L1
Hydrogenase
DNA-PK
BACE
Na+/Ca2+ Exchanger
Histone Demethylase
Lipase
Necroptosis
gp120/CD4
MIF
TOPK
Factor Xa
VDA
OCT
c-Myc
Hck
Liver X Receptor
NR4A
IDO
IAP
CSF-1R
Immunology/Inflammation related
Adiponectin Receptor
PAFR
MTH1
GRK
Glucagon Receptor
Arp2/3 Complex
PROTAC Linker
HCN Channel
ACK1
Bradykinin Receptor
HCAR
PTEN
Chk
Somatostatin
PAD
cAMP
Epigenetic Reader Domain
DUB
Indoleamine 2,3-Dioxygenase (IDO)
Lipid
Glutathione reductase
STING
GluCls
Pyroptosis
Casein Kinase
Neprilysin
PDK
Platelet aggregation
NADPH-oxidase
S6 Kinase
Imidazoline Receptor
p53
PGC-1α

Keywords