购物车
  • 全部删除
  • TargetMol
    您的购物车当前为空
TargetMol | Compound Library

抗癌化合物库现货

Anti-Cancer Compound Library

Rating icon 很棒
产品编号 L2100

在过去的几十年中癌症的研究和治疗取得了巨大的成功,但癌症仍然是人类面临的巨大挑战,给患者身心健康带来巨大的痛苦。癌细胞具有许多显著不同的生物学特征,表现出无限的增殖潜能,维持自身生长信号的持续稳定,逃避应激信号(例如治疗药物)诱导的细胞凋亡,刺激血管生长,为肿瘤提供营养,同时逃避免疫系统防御和诱导局部慢性炎症,发挥其侵袭和转移能力,表现出异常的代谢活动,并通过突变和表观遗传机制显著改变全基因组的稳定性。 我们根据上述癌细胞显著不同的特征和异常的代谢活动,精心筛选了 9332 个肿瘤相关的小分子化合物,这些化合物都是调节肿瘤细胞代谢、增殖、侵袭、转移通路上的小分子,可用于肿瘤相关的研究以及抗肿瘤药物的筛选,可用于高通量、高内涵筛选。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
资源下载
化合物库相关信息
Excel
SDF
联系我们获取更多批次信息

产品编号 L2100

抗癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 9332种肿瘤相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 产品经过临床验证和临床实验,具有生物安全保障和一定的生物活性;
  • 是肿瘤发生机理研究、抗肿瘤药物筛选的有效工具;?
  • 靶点含PI3K、HDAC、mTOR、CDK、Aurora Kinase、JAK等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS检测技术保证产品高纯度和高质量,减少假阳性发生概率。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

使用TargetMol产品
发表顶级期刊文献

引用更多关于TargetMol产品的科学文献吧!

查看更多

Library Customization | TargetMol 化合物库定制

Compound Library | TargetMol
您可以通过点击按钮
定制您专属的化合物!
联系专属定制

Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
Antibacterial
NF-κB
DNA/RNA Synthesis
COX
Adrenergic Receptor
CDK
Dopamine Receptor
PI3K
EGFR
Potassium Channel
Reactive Oxygen Species
Epigenetic Reader Domain
Histamine Receptor
Calcium Channel
Antibiotic
Cytochromes P450
VEGFR
Sodium Channel
Histone Methyltransferase
HDAC
GABA Receptor
Parasite
TRP/TRPV Channel
JAK
PPAR
mTOR
Akt
ERK
Wnt/beta-catenin
AChR
HIV Protease
GPCR
Antifungal
PARP
Prostaglandin Receptor
Estrogen Receptor/ERR
PKC
Src
FLT
p38 MAPK
STAT
Microtubule Associated
Adenosine Receptor
AMPK
PDGFR
FGFR
GSK-3
Dehydrogenase
Topoisomerase
TNF
Estrogen/progestogen Receptor
Opioid Receptor
Bcl-2 Family
Caspase
Raf
Glucocorticoid Receptor
Influenza Virus
Antioxidant
iGluR
c-Met/HGFR
Androgen Receptor
Ferroptosis
Nucleoside Antimetabolite/Analog
c-Kit
HSP
Sirtuin
Bcr-Abl
MMP
ALK
Cannabinoid Receptor
ATPase
Histone Demethylase
TGF-beta/Smad
Aurora Kinase
Ras
Phosphatase
IL Receptor
JNK
ROCK
PDE
Tyrosine Kinases
DUB
MAPK
MEK
P-gp
NO Synthase
ROS
p53
IκB/IKK
Mitophagy
NMDAR
SARS-CoV
Virus Protease
RIP kinase
Lipoxygenase
Serine/threonin kinase
S1P Receptor
HIF/HIF Prolyl-Hydroxylase
PKA
HSV
CXCR
NOD
IGF-1R
DNA-PK
Hedgehog/Smoothened
Antiviral
Nrf2
LPL Receptor
TLR
Histone Acetyltransferase
c-RET
E1/E2/E3 Enzyme
Drug Metabolite
P2X Receptor
S6 Kinase
FAK
ATM/ATR
Cholinesterase (ChE)
Casein Kinase
HIF
HER
PERK
PLK
Chloride channel
Mitochondrial Metabolism
Sigma receptor
TAM Receptor
Proteasome
NOS
Chk
GluR
Interleukin
Neurokinin receptor
DNA Methyltransferase
Proton pump
RAAS
HBV
Pim
Serotonin Transporter
Norepinephrine
HCV Protease
Gamma-secretase
Trk receptor
Beta Amyloid
Phospholipase
Tyrosinase
DNA Alkylator/Crosslinker
Rho
Protease-activated Receptor
Mdm2
DHFR
MAO
Endothelin Receptor
Carbonic Anhydrase
Glucagon Receptor
PDK
IRAK
PROTACs
DYRK
Antifection
SGLT
Retinoid Receptor
Syk
P2Y Receptor
Fatty Acid Synthase
PD-1/PD-L1
Smo
Neuropeptide Y Receptor
c-Myc
Guanylate cyclase
cAMP
CaMK
transporter
Reverse Transcriptase
c-Fms
Kras
Transferase
DNA
LPA Receptor
Anti-infection
CFTR
Integrin
IRE1
DNA Alkylation
OX Receptor
ADC Cytotoxin
NADPH
Cholecystokinin Receptor
Leukotriene Receptor
HMG-CoA Reductase
ROS Kinase
Monoamine Oxidase
YAP
Progesterone Receptor
Serine Protease
Antifolate
IAP
ABC Transporter
Vasopressin Receptor
PI4K
Kinesin
GTPase
MRP
Indoleamine 2,3-Dioxygenase (IDO)
NOD-like Receptor (NLR)
MicroRNA
BTK
GHSR
Monocarboxylate transporter
Reductase
CSF-1R
GPCR19
Aromatase
Neurotensin Receptor
Immunology/Inflammation related
GRK
CCR
Bradykinin Receptor
Somatostatin
Ligand for E3 Ligase
Glutathione Peroxidase
Melatonin Receptor
Aryl Hydrocarbon Receptor
Telomerase
AhR
FXR
LIM Kinase
Myosin
Glucosidase
Monoamine Transporter
PAD
BCRP
MNK
STING
Free radical scavengers
Ephrin Receptor
Melanocortin Receptor
LTR
Na+/Ca2+ Exchanger
IFNAR
CaSR
GNRH Receptor
SIK
Bombesin Receptor
PAK
PTEN
Wee1
PGE Synthase
Thrombin
Arrestin
BACE
Tie-2
OCT
Cysteine Protease
Liver X Receptor
Glucokinase
Glutaminase
UGT
LDL
Molecular Glues
Isocitrate Dehydrogenase (IDH)
Acyltransferase
Methionine Adenosyltransferase (MAT)
GPX
Hydroxylase
APC/C
MLK
Melanin-concentrating Hormone Receptor (MCHR)
CRM1
Amino Acids and Derivatives
Ligands for Target Protein for PROTAC
NAMPT
PYK2
Annexin A
PAFR
MT Receptor
Lipid
OAT
Survivin
LRRK2
CRFR
MELK
RSV
ribosome
SGK
Apelin receptor
NPC1L1
TOPK
Cell Cycle Arrest
MTH1
DPP-4
FAAH
ACK1
Xanthine Oxidase
Beta-Secretase
Porcupine
ASK
GST
Carboxypeptidase
CRISPR/Cas9
Oxytocin Receptor
CGRP Receptor
Discoidin Domain Receptor (DDR)
Platelet aggregation
BMI-1
PKM
RAR/RXR
MALT
ROR
Hck
RANKL/RANK
IDO
Adiponectin Receptor
DNA gyrase
Hexokinase
ATP Citrate Lyase
Aminopeptidase
Decarboxylase
TSH Receptor
PAI-1
Pyroptosis
Hippo pathway
Aquaporin
Adenosine Deaminase
p97
Factor Xa
AAK1
VDAC
Haspin Kinase
Na-K-Cl cotransporter
HCN Channel
Epoxide Hydrolase
KSP
CD73
HuR
KLF
Complement System
Imidazoline Receptor
Adenylyl Cyclase
EBI2/GPR183
NEDD8
MyD88
Arginase
Cell wall
Lipase
gp120/CD4
VDA
Galectin
Thrombopoietin Receptor
OXPHOS
PSMA
Glutathione reductase
AIM2
GluCls
Protease
RXFP receptor
Gap Junction Protein
DAPK
NADPH-oxidase
Lysosomal Autophagy
Vitamin
IKZF
FOXO3
Advanced Glycation End Products
Transaminase
Hydrogenase
CD38
CYP19A1
Piezo Channel
NUDIX hydrolase
Dynamin
Neuropeptide W
Necroptosis
N-Acetylglucosaminyltransferase
Stemness kinase
Amylase
FLAP
Endonuclease
Phosphorylase
GlyT
Anion Exchanger
PROTAC Linker
Thioredoxin
Stearoyl-CoA Desaturase (SCD)
Angiotensin-converting Enzyme (ACE)
Transketolase
Huntingtin
cGAS
hCE
NEDD4-1
Neprilysin
Glyoxalase
Sodium-dependent phosphate transporter

Keywords