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TargetMol | Compound Library

铜死亡化合物库现货

Cuproptosis Compound Library

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产品编号 L8710

铜离子是所有生物必不可少的辅助因子,但当其浓度超过一定阈值时,就会对机体产生毒害作用。铜死亡的发生机制明显区别于已知的细胞凋亡、焦亡、坏死及铁死亡的细胞死亡方式:铜离子通过直接结合三羧酸(TCA)循环途径中的脂酰化成分,导致脂酰化蛋白异常聚集以及铁硫簇蛋白的丢失,从而导致蛋白质毒性应激反应并导致细胞死亡。铜死亡与肌萎缩侧索硬化症(ALS)、乳腺癌、黑色素瘤、成神经细胞瘤、和前列腺癌等疾病有关。 TargetMol 铜死亡化合物库集合了 400 种与铜死亡相关的化合物,可以用于铜死亡机制及相关疾病研究

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产品编号 L8710

铜死亡化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 400 种与铜死亡相关的活性小分子,可用于高通量和高内涵筛选;
  • 靶向FDX1,胞浆金属伴侣(ATOX1),CCS (copper chaperones),线粒体呼吸等;
  • 部分化合物已被FDA批准上市;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库定制

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Library Customization | TargetMol 化合物库组成

Reactive Oxygen Species
Autophagy
Apoptosis
BCL
Endogenous Metabolite
Mitophagy
ROS
Mitochondrial Metabolism
Antibacterial
COX
NF-κB
Ferroptosis
HIV Protease
Antioxidant
PDE
Antifungal
Caspase
IAP
Antibiotic
Parasite
HSP
Influenza Virus
Dehydrogenase
Topoisomerase
IL Receptor
ROS Kinase
PKM
Calcium Channel
HIF/HIF Prolyl-Hydroxylase
NO Synthase
ATPase
p38 MAPK
Estrogen/progestogen Receptor
PARP
ALK
HDAC
P450
TNF
PI3K
PPAR
MMP
Xanthine Oxidase
Akt
Nrf2
AMPK
GABA Receptor
p53
NOS
c-Met/HGFR
NADPH
Virus Protease
PKC
E1/E2/E3 Enzyme
DNA/RNA Synthesis
Histamine Receptor
JNK
Wnt/beta-catenin
VEGFR
ERK
Gamma-secretase
JAK
HSV
Lipoxygenase
mTOR
P-gp
Trk receptor
IκB/IKK
5-HT Receptor
Potassium Channel
FLT
Sodium Channel
Microtubule Associated
Chloride channel
Monocarboxylate transporter
ROR
HCV Protease
Dynamin
RAAS
HBV
Estrogen Receptor/ERR
Tyrosine Kinases
Cysteine Protease
Adrenergic Receptor
MAO
IRE1
Opioid Receptor
PDGFR
Epigenetic Reader Domain
IGF-1R
Interleukin
OXPHOS
TLR
SARS-CoV
Beta Amyloid
Reverse Transcriptase
STAT
PDK
Phospholipase
AChR
c-Kit
Anti-infection
HMG-CoA Reductase
CFTR
Proteasome
Mdm2
CAT
Carbonic Anhydrase
Src
MyD88
Ligands for Target Protein for PROTAC
YAP
Adenosine Receptor
IFNAR
aconitase
RAR/RXR 
Histone Demethylase
Glutathione Peroxidase
Phosphatase
Melatonin Receptor
PKA
FXR
TRP/TRPV Channel
Amylase
Glucocorticoid Receptor
Immunology/Inflammation related
Annexin A
UGT
CDK
Drug Metabolite
Phosphorylase
NMDAR
Hexokinase
Hedgehog/Smoothened
FAAH
Somatostatin
GluR
cAMP
CaMK
DNA
Androgen Receptor
TGF-beta/Smad
SGLT
Glutathione reductase
AChE
Antiviral
Prostaglandin Receptor
STING
LRRK2
Aminopeptidase
Free radical scavengers
Sirtuin
Histone Acetyltransferase
RSV
Casein Kinase
ATM/ATR
GST
Retinoid Receptor
Aromatase
CRISPR/Cas9
GPR
HIF
MEK
FGFR
Discoidin Domain Receptor (DDR)
Platelet aggregation
Syk
NOD
NADPH-oxidase
IRAK
S6 Kinase
Tyrosinase
Thrombin
NOD-like Receptor (NLR)
AhR
Monoamine Oxidase

Supporting Files | TargetMol 化合物库信息

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IACS-010759MIM1EnsifentrineLuteolinPKR-IN-2Sulcotrione3-MethyladenineSalsalateGSK5182Methyl gallate
Empty624-49-71092351-67-12365172-82-1607-91-079595-97-4510-30-5149647-78-9144060-53-756396-35-1551-15-5Empty
Dimethyl fumarateTorkinibDesmorpholinyl Navitoclax-NH-MeMyristicinnorbergeninEchinocystic acidVorinostatFebuxostatUK-5099Liquiritin
Empty32619-42-4139-85-57336-33-6301356-95-610236-47-2517-89-51333327-56-277671-31-9478-43-32143096-93-7Empty
OleuropeinProtocatechualdehyde3-demethylcolchicineCID5721353NaringinShikoninTRC051384 HClEnoximoneRheinNavitoclax-piperazine
Empty66170-10-35053-08-7335165-68-92086-83-1501-36-0478-01-3147526-32-71799633-27-4957-66-41617-53-4Empty
L-Ascorbic acid 2-phosphate trisodiumFenspiride hydrochlorideBAI1BerberineResveratrolNobiletinPitavastatin calciumS63845IsolinderalactoneAmentoflavone
Empty303-97-920633-67-428822-58-41800405-30-477883-43-3113-24-6480-44-4292057-76-2100823-03-836052-37-6Empty
Coenzyme Q9Calycosin-7-O-β-D-glucosideIBMXKL1333Doxazosin mesylateSodium 2-oxopropanoateAcacetinIMB-XH1TC11Alpinetin
Empty1208313-97-6923564-51-6546141-08-6877399-52-5118024-26-3569-83-51357576-48-7104206-82-83943-89-3370-86-5Empty
BD-AcAc 2NavitoclaxURB-597CrizotinibBlumeatin1-[2,4-Dihydroxy-6-methoxy-3-(3-methyl-2-buten-1-yl)phenyl]-3-(4-hydroxyphenyl)-2-propen-1-oneAZD4320MesotrioneEthyl 3,4-dihydroxybenzoateFCCP
Empty54-85-394164-88-28047-67-43943-74-61134156-31-2119168-77-376150-91-969-72-733237-37-510163-15-2Empty
IsoniazidPKM2-IN-1Iron sucroseMethyl VanillateVER-155008TebufenpyradTCPOBOPSalicylic acidRutaevinDisodium monofluorophosphate
Empty143390-89-02465-59-041753-43-91454846-35-513005-09-953846-50-730964-13-7917111-44-575747-14-71426138-42-2Empty
Kresoxim-MethylOxypurinolGinsenoside Rb1LorlatinibDehydrocorydaline nitrate8-​PrenylnaringeninCynarinLexibulinTanespimycinFX1