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Cuproptosis Compound Library
铜离子是所有生物必不可少的辅助因子,但当其浓度超过一定阈值时,就会对机体产生毒害作用。铜死亡的发生机制明显区别于已知的细胞凋亡、焦亡、坏死及铁死亡的细胞死亡方式:铜离子通过直接结合三羧酸(TCA)循环途径中的脂酰化成分,导致脂酰化蛋白异常聚集以及铁硫簇蛋白的丢失,从而导致蛋白质毒性应激反应并导致细胞死亡。铜死亡与肌萎缩侧索硬化症(ALS)、乳腺癌、黑色素瘤、成神经细胞瘤、和前列腺癌等疾病有关。 TargetMol 铜死亡化合物库集合了 400 种与铜死亡相关的化合物,可以用于铜死亡机制及相关疾病研究
Empty | 1570496-34-2 | 509102-00-5 | 1884461-72-6 | 491-70-3 | 1628428-01-2 | 99105-77-8 | 5142-23-4 | 552-94-3 | 877387-37-6 | 99-24-1 | Empty |
IACS-010759 | MIM1 | Ensifentrine | Luteolin | PKR-IN-2 | Sulcotrione | 3-Methyladenine | Salsalate | GSK5182 | Methyl gallate | ||
Empty | 624-49-7 | 1092351-67-1 | 2365172-82-1 | 607-91-0 | 79595-97-4 | 510-30-5 | 149647-78-9 | 144060-53-7 | 56396-35-1 | 551-15-5 | Empty |
Dimethyl fumarate | Torkinib | Desmorpholinyl Navitoclax-NH-Me | Myristicin | norbergenin | Echinocystic acid | Vorinostat | Febuxostat | UK-5099 | Liquiritin | ||
Empty | 32619-42-4 | 139-85-5 | 7336-33-6 | 301356-95-6 | 10236-47-2 | 517-89-5 | 1333327-56-2 | 77671-31-9 | 478-43-3 | 2143096-93-7 | Empty |
Oleuropein | Protocatechualdehyde | 3-demethylcolchicine | CID5721353 | Naringin | Shikonin | TRC051384 HCl | Enoximone | Rhein | Navitoclax-piperazine | ||
Empty | 66170-10-3 | 5053-08-7 | 335165-68-9 | 2086-83-1 | 501-36-0 | 478-01-3 | 147526-32-7 | 1799633-27-4 | 957-66-4 | 1617-53-4 | Empty |
L-Ascorbic acid 2-phosphate trisodium | Fenspiride hydrochloride | BAI1 | Berberine | Resveratrol | Nobiletin | Pitavastatin calcium | S63845 | Isolinderalactone | Amentoflavone | ||
Empty | 303-97-9 | 20633-67-4 | 28822-58-4 | 1800405-30-4 | 77883-43-3 | 113-24-6 | 480-44-4 | 292057-76-2 | 100823-03-8 | 36052-37-6 | Empty |
Coenzyme Q9 | Calycosin-7-O-β-D-glucoside | IBMX | KL1333 | Doxazosin mesylate | Sodium 2-oxopropanoate | Acacetin | IMB-XH1 | TC11 | Alpinetin | ||
Empty | 1208313-97-6 | 923564-51-6 | 546141-08-6 | 877399-52-5 | 118024-26-3 | 569-83-5 | 1357576-48-7 | 104206-82-8 | 3943-89-3 | 370-86-5 | Empty |
BD-AcAc 2 | Navitoclax | URB-597 | Crizotinib | Blumeatin | 1-[2,4-Dihydroxy-6-methoxy-3-(3-methyl-2-buten-1-yl)phenyl]-3-(4-hydroxyphenyl)-2-propen-1-one | AZD4320 | Mesotrione | Ethyl 3,4-dihydroxybenzoate | FCCP | ||
Empty | 54-85-3 | 94164-88-2 | 8047-67-4 | 3943-74-6 | 1134156-31-2 | 119168-77-3 | 76150-91-9 | 69-72-7 | 33237-37-5 | 10163-15-2 | Empty |
Isoniazid | PKM2-IN-1 | Iron sucrose | Methyl Vanillate | VER-155008 | Tebufenpyrad | TCPOBOP | Salicylic acid | Rutaevin | Disodium monofluorophosphate | ||
Empty | 143390-89-0 | 2465-59-0 | 41753-43-9 | 1454846-35-5 | 13005-09-9 | 53846-50-7 | 30964-13-7 | 917111-44-5 | 75747-14-7 | 1426138-42-2 | Empty |
Kresoxim-Methyl | Oxypurinol | Ginsenoside Rb1 | Lorlatinib | Dehydrocorydaline nitrate | 8-Prenylnaringenin | Cynarin | Lexibulin | Tanespimycin | FX1 |