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高选择性抑制剂库

高选择性抑制剂库

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产品编号 L2010 Highly Selective Inhibitor Library
  库化合物信息   Excel SDF

高选择性抑制剂能够高度选择性地影响目标分子或通路,而对其他非目标分子的影响相对较小。这种选择性是指药物在生物体内能够特异性地与目标分子相互作用,而对非目标分子产生较小或几乎没有影响。与非选择性抑制剂相比,高选择性抑制剂的优势在于其更精确地作用于目标靶点,从而降低了对非目标靶点的干扰,减少了可能的副作用和毒性。高选择性抑制剂在药物研发中的应用广泛,特别是在癌症治疗和其他复杂疾病的治疗方面,应用于药物开发中,可以更有效地干预病理过程,提高治疗的效果,并降低不良反应的发生率。

TargetMol 收集了580种高选择性抑制剂,绝大部分抑制剂相对于其他靶点的选择性至少高一百倍,是药物开发的有效工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品描述

  • xunm种具有高选择性的抑制剂集合;
  • 涵盖170种药物靶点;
  • 部分抑制剂已得到FDA批准上市;
  • 涵盖多种信号通路,如离子通道; NF-κB; PI3K/Akt/mTOR signaling; MAPK等
  • 结构多样,生物活性强,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

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包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2010)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Apoptosis (97)
Autophagy (63)
EGFR (33)
PI3K (25)
Epigenetic Reader Domain (20)
Histone Methyltransferase (20)
CDK (19)
BTK (18)
mTOR (15)
c-Met/HGFR (14)
GSK-3 (14)
Proteasome (14)
Aurora Kinase (13)
FGFR (13)
DPP-4 (12)
MEK (11)
Src (11)
HDAC (11)
Raf (11)
FLT (10)
PDGFR (10)
JAK (10)
Antibacterial (10)
VEGFR (9)
PARP (9)
Chk (8)
HIV Protease (8)
COX (8)
SGLT (8)
ERK (7)
TRP/TRPV Channel (7)
Cysteine Protease (7)
PLK (7)
Antibiotic (7)
PDE (7)
BCL (7)
PPAR (6)
ATM/ATR (6)
IκB/IKK (6)
SARS-CoV (6)
TGF-beta/Smad (6)
Histone Demethylase (6)
HER (6)
Trk receptor (6)
DNA/RNA Synthesis (6)
DNA-PK (6)
Ras (5)
PKC (5)
Ferroptosis (5)
Wnt/beta-catenin (5)
Virus Protease (5)
Serine Protease (5)
Phosphatase (5)
MMP (5)
P450 (5)
Mitophagy (5)
p38 MAPK (5)
Histone Acetyltransferase (5)
5-HT Receptor (5)
ALK (5)
c-Kit (5)
Dehydrogenase (5)
c-Fms (5)
Adrenergic Receptor (5)
Akt (4)
Lipase (4)
Sirtuin (4)
CSF-1R (4)
ROCK (4)
RIP kinase (4)
TAM Receptor (4)
MAO (4)
GPR (4)
Casein Kinase (4)
PDK (4)
Ligands for Target Protein for PROTAC (4)
FAAH (4)
PERK (4)
DUB (4)
AChR (4)
Potassium Channel (4)
Tyrosine Kinases (4)
PKA (4)
GluR (3)
Syk (3)
Influenza Virus (3)
Factor Xa (3)
STAT (3)
S1P Receptor (3)
Kinesin (3)
JNK (3)
Monoamine Oxidase (3)
MNK (3)
E1/E2/E3 Enzyme (3)
S6 Kinase (3)
Serine/threonin kinase (3)
iGluR (3)
IGF-1R (3)
Thrombin (3)
Caspase (3)
Prostaglandin Receptor (3)
HSP (3)
HCV Protease (3)
RAAS (3)
Pim (2)
Mitochondrial Metabolism (2)
cAMP (2)
Parasite (2)
Proton pump (2)
Phosphorylase (2)
Reactive Oxygen Species (2)
Cannabinoid Receptor (2)
NOS (2)
NOD-like Receptor (NLR) (2)
NADPH (2)
NOD (2)
Bcr-Abl (2)
Neurokinin receptor (2)
MAPK (2)
Endothelin Receptor (2)
Dopamine Receptor (2)
AMPK (2)
GRK (2)
transporter (2)
Glutathione Peroxidase (2)
Tie-2 (2)
CXCR (2)
HSV (2)
Hydroxylase (2)
IDO (2)
Adenosine Receptor (2)
Indoleamine 2,3-Dioxygenase (IDO) (2)
Integrase (2)
Sodium Channel (2)
DYRK (2)
Isocitrate Dehydrogenase (IDH) (2)
KSP (2)
CaMK (2)
Estrogen/progestogen Receptor (2)
LPL Receptor (2)
Estrogen Receptor/ERR (2)
LRRK2 (2)
Protease-activated Receptor (1)
Calcium Channel (1)
ACK (1)
Wee1 (1)
Progesterone Receptor (1)
Vasopressin Receptor (1)
Antifungal (1)
Telomerase (1)
Transferase (1)
BMI-1 (1)
Topoisomerase (1)
TLR (1)
PTEN (1)
BCRP (1)
SGK (1)
Reverse Transcriptase (1)
Rho (1)
ROS (1)
SIK (1)
Sigma receptor (1)
ATPase (1)
ASK (1)
Porcupine (1)
NMDAR (1)
Platelet aggregation (1)
HIF (1)
AChE (1)
IRE1 (1)
IRAK (1)
Interleukin (1)
Immunology/Inflammation related (1)
IFNAR (1)
DAPK (1)
Decarboxylase (1)
Histamine Receptor (1)
HIF/HIF Prolyl-Hydroxylase (1)
DNA (1)
LPA Receptor (1)
DNA Methyltransferase (1)
GlyT (1)
Glutaminase (1)
Glucocorticoid Receptor (1)
Galectin (1)
GABA Receptor (1)
Dynamin (1)
Fatty Acid Synthase (1)
FAK (1)
FABP (1)
Lipoxygenase (1)
MALT (1)
PKM (1)
NO Synthase (1)
Phospholipase (1)
Carbonic Anhydrase (1)
P-gp (1)
PD-1/PD-L1 (1)
CCR (1)
PAK (1)
CD73 (1)
OX Receptor (1)
cGAS (1)
Opioid Receptor (1)
Epoxide Hydrolase (1)
Mdm2 (1)
NF-κB (1)
Neuropeptide Y Receptor (1)
NAMPT (1)
Chloride channel (1)
MTH1 (1)
Monoamine Transporter (1)
MLK (1)
Complement System (1)
Microtubule Associated (1)
c-RET (1)
YAP (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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