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TargetMol | Compound Library

药物功能重定位化合物库现货

Drug Repurposing Compound Library

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产品编号 L9200

传统的药物开发涉及从头确认和验证新分子实体,这是一个耗时且成本高昂的过程,随着对药物安全性及有效性的要求不断提高,开发新药的成本还将持续上涨。由于时间和成本大幅降低,近年来药物功能重定位受到越来越多关注,高内涵筛选、新的生物标志物发现和生物信息学的快速发展为基于靶点或细胞的药物重定位创造了机会。 TargetMol 药物功能重定位化合物库收集了4960 种已上市和进入临床期的药物,这些化合物经过大量的临床前研究实验,具有活性高、毒性低和机制明确的特点,适用于药物筛选的同时,也是细胞诱导分化的有力工具。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L9200

药物功能重定位化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 4960种全球上市药物和临床药物的独特集合,可用于高通量筛选和高内涵筛选,是老药新用、新的药物靶点筛选和细胞诱导的有效工具。
  • 是整个行业规模领先的药物功能重定位化合物库;
  • 所有上市化合物得到FDA、EMA、NMPA等权威部门审批或收录在USP、EP、BP、JP、CP等药典文献中;
  • 涵盖多个研究领域:肿瘤、心血管药物、抗炎/免疫、神经系统药物、呼吸系统药物等;
  • 靶点多样,包括5-HT Receptor、Sodium Channel、p38 MAPK、PI3K、MEK等;
  • 详细的说明书,化合物结构、靶点信息、适应症信息、活性描述等;
  • 结构多样,药效显著,可渗透细胞;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

Autophagy
Antibacterial
Apoptosis
Antibiotic
Endogenous Metabolite
5-HT Receptor
Adrenergic Receptor
AChR
Dopamine Receptor
Histamine Receptor
COX
HIV Protease
Parasite
DNA/RNA Synthesis
Sodium Channel
Antifungal
Potassium Channel
Calcium Channel
VEGFR
EGFR
Topoisomerase
PDE
PI3K
Glucocorticoid Receptor
Reactive Oxygen Species
SARS-CoV
Cytochromes P450
Dehydrogenase
CDK
Estrogen/progestogen Receptor
HCV Protease
Influenza Virus
FLT
Ferroptosis
PPAR
NF-κB
GABA Receptor
PDGFR
Microtubule Associated
JAK
c-Kit
HDAC
FGFR
RAAS
c-Met/HGFR
Estrogen Receptor/ERR
mTOR
Prostaglandin Receptor
HBV
Mitophagy
Nucleoside Antimetabolite/Analog
Androgen Receptor
Src
Adenosine Receptor
Reverse Transcriptase
Tyrosine Kinases
iGluR
Serotonin Transporter
NMDAR
Bcr-Abl
Cholinesterase (ChE)
GPR
TRP/TRPV Channel
HSV
Norepinephrine
Proteasome
HER
Virus Protease
MAO
Raf
GluR
Antiviral
ATPase
PARP
ribosome
TNF
Phosphatase
Progesterone Receptor
Epigenetic Reader Domain
Akt
HSP
p38 MAPK
Antioxidant
ROS
Opioid Receptor
Beta Amyloid
Carbonic Anhydrase
Transferase
PKC
IL Receptor
Aurora Kinase
MMP
P-gp
ALK
HIF/HIF Prolyl-Hydroxylase
Proton pump
MEK
Histone Methyltransferase
Antifection
DPP-4
TLR
c-RET
Monoamine Oxidase
Thyroid hormone receptor(THR)
DNA Alkylator/Crosslinker
Drug Metabolite
Mitochondrial Metabolism
Endothelin Receptor
ERK
Interleukin
Thrombin
Trk receptor
Bcl-2 Family
AMPK
Phospholipase
HMG-CoA Reductase
GSK-3
P2X Receptor
CXCR
Retinoid Receptor
c-Fms
Integrin
MRP
GNRH Receptor
Caspase
ROCK
CCR
Lipoxygenase
SGLT
STAT
TAM Receptor
S1P Receptor
Factor Xa
PKA
Gamma-secretase
Vasopressin Receptor
Chk
Neurokinin receptor
FAK
NO Synthase
DNA-PK
NADPH
E1/E2/E3 Enzyme
Guanylate cyclase
DNA Alkylation
HIF
Cannabinoid Receptor
Syk
CFTR
p53
LPL Receptor
Reductase
Wnt/beta-catenin
Serine Protease
Antifolate
TGF-beta/Smad
Nrf2
DHFR
Amino Acids and Derivatives
P2Y Receptor
Glutathione Peroxidase
FXR
DNA gyrase
Hedgehog/Smoothened
IGF-1R
RSV
Sigma receptor
ROS Kinase
NOS
Histone Demethylase
CSF-1R
IAP
BTK
ATM/ATR
Hydroxylase
PLK
Tyrosinase
ADC Cytotoxin
Mdm2
Chloride channel
CETP
Leukotriene Receptor
ABC Transporter
OX Receptor
CaMK
Indoleamine 2,3-Dioxygenase (IDO)
DNA Methyltransferase
S6 Kinase
BACE
JNK
Cholecystokinin Receptor
Cysteine Protease
Glucosidase
Smo
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Ligand for E3 Ligase
Kinesin
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RIP kinase
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DNA
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GlyT
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Molecular Glues
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Fatty Acid Synthase
PAK
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PGE Synthase
IκB/IKK
GHSR
CGRP Receptor
Gap Junction Protein
NOD
IRAK
AhR
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IFNAR
Tie-2
IDO
MT Receptor
FAAH
MAPK
GPCR19
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CRFR
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Complement System
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Imidazoline Receptor
PROTACs
CRM1
DprE1
YAP
Cell wall
Melatonin Receptor
CaSR
Serine/threonin kinase
Annexin A
UGT
Neuropeptide Y Receptor
Somatostatin
Wee1
Lipid
OAT
STING
Decarboxylase
Neprilysin
GST
Acetyl-CoA Carboxylase
Kras
LPA Receptor
PDK
Oxytocin Receptor
Anti-infection
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PD-1/PD-L1
MicroRNA
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Arginase
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NAMPT
PYK2
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LDL
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Hexokinase
Epoxide Hydrolase
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transporter
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GSNOR
NEDD8
Ligands for Target Protein for PROTAC
PERK
Lipase
TOPK
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c-Myc
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IRE1
FLAP
Integrase
HCN Channel
Stearoyl-CoA Desaturase (SCD)
Thrombopoietin Receptor
ATP Citrate Lyase
BCRP
Glutathione reductase
Porcupine
CD73
GluCls
PAI-1
Pyroptosis
Aquaporin
Discoidin Domain Receptor (DDR)
p97
MLK
Apelin receptor
Adenylyl Cyclase
NPC1L1
Hydrogenase
RAR/RXR
MALT
Dynamin
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Arrestin
DYRK
gp120/CD4
GTPase
N-Acetylglucosaminyltransferase
AAK1
VDAC
Hck
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LIM Kinase
Stemness kinase
Immunology/Inflammation related
SIK
Adiponectin Receptor
PAFR
MTH1
Fas/FasL
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PROTAC Linker
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ACK1
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ASK
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SGK
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BMI-1
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