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κM-Conotoxin RIIIJ(κM-RIIIJ)是一种针对Kv1.2的选择性抑制剂,具有33 nM的IC50值。
κM-Conotoxin RIIIJ(κM-RIIIJ)是一种针对Kv1.2的选择性抑制剂,具有33 nM的IC50值。
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 5 mg | 待询 | 待询 | |
| 50 mg | 待询 | 待询 |
κM-Conotoxin RIIIJ 相关产品
| 产品描述 | κM-Conotoxin RIIIJ (κM-RIIIJ) selectively inhibits Kv1.2 channels, exhibiting an IC50 value of 33 nM [1]. |
| 别名 | κM-RIIIJ |
| 分子量 | 2807.3 |
| 分子式 | C117H184N32O36S6 |
| Sequence | Leu-{Hyp}-{Hyp}-Cys-Cys-Thr-{Hyp}-{Hyp}-Lys-Lys-His-Cys-{Hyp}-Ala-{Hyp}-Ala-Cys-Lys-Tyr-Lys-{Hyp}-Cys-Cys-Lys-Ser (Disulfide bridge:Cys4-Cys17, Cys5-Cys22, Cys12-Cys23) |
| Sequence Short | L-{Hyp}-{Hyp}-CCT-{Hyp}-{Hyp}-KKHC-{Hyp}-A-{Hyp}-ACKYK-{Hyp}-CCKS (Disulfide bridge:Cys4-Cys17, Cys5-Cys22, Cys12-Cys23) |
| 存储 | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
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