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Penthiopyrad

Name: Penthiopyrad
Brand: TargetMol
SKU: T16470
Price: 108 CNY
Availability: InStock
Rating: 5 (10 reviews)

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很棒

纯度: 99.88%

货号 T16470Cas号 183675-82-3

别名 吡噻菌胺, Vertisan, MTF-753

Penthiopyrad (MTF-753) 显示出广谱的抗真菌活性并抑制真菌呼吸。 Penthiopyrad 可用于叶面和土传植物病害的研究。

为众多的药物研发团队赋能，

让新药发现更简单！

Penthiopyrad

一键复制产品信息

很棒

纯度: 99.88%

货号 T16470 别名 吡噻菌胺, Vertisan, MTF-753Cas号 183675-82-3

Penthiopyrad (MTF-753) 显示出广谱的抗真菌活性并抑制真菌呼吸。 Penthiopyrad 可用于叶面和土传植物病害的研究。

规格	价格	库存
1 mg	¥ 108	现货
5 mg	¥ 198	现货
10 mg	¥ 289	现货
25 mg	¥ 579	现货
50 mg	¥ 953	现货
100 mg	¥ 1,490	现货
200 mg	¥ 2,190	现货
1 mL x 10 mM (in DMSO)	¥ 223	现货

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TargetMol的所有产品仅用作科学研究或药证申报，不能被用于人体，我们不向个人提供产品和服务。请您遵守承诺用途，不得违反法律法规规定用于任何其他用途。

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纯度: 99.88%

颜色: 白色

性状: Solid

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COA LCMS HNMR 产品操作手册

产品介绍

Penthiopyrad AI Summary

Penthiopyrad exhibits a broad range of bioactivities, particularly as a potent fungicide and antifungal agent. It shows significant efficacy against multiple fungal pathogens including powdery mildew (Podosphaera xanthii), Magnaporthe grisea (rice blast), Puccinia recondita (wheat brown rust), and Botryotinia fuckeliana (gray mold). Demonstrated under greenhouse conditions, it effectively reduces disease severity on various plant species such as Lagenaria siceraria and Cucurbita pepo, with efficacy varying between 0.03% to 14.6%. The compound also exhibits exceptional activity against sterol 14alpha-demethylation inhibitor-resistant strains of Oculimacula yallundae and boscalid-resistant Alternaria alternata, achieving high inhibition percentages of up to 90.53%. Beyond its fungicidal properties, Penthiopyrad also shows notable bioactivity in inhibiting mitochondrial enzymes in porcine hearts, including succinate-cytochrome c reductase (IC50 of 1321.0 nM) and succinate-ubiquinone oxidoreductase (IC50 of 1190.0 nM), and selectively inhibiting cytochrome b-c1 complex activity. Additionally, it exhibits antiviral properties against SARS-CoV-2, inhibiting the SARS-CoV-2 3CL-Pro protease by 6.27% at a 20 µM concentration and reducing virus-induced cytotoxicity in VERO-6 cells. These diverse activities suggest that Penthiopyrad holds potential as a broad-spectrum agrochemical and pharmacological agent with applications ranging from plant disease management to antiviral therapies..

Note: Summary generated by AI. Data source: ChEMBL

生物活性

产品描述	Penthiopyrad (MTF-753) shows a broad spectrum of antifungal activity and suppresses fungal respiration. Penthiopyrad can be used in studies about foliar and soil-borne plant diseases.
别名	吡噻菌胺, Vertisan, MTF-753

化学信息

分子量	359.41
分子式	C₁₆H₂₀F₃N₃OS
CAS No.	183675-82-3
Smiles	CC(C)CC(C)c1sccc1NC(=O)c1cn(C)nc1C(F)(F)F
密度	1.3g/cm3

储存&溶解度

存储

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

溶解度信息

DMSO: 90 mg/mL (250.41 mM), Sonication is recommended.

体内实验配方

10% DMSO+40% PEG300+5% Tween 80+45% Saline: 3.3 mg/mL (9.18 mM), Sonication is recommended.

请按顺序添加溶剂，在添加下一种溶剂之前，尽可能使溶液澄清。如有必要，可通过加热、超声、涡旋处理进行溶解。工作液建议现配现用。以上配方仅供参考，体内配方并不是绝对的，请根据不同情况进行调整。

溶液配制表

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.7823 mL	13.9117 mL	27.8234 mL	139.1169 mL
5 mM	0.5565 mL	2.7823 mL	5.5647 mL	27.8234 mL
10 mM	0.2782 mL	1.3912 mL	2.7823 mL	13.9117 mL
20 mM	0.1391 mL	0.6956 mL	1.3912 mL	6.9558 mL
50 mM	0.0556 mL	0.2782 mL	0.5565 mL	2.7823 mL
100 mM	0.0278 mL	0.1391 mL	0.2782 mL	1.3912 mL

计算器

摩尔浓度计算器
稀释计算器
配液计算器
分子量计算器

体内实验配液计算器

请在以下方框中输入您的动物实验信息后点击计算，可以得到母液配置方法和体内配方的制备方法：

比如您的给药剂量是10 mg/kg，每只动物体重20 g，给药体积100 μL，一共给药动物10只，您使用的配方为 10% DMSO + 40% PEG300 + 5% Tween 80 + 45% Saline / PBS / ddH₂O，那么您的工作液浓度为2 mg/mL。

母液配置方法：2 mg 药物溶于 100 μL DMSO （母液浓度为 20 mg/mL ）, 如您需要配置的浓度超过该产品的溶解度，请先与我们联系。