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抑制剂库

抑制剂库

产品编号 L2000 Inhibitor Library
  库化合物信息   Excel SDF

细胞信号控制细胞基本活动,调控细胞行为。细胞感知并准确响应微环境的变化是发育、组织修复和免疫的基础,也是正常组织稳态的基础。细胞信号间相互作用异常或细胞信息处理错误是导致癌症、自身免疫和糖尿病等疾病的原因。深入了解细胞信号传导,疾病可得到更有效的治疗。

TargetMol 抑制剂库是由7618 个靶向小分子化合物组成的集合,每一个化合物都有明确的抑制靶点,靶点所处的信号通路也因此被阻断,TargetMol 抑制剂库是研究信号通路及相关疾病的有力工具,可用于高通量筛选和高内涵筛选。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
我们的产品含有多种规格,如需了解具体的规格以及价格信息,请联系我们咨询订购,对于大额的订购,我们还有额外的优惠!
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如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 7618个小分子抑制剂的独特集合,主要用于细胞信号研究、新药筛选、高通量筛选和高内涵筛选;
  • 通过临床前研究和临床实验,生物活性和安全性已经得到验证;部分抑制剂已经被FDA批准上市;
  • 作用于MAPK、PI3K、JAK、HDAC、VEGFR、CDK等靶点,阻断相关信号通路;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2000)
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化合物库组成

Apoptosis (762)
Autophagy (583)
Antibacterial (436)
Antibiotic (252)
5-HT Receptor (214)
Endogenous Metabolite (200)
COX (192)
CDK (176)
DNA/RNA Synthesis (167)
NF-κB (160)
HIV Protease (159)
PI3K (159)
AChR (156)
EGFR (149)
Dopamine Receptor (143)
VEGFR (141)
Parasite (129)
Antifungal (128)
Adrenergic Receptor (127)
Epigenetic Reader Domain (125)
P450 (121)
PDE (120)
Dehydrogenase (120)
Histamine Receptor (118)
Histone Methyltransferase (107)
HDAC (106)
Potassium Channel (103)
Calcium Channel (96)
JAK (91)
FLT (89)
Src (88)
PDGFR (87)
mTOR (87)
Influenza Virus (86)
Sodium Channel (82)
Topoisomerase (82)
Microtubule Associated (80)
Phosphatase (78)
SARS-CoV (75)
FGFR (74)
Akt (73)
ERK (73)
STAT (72)
TRP/TRPV Channel (72)
AChE (71)
Reactive Oxygen Species (70)
Raf (69)
c-Kit (67)
PKC (67)
p38 MAPK (66)
PARP (66)
TNF (65)
Wnt/beta-catenin (62)
c-Met/HGFR (62)
HCV Protease (61)
Prostaglandin Receptor (59)
RAAS (58)
Bcr-Abl (58)
Ferroptosis (58)
Proteasome (57)
GABA Receptor (57)
Ras (56)
BCL (53)
GSK-3 (53)
Aurora Kinase (52)
MMP (52)
Virus Protease (50)
ALK (50)
Lipoxygenase (49)
MAO (49)
PPAR (47)
Adenosine Receptor (46)
HSP (46)
NMDAR (46)
Phospholipase (45)
NO Synthase (45)
Tyrosinase (44)
IL Receptor (43)
Antioxidant (43)
TGF-beta/Smad (42)
MEK (41)
iGluR (41)
JNK (41)
DUB (41)
E1/E2/E3 Enzyme (41)
Beta Amyloid (41)
GluR (40)
ATPase (39)
Mitophagy (39)
Tyrosine Kinases (39)
Monoamine Oxidase (39)
BTK (38)
GPR (38)
CCR (38)
Caspase (38)
Casein Kinase (38)
HER (37)
DNA-PK (37)
Reverse Transcriptase (37)
HSV (36)
P-gp (36)
Serine/threonin kinase (36)
ROCK (36)
MAPK (36)
HBV (35)
IκB/IKK (35)
Histone Demethylase (35)
CXCR (34)
Sirtuin (34)
AMPK (34)
HIF/HIF Prolyl-Hydroxylase (34)
Androgen Receptor (34)
Serotonin Transporter (34)
Transferase (33)
Interleukin (33)
Mitochondrial Metabolism (33)
Estrogen Receptor/ERR (33)
Cysteine Protease (33)
Estrogen/progestogen Receptor (33)
c-RET (32)
CaMK (32)
Nucleoside Antimetabolite/Analog (32)
TAM Receptor (32)
Integrin (32)
HIF (31)
TLR (31)
PKA (31)
Anti-infection (30)
NOS (29)
ROS (29)
Serine Protease (28)
Gamma-secretase (28)
Carbonic Anhydrase (28)
S6 Kinase (27)
Trk receptor (27)
Histone Acetyltransferase (27)
IGF-1R (27)
Proton pump (27)
Drug Metabolite (27)
Opioid Receptor (27)
P2X Receptor (26)
Norepinephrine (26)
Hedgehog/Smoothened (25)
FAK (25)
FAAH (25)
PLK (25)
c-Fms (24)
Reductase (24)
RIP kinase (24)
DPP-4 (23)
Glucosidase (23)
Indoleamine 2,3-Dioxygenase (IDO) (23)
DNA Methyltransferase (23)
Cannabinoid Receptor (23)
ribosome (22)
Syk (22)
Glucocorticoid Receptor (22)
Fatty Acid Synthase (21)
Antiviral (21)
p53 (21)
Kinesin (20)
Neurokinin receptor (20)
Pim (20)
Chk (20)
ATM/ATR (20)
SGLT (19)
Antifection (19)
HMG-CoA Reductase (19)
Nrf2 (19)
LPL Receptor (19)
S1P Receptor (18)
Chloride channel (18)
LRRK2 (18)
transporter (17)
Lipase (17)
Complement System (17)
Acyltransferase (17)
NOD (17)
Mdm2 (17)
Smo (17)
PAK (17)
Endothelin Receptor (17)
PDK (17)
OX Receptor (16)
Leukotriene Receptor (16)
Epoxide Hydrolase (16)
NADPH (16)
MRP (16)
IRAK (15)
NOD-like Receptor (NLR) (15)
P2Y Receptor (15)
Xanthine Oxidase (15)
Rho (15)
Glutathione Peroxidase (15)
BACE (14)
IRE1 (14)
Hydroxylase (14)
DYRK (14)
c-Myc (14)
Thrombin (13)
Retinoid Receptor (13)
CSF-1R (13)
Sigma receptor (13)
cAMP (13)
LTR (13)
Glucokinase (13)
PI4K (13)
PGE Synthase (13)
Aryl Hydrocarbon Receptor (12)
LPA Receptor (12)
PD-1/PD-L1 (12)
Ephrin Receptor (12)
Immunology/Inflammation related (12)
Aminopeptidase (12)
Antifolate (12)
PERK (12)
Protease-activated Receptor (12)
Acetyl-CoA Carboxylase (11)
AhR (11)
IDO (11)
Aromatase (11)
Neuropeptide Y Receptor (11)
Beta-Secretase (11)
Stearoyl-CoA Desaturase (SCD) (11)
Isocitrate Dehydrogenase (IDH) (11)
Factor Xa (11)
ROS Kinase (11)
STING (11)
GTPase (10)
Myosin (10)
DHFR (10)
PAI-1 (10)
Discoidin Domain Receptor (DDR) (10)
Vasopressin Receptor (10)
Melanocortin Receptor (9)
GNRH Receptor (9)
IAP (9)
SGK (9)
ATP Citrate Lyase (9)
Monoamine Transporter (9)
Telomerase (9)
RSV (9)
cholecystokinin (9)
Monocarboxylate transporter (9)
NAMPT (8)
CETP (8)
DNA gyrase (8)
YAP (8)
BCRP (8)
Porcupine (8)
PAD (8)
Phosphorylase (8)
NADPH-oxidase (7)
PTEN (7)
p97 (7)
ROR (7)
Na+/Ca2+ Exchanger (7)
Neprilysin (7)
GRK (7)
Lipid (7)
CFTR (7)
Tie-2 (7)
DNA (7)
ASK (7)
Ligands for Target Protein for PROTAC (7)
MLK (6)
MNK (6)
Guanylate cyclase (6)
Dynamin (6)
Adenylyl cyclase (6)
MAGL (6)
OAT (6)
SIK (6)
Platelet aggregation (6)
ABC (6)
TOPK (5)
Adenosine deaminase (5)
CAT (5)
APC (5)
Aquaporin (5)
Neurotensin Receptor (5)
BMI-1 (5)
Bradykinin Receptor (5)
Thyroid hormone receptor(THR) (5)
LIM Kinase (5)
GlyT (5)
Liver X Receptor (5)
GPX (5)
PAFR (5)
CRFR (5)
Carboxypeptidase (5)
cGAS (5)
CRISPR/Cas9 (5)
FLAP (5)
Wee1 (5)
CRM1 (5)
Progesterone Receptor (5)
MELK (5)
MTH1 (5)
DprE1 (5)
Glutaminase (5)
Gap Junction Protein (5)
UGT (5)
DNA Alkylator/Crosslinker (5)
Glucagon Receptor (5)
GST (5)
Arginase (4)
VDAC (4)
PYK2 (4)
IFNAR (4)
ACK (4)
CaSR (4)
Decarboxylase (4)
NPC1L1 (4)
Hck (4)
MALT (4)
Amino Acids and Derivatives (4)
Methionine Adenosyltransferase (MAT) (4)
DNA Alkylation (4)
Ligand for E3 Ligase (4)
LDL (4)
Bombesin Receptor (4)
Survivin (4)
Angiotensin-converting Enzyme (ACE) (4)
CGRP Receptor (4)
NEDD8 (4)
Galectin (4)
MT Receptor (4)
KSP (4)
CD73 (3)
PKM (3)
AAK1 (AP2 associated kinase 1) (3)
Hexokinase (3)
Melatonin Receptor (3)
MyD88 (3)
CD38 (3)
Hippo pathway (3)
Pyroptosis (3)
OXPHOS (3)
Imidazoline Receptor (3)
FXR (3)
RANKL/RANK (2)
RAR/RXR  (2)
hCE (2)
GHSR (2)
Na-K-Cl cotransporter (2)
Transaminase (2)
KLF (2)
Integrase (2)
Prolyl Endopeptidase (PREP) (2)
Melanin-concentrating Hormone Receptor (MCHR) (2)
TSH Receptor (2)
Necroptosis (2)
advanced glycation end products (2)
Apelin receptor (2)
Fas/FasL (2)
EBI2/GPR183 (2)
Somatostatin (2)
LHRH (2)
Oxytocin Receptor (2)
Haspin Kinase (2)
Free radical scavengers (2)
HCN Channel (2)
PROTACs (1)
PROTAC Linker (1)
Protease (1)
Cell wall (1)
Fer/FerT kinase (1)
gp120/CD4 (1)
lysosomal autophagy (1)
Neuropeptide W (1)
Taste receptor (1)
Stemness kinase (1)
GPCR19 (1)
Thioredoxin (1)
stilbene oxidase (1)
Anion Exchanger (1)
VDA (1)
cell cycle arrest (1)
PGC-1α (1)
N-Acetylglucosaminyltransferase (1)
DAPK (1)
aconitase (1)
GSNOR (1)
NUDIX hydrolase (1)
GluCls (1)
FABP (1)
Molecular Glues (1)
Annexin A (1)
FOXO1 (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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