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- 9730个小分子抑制剂的独特集合，主要用于细胞信号研究、新药筛选、高通量筛选和高内涵筛选；
- 通过临床前研究和临床实验，生物活性和安全性已经得到验证；部分抑制剂已经被FDA批准上市；
- 作用于MAPK、PI3K、JAK、HDAC、VEGFR、CDK等靶点，阻断相关信号通路；
- 结构多样，药效显著，可渗透细胞；
- 详细的说明书，化合物结构、靶点信息、IC50值、活性描述等；
- NMR、HPLC/LCMS等多种检测技术保证产品结构正确，纯度高，减少假阳性。
抑制剂库
Inhibitor Library
很棒细胞信号控制细胞基本活动，调控细胞行为。细胞感知并准确响应微环境的变化是发育、组织修复和免疫的基础，也是正常组织稳态的基础。细胞信号间相互作用异常或细胞信息处理错误是导致癌症、自身免疫和糖尿病等疾病的原因。深入了解细胞信号传导，疾病可得到更有效的治疗。 TargetMol 抑制剂库是由9730 个靶向小分子化合物组成的集合，每一个化合物都有明确的抑制靶点，靶点所处的信号通路也因此被阻断，TargetMol 抑制剂库是研究信号通路及相关疾病的有力工具，可用于高通量筛选和高内涵筛选。
TargetMol 的所有产品和服务仅用于科学研究，不能被用于人体，我们也不向个人提供产品和服务。
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化合物库相关信息
Excel
SDF
联系我们获取更多批次信息产品编号 L2000
抑制剂库规格
- 1 mg
- 30 μL x 10 mM (in DMSO)
- 50 μL x 10 mM (in DMSO)
- 100 μL x 10 mM (in DMSO)
- 250 μL x 10 mM (in DMSO)
询价 & 定制
产品描述
包装和储存
- 可选用DMSO耐受的96/384孔板或2D 条形码编码管；
- 干粉蓝冰运输，DMSO溶液干冰运输；
- 排布：96孔板：1st & 12th 空白对照，384孔板：1st & 2nd & 23th & 24th空白对照。
SCI 文献
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化合物库组成
Apoptosis
Autophagy
Antibacterial
5-HT Receptor
CDK
COX
Antibiotic
AChR
PI3K
EGFR
HIV Protease
Endogenous Metabolite
DNA/RNA Synthesis
Adrenergic Receptor
Dopamine Receptor
Calcium Channel
PDE
NF-κB
VEGFR
Epigenetic Reader Domain
Dehydrogenase
Histamine Receptor
Histone Methyltransferase
Cytochromes P450
Potassium Channel
Sodium Channel
Parasite
HDAC
Phosphatase
JAK
Antifungal
mTOR
Src
FLT
Microtubule Associated
Topoisomerase
TRP/TRPV Channel
SARS-CoV
PDGFR
Cholinesterase (ChE)
PARP
FGFR
PKC
Raf
Wnt/beta-catenin
Akt
STAT
p38 MAPK
Influenza Virus
HCV Protease
RAAS
ERK
c-Kit
GSK-3
Prostaglandin Receptor
MAO
GABA Receptor
c-Met/HGFR
Lipoxygenase
Bcr-Abl
ALK
TNF
NMDAR
MMP
Proteasome
Reactive Oxygen Species
Adenosine Receptor
GluR
Bcl-2 Family
DUB
HSP
Phospholipase
Ferroptosis
Aurora Kinase
Histone Demethylase
Virus Protease
TGF-beta/Smad
Tyrosinase
GPR
ROCK
iGluR
IL Receptor
MAPK
Ras
Transferase
Tyrosine Kinases
ATPase
HER
E1/E2/E3 Enzyme
CCR
Integrin
PKA
Casein Kinase
MEK
NO Synthase
Beta Amyloid
JNK
PPAR
Caspase
Antiviral
Monoamine Oxidase
Serine/threonin kinase
Carbonic Anhydrase
Serotonin Transporter
IκB/IKK
Reverse Transcriptase
Antioxidant
Mitophagy
Cysteine Protease
Androgen Receptor
DNA-PK
HBV
Mitochondrial Metabolism
HSV
AMPK
CXCR
Sirtuin
c-RET
Reductase
NOS
ROS
Norepinephrine
HIF
TAM Receptor
Estrogen/progestogen Receptor
RIP kinase
P2X Receptor
IGF-1R
P-gp
Estrogen Receptor/ERR
Serine Protease
CaMK
Histone Acetyltransferase
Nucleoside Antimetabolite/Analog
Gamma-secretase
Drug Metabolite
Glucosidase
TLR
HIF/HIF Prolyl-Hydroxylase
Interleukin
Trk receptor
FAK
Proton pump
Hedgehog/Smoothened
FAAH
Acyltransferase
c-Fms
PLK
S6 Kinase
Cannabinoid Receptor
Opioid Receptor
ATM/ATR
Neurokinin receptor
Syk
p53
Glucocorticoid Receptor
DPP-4
Endothelin Receptor
NOD
HMG-CoA Reductase
Pim
Chk
Fatty Acid Synthase
Kinesin
Chloride channel
DYRK
Antifection
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
Anti-infection
IRAK
LTR
NADPH
Rho
Leukotriene Receptor
LRRK2
transporter
Thrombin
Mdm2
LPL Receptor
BACE
Lipase
Factor Xa
Xanthine Oxidase
PDK
DNA Methyltransferase
Immunology/Inflammation related
Nrf2
Sigma receptor
PD-1/PD-L1
S1P Receptor
BTK
P2Y Receptor
PERK
Glutathione Peroxidase
Smo
cAMP
Kras
Hydroxylase
DHFR
MRP
PAK
Epoxide Hydrolase
Retinoid Receptor
Cholecystokinin Receptor
Glucokinase
OX Receptor
LPA Receptor
PI4K
Complement System
ROS Kinase
YAP
c-Myc
IRE1
Neuropeptide Y Receptor
ribosome
GTPase
Aryl Hydrocarbon Receptor
IAP
CSF-1R
Myosin
Ephrin Receptor
Aromatase
AhR
Antifolate
DNA
PGE Synthase
Aminopeptidase
Protease-activated Receptor
ABC Transporter
Monoamine Transporter
Telomerase
Beta-Secretase
RSV
Discoidin Domain Receptor (DDR)
ADC Cytotoxin
MicroRNA
Monocarboxylate transporter
CETP
Glutaminase
IDO
Isocitrate Dehydrogenase (IDH)
Stearoyl-CoA Desaturase (SCD)
Vasopressin Receptor
Acetyl-CoA Carboxylase
Platelet aggregation
NOD-like Receptor (NLR)
GRK
DNA gyrase
Bradykinin Receptor
Lipid
PAI-1
Melanocortin Receptor
NADPH-oxidase
CFTR
MLK
GNRH Receptor
LIM Kinase
NAMPT
ATP Citrate Lyase
BCRP
MNK
STING
Neprilysin
SGK
Dynamin
Ligands for Target Protein for PROTAC
Tie-2
PAFR
LDL
Glucagon Receptor
Phosphorylase
GlyT
PAD
OAT
Porcupine
ASK
Carboxypeptidase
Adenylyl Cyclase
CRM1
Na+/Ca2+ Exchanger
AAK1
Neurotensin Receptor
PYK2
SIK
UGT
MAGL
DNA Alkylation
Angiotensin-converting Enzyme (ACE)
Wee1
CRFR
GST
GPX
APC/C
p97
Thyroid hormone receptor(THR)
ROR
Progesterone Receptor
FLAP
MT Receptor
Guanylate cyclase
cGAS
MELK
Methionine Adenosyltransferase (MAT)
Ligand for E3 Ligase
Protease
CGRP Receptor
Gap Junction Protein
Melanin-concentrating Hormone Receptor (MCHR)
PROTACs
MALT
Amino Acids and Derivatives
MyD88
DprE1
DNA Alkylator/Crosslinker
Amylase
MTH1
Bombesin Receptor
ACK1
Survivin
CD73
Decarboxylase
Pyroptosis
Hippo pathway
CRISPR/Cas9
Aquaporin
GHSR
Adenosine Deaminase
DAPK
BMI-1
Advanced Glycation End Products
NPC1L1
CD38
NEDD8
Melatonin Receptor
Galectin
CaSR
VDAC
Hexokinase
HCN Channel
PTEN
KSP
Imidazoline Receptor
Apelin receptor
Transaminase
Arginase
Arrestin
IFNAR
Necroptosis
TOPK
Hck
Liver X Receptor
Haspin Kinase
OXPHOS
TSH Receptor
HuR
Oxytocin Receptor
PKM
GSNOR
NUDIX hydrolase
EBI2/GPR183
Glutaminyl Cyclase
gp120/CD4
Kisspeptin
FXR
FOXO1
Prolyl Endopeptidase (PREP)
Na-K-Cl cotransporter
Molecular Glues
Integrase
Somatostatin
Transketolase
AIM2
hCE
KLF
Drug-Linker Conjugates for ADC
Taste receptor
stilbene oxidase
RAR/RXR
Piezo Channel
Procollagen C Proteinase
Aconitase
Neuropeptide W
Cell wall
LHRH
VDA
OCT
N-Acetylglucosaminyltransferase
Stemness kinase
RANKL/RANK
Adiponectin Receptor
Fas/FasL
FABP
PACAP
Anion Exchanger
Thioredoxin
Mucin
PSMA
Glutathione reductase
MRGPR
GPCR19
CPT
GluCls
Fer/FerT kinase
Lysosomal Autophagy
Glyoxalase
Sodium-dependent phosphate transporter
Vitamin
PGC-1α
化合物库信息
| Empty | 99-93-4 | 99899-45-3 | 99873-43-5 | 99755-59-6 | 99754-06-0 | 99-66-1 | 99614-02-5 | 99614-01-4 | 99522-79-9 | 99464-64-9 | Empty |
| 4-Hydroxyacetophenone | SM-2470 | Droxinostat | Rotigotine- | ONO-RS-082 | Valproic Acid | Ondansetron | Ondansetron hydrochloride | Pranidipine | Ampiroxicam | ||
| Empty | 99390-76-8 | 99365-23-8 | 99353-00-1 | 99-32-1 | 99300-78-4 | 99291-25-5 | 99254-95-2 | 99248-32-5 | 99-24-1 | 99201-87-3 | Empty |
| BMY-27709 | Prosaikogenin G | Methyl rosmarinate | Chelidonic acid | Venlafaxine hydrochloride | Levodropropizine | McN5691 | Donetidine | Methyl gallate | Anpirtoline hydrochloride | ||
| Empty | 99-14-9 | 99134-29-9 | 99105-77-8 | 99009-20-8 | 98991-32-3 | 98-98-6 | 989-51-5 | 989-30-0 | 98769-84-7 | 98717-15-8 | Empty |
| Tricarballylic acid | L 651896 | Sulcotrione | Pyrazoloacridine | CHBO4 | PCL 016 | (-)-Epigallocatechin Gallate | 3-Epiursolic acid | Reboxetine mesylate | Ropivacaine hydrochloride | ||
| Empty | 98665-15-7 | 98636-73-8 | 985-12-6 | 98410-36-7 | 98319-26-7 | 982-57-0 | 98207-12-6 | 98206-09-8 | 981-15-7 | 98-10-2 | Empty |
| Ganoderic acid F | Nitrocaramiphen hydrochloride | Drotaverine hydrochloride | Palatrigine | Finasteride | Chloramphenicol succinate sodium | Lobuprofen | Eltoprazine hydrochloride | Ailanthone | Benzenesulfonamide | ||
| Empty | 98079-52-8 | 980-71-2 | 979-92-0 | 97938-31-3 | 978-62-1 | 977-96-8 | 97-77-8 | 97743-99-2 | 97730-95-5 | 97682-44-5 | Empty |
| Lomefloxacin hydrochloride | Brompheniramine maleate | SAH | Leachianone A | IMD-0354 | Decynium 22 | Disulfiram | rac Desmethyl Citalopram Hydrochloride | DPI 201-106 | Irinotecan | ||
| Empty | 97677-19-5 | 976-71-6 | 97657-92-6 | 973-67-1 | 97240-79-4 | 97230-47-2 | 97230-46-1 | 969-33-5 | 968-81-0 | 96847-55-1 | Empty |
| Alconil | Canrenone | Latrepirdine dihydrochloride | 5,6,7-TRIMETHOXYFLAVONE | Topiramate | Picfeltarraenin IA | Picfeltarraenin IB | Cyproheptadine hydrochloride | Acetohexamide | Dextromilnacipran | ||
| Empty | 96829-58-2 | 96736-11-7 | 96609-16-4 | 96574-01-5 | 96566-25-5 | 96553-02-5 | 965-52-6 | 96-50-4 | 96489-71-3 | 964-52-3 | Empty |
| Orlistat | Nourseothricin sulfate | Lifibrol | Salvianolic acid A | Ablukast | Gypsogenin-3-O-glucuronide | Nifuroxazide | Aminothiazole | Pyridaben | Moxisylyte hydrochloride | ||
| Empty | 96441-14-4 | 96224-26-9 | 96206-92-7 | 96201-88-6 | 96187-53-0 | 960404-48-2 | 960374-59-8 | 960293-88-3 | 96020-91-6 | 960203-27-4 | Empty |
| Labetalone hydrochloride | CL 277082 | MPEP | Brequinar sodium | Brequinar | Dapagliflozin ((2S)-1,2-propanediol, hydrate) | ONX-0914 | BI605906 | Eflornithine hydrochloride hydrate | Vortioxetine hydrobromide |
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