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T-10418是一种高效和选择性的G2A/GPR132 激动剂(EC50=0.82 μM),能增强在小鼠原代感觉神经元中的TRPV1反应,可用于研究神经性疼痛和炎症。
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T-10418是一种高效和选择性的G2A/GPR132 激动剂(EC50=0.82 μM),能增强在小鼠原代感觉神经元中的TRPV1反应,可用于研究神经性疼痛和炎症。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 1,280 | In stock | |
5 mg | ¥ 3,190 | In stock | |
10 mg | ¥ 4,590 | In stock | |
25 mg | ¥ 6,930 | In stock | |
50 mg | ¥ 9,550 | In stock | |
100 mg | ¥ 12,800 | In stock | |
200 mg | ¥ 17,300 | In stock | |
1 mL x 10 mM (in DMSO) | ¥ 2,650 | In stock |
T-10418 相关产品
产品描述 | T-10418 is a highly potent and selective G2A/GPR132 agonist (EC50 = 0.82 μM) that enhances TRPV1 responses in mouse primary sensory neurons, making it suitable for studying neuropathic pain and inflammation. |
体外活性 | 方法: |
分子量 | 376.41 |
分子式 | C22H20N2O4 |
CAS No. | 1608784-68-4 |
Smiles | C(N[C@H](CC1=CC=CC=C1)C(O)=O)(=O)C2=CC(OCC=3C=CC=NC3)=CC=C2 |
颜色 | Yellow |
物理性状 | Solid |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 80 mg/mL (212.53 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO
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以上为“体内实验配液计算器”的使用方法举例,并不是具体某个化合物的推荐配制方式,请根据您的实验动物和给药方式选择适当的溶解方案。
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