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CBM-301940 (compound 5) 是一种高效和具有口服活性的MCD(Malonyl-CoA Decarboxylase)抑制剂,IC50=23 nM,改善了大鼠心脏缺血/再灌注模型的心脏效率和功能,具有心脏保护功能。
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CBM-301940 (compound 5) 是一种高效和具有口服活性的MCD(Malonyl-CoA Decarboxylase)抑制剂,IC50=23 nM,改善了大鼠心脏缺血/再灌注模型的心脏效率和功能,具有心脏保护功能。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 945 | In stock | |
5 mg | ¥ 2,080 | In stock | |
10 mg | ¥ 3,330 | In stock | |
25 mg | ¥ 5,660 | In stock | |
50 mg | ¥ 8,490 | In stock | |
100 mg | ¥ 12,700 | In stock |
产品描述 | CBM-301940 (compound 5) is a potent and orally active MCD (Malonyl-CoA Decarboxylase) inhibitor with IC50=23 nM that improves cardiac efficiency and function with cardioprotective properties in a rat cardiac ischemia/reperfusion model. |
靶点活性 | Malonyl-CoA decarboxylase (MCD):23 nM |
体外活性 | CBM-301940(化合物5)是一种口服活性的丙二酸辅酶A脱羧酶(MCD)抑制剂,其 IC₅₀ 值为 23 nM[1]。 |
别名 | CBM301940 |
分子量 | 422.32 |
分子式 | C15H20F6N2O5 |
CAS No. | 902146-11-6 |
Smiles | O=C(NC(C)CC(=O)OC(C)(C)C)C1=NOC(C1)C(O)(C(F)(F)F)C(F)(F)F |
存储 | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
以上为“体内实验配液计算器”的使用方法举例,并不是具体某个化合物的推荐配制方式,请根据您的实验动物和给药方式选择适当的溶解方案。
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