YAP-TEAD-IN-1 TFA

Name: YAP-TEAD-IN-1 TFA
Brand: TargetMol
SKU: TP2160L
Rating: 4.5 (1 reviews)

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产品编号 TP2160LCas号 1659305-79-9

YAP-TEAD-IN-1 TFA, a competitive inhibitor of the YAP–TEAD interaction (IC50: 25 nM), exhibits higher binding affinity to TEAD1 (Kd: 15 nM) compared to YAP (50-171) (Kd: 40 nM).

YAP-TEAD-IN-1 TFA

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产品编号 TP2160LCas号 1659305-79-9

YAP-TEAD-IN-1 TFA, a competitive inhibitor of the YAP–TEAD interaction (IC50: 25 nM), exhibits higher binding affinity to TEAD1 (Kd: 15 nM) compared to YAP (50-171) (Kd: 40 nM).

规格	价格	库存	数量
10 mg	¥ 1,650	5日内发货

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产品介绍

生物活性

产品描述	YAP-TEAD-IN-1 TFA, a competitive inhibitor of the YAP–TEAD interaction (IC50: 25 nM), exhibits higher binding affinity to TEAD1 (Kd: 15 nM) compared to YAP (50-171) (Kd: 40 nM).
靶点活性	YAP-TEAD:25 nM
体外活性	In a GST pull-down assay, YAP-TEAD-IN-1 (2 μM) is against endogenous YAP binding to GST-TEAD (1209-426), the Kd of His-YAP1209-426 is determined to be 40 nM.

化学信息

分子式	C₉₃H₁₄₄ClN₂₃O₂₁S₂.xC₂HF₃O₂
CAS No.	1659305-79-9
密度	1.31g/cm3
Sequence	Ac-Val-Pro-{Phe(3-Cl)}-{Hcy}-Leu-Arg-Lys-{Nle}-Pro-Ala-Ser-Phe-Cys-Lys-Pro-Pro-Glu-NH2 (Disulfide bridge:Hcy4-Cys13)
Sequence Short	Ac-VP-{Phe(3-Cl)}-{Hcy}-LRK-{Nle}-PASFCKPPE-NH2 (Disulfide bridge:Hcy4-Cys13)