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肠道微生物代谢化合物库

肠道微生物代谢化合物库

产品编号 L2540 Gut Microbial Metabolite Library
  库化合物信息   Excel SDF

肠道菌群在人体内形成了错综复杂的微生态系统,肠道微生物基因组中富含参与碳水化合物、氨基酸、甲烷、维生素和短链脂肪酸代谢的基因,其中很大一部分是人体自身所不具备的,表明肠道微生物是人体代谢的重要参与者,人体代谢平衡状况与肠道菌群的结构组成变化密不可分。

肠道菌群与人类健康息息相关,肠道菌群异常可能导致多种代谢疾病发生,包括肥胖、2型糖尿病、非酒精性脂肪肝、代谢性心脏病和营养不良等。此外,由于肠道是人体内重要的免疫器官,肠道微生物与宿主在肠道黏膜表面的交流促进了免疫系统的建立和发展,成为人体重要的免疫屏障。肠道菌群代谢产物和衍生物可作为菌群的“信使”,影响宿主能量稳态、机体肥胖、葡萄糖耐量、炎症和内分泌调节等,调控宿主代谢。因此研究肠道微生物代谢产物可能有助于发现某些疾病发病机制及开发有效治疗方法。

TargetMol 肠道微生物代谢化合物库收集了614 种肠道微生物代谢物,可以用于肠道菌群的相关研究及药物开发。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 614 种肠道微生物代谢物的集合,可以用于高通量和高内涵筛选;
  • 包含脂肪酸、氨基酸、维生素、糖类、脂质等化合物类型;
  • 研究肠道菌群代谢和相关药物开发的有效工具;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

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包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2540)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Endogenous Metabolite (508)
Apoptosis (36)
Autophagy (27)
Antibacterial (26)
Antioxidant (12)
Influenza Virus (12)
Reactive Oxygen Species (11)
Antifungal (9)
Amino Acids and Derivatives (9)
PPAR (9)
Ferroptosis (9)
DNA/RNA Synthesis (7)
Antibiotic (7)
5-HT Receptor (6)
NF-κB (6)
Calcium Channel (5)
Nrf2 (5)
TNF (5)
COX (5)
Dehydrogenase (5)
iGluR (5)
Caspase (4)
Parasite (4)
Virus Protease (4)
Nucleoside Antimetabolite/Analog (4)
Mitophagy (4)
NO Synthase (4)
TRP/TRPV Channel (4)
Adenosine Receptor (4)
P450 (4)
Tyrosinase (4)
Akt (3)
GPCR19 (3)
MMP (3)
ERK (3)
Chloride channel (3)
ROS (3)
AMPK (3)
NMDAR (3)
GABA Receptor (3)
PDE (3)
AhR (3)
Histone Acetyltransferase (3)
HIV Protease (3)
p38 MAPK (3)
PI3K (3)
Histamine Receptor (3)
FXR (3)
Phosphatase (3)
Arginase (2)
Potassium Channel (2)
Mitochondrial Metabolism (2)
PARP (2)
Transferase (2)
FGFR (2)
Estrogen/progestogen Receptor (2)
Adrenergic Receptor (2)
GluR (2)
Epigenetic Reader Domain (2)
Imidazoline Receptor (2)
Aryl Hydrocarbon Receptor (2)
HDAC (2)
PKC (1)
GPR (1)
P2Y Receptor (1)
Reductase (1)
Decarboxylase (1)
aconitase (1)
Beta Amyloid (1)
HIF (1)
Dopamine Receptor (1)
ROR (1)
PLK (1)
Histone Demethylase (1)
DHFR (1)
Monocarboxylate transporter (1)
Cannabinoid Receptor (1)
AChR (1)
Neurokinin receptor (1)
Anti-infection (1)
NOD (1)
Carbonic Anhydrase (1)
HIF/HIF Prolyl-Hydroxylase (1)
ATPase (1)
CFTR (1)
Sirtuin (1)
P-gp (1)
Trk receptor (1)
IL Receptor (1)
MAO (1)
Glucokinase (1)
Glucocorticoid Receptor (1)
LDL (1)
Drug Metabolite (1)
MT Receptor (1)
Phosphorylase (1)
GlyT (1)
Antifection (1)
Wnt/beta-catenin (1)
Estrogen Receptor/ERR (1)
HBV (1)
Fatty Acid Synthase (1)
HSV (1)
Melatonin Receptor (1)
Prostaglandin Receptor (1)
JNK (1)
HSP (1)
Antiviral (1)
Lipase (1)
Acyltransferase (1)
AChE (1)
MAPK (1)
ATP Citrate Lyase (1)
Lipoxygenase (1)
EGFR (1)
TGF-beta/Smad (1)
Glutathione Peroxidase (1)
mTOR (1)
CaMK (1)
IGF-1R (1)
Opioid Receptor (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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