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Adenosine receptor A1 antagonist 5
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很棒纯度: 99.97%
货号 T22466Cas号 85872-53-3
Adenosine receptor A1 antagonist 5 可作为一种腺苷拮抗剂，是一种氧嘌呤，可作为杀虫剂和虫害防治剂，对血压升高有抑制作用。
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Adenosine receptor A1 antagonist 5
一键复制产品信息 很棒纯度: 99.97%
货号 T22466Cas号 85872-53-3
Adenosine receptor A1 antagonist 5 可作为一种腺苷拮抗剂，是一种氧嘌呤，可作为杀虫剂和虫害防治剂，对血压升高有抑制作用。
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 1 mg | ¥ 288 | 现货 | |
| 5 mg | ¥ 700 | 现货 | |
| 10 mg | ¥ 1,020 | 现货 | |
| 25 mg | ¥ 1,720 | 现货 | |
| 50 mg | ¥ 2,470 | 现货 | |
| 100 mg | ¥ 3,430 | 现货 | |
| 200 mg | ¥ 4,610 | 现货 |
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产品介绍
Adenosine receptor A1 antagonist 5 AI Summary
Adenosine receptor A1 antagonist 5 exhibits bioactivity primarily as a ligand for adenosine receptors, displaying high binding affinity for the A1 adenosine receptor (Ki = 2.75 nM in rat cortex) and moderate binding affinity for the A2A adenosine receptor (Ki = 116.0 nM in rat striatal membranes). It also shows significant binding affinity for the human HEK293 adenosine A2B receptor (Ki = 18.9 nM). The compound acts as an antagonist at these receptors, inhibiting adenyl cyclase stimulation in various membranes, such as human platelet and rat PC12 membranes, with Ki values indicating a preference for A1 receptors over A2 receptors. Additionally, Adenosine receptor A1 antagonist 5 demonstrates a range of bioactivities, including inhibition of [3H]-PIA binding at adenosine A1 receptors, antagonism at both adenosine A1 and A2 receptors, and inhibition of adenylate cyclase stimulation. Beyond its role in adenosine receptor interaction, the compound shows diverse activity across various biological targets, including inhibitory effects on SARS-CoV-2 cytotoxicity, inhibition of HSD17B4 and JMJD2E, antiviral properties against Lassa and Marburg viruses, and modulation of Cytochrome P450 enzymes..
Note: Summary generated by AI. Data source: ChEMBL 
生物活性
化学信息
储存&溶解度
| 产品描述 | Adenosine receptor A1 antagonist 5 acts as an adenosine antagonist, is an oxypurine, acts as an insecticide and pest control agent, and has an inhibitory effect on elevated blood pressure. |
| 分子量 | 312.37 |
| 分子式 | C17H20N4O2 |
| CAS No. | 85872-53-3 |
| Smiles | C(CC)N1C2=C(NC(=N2)C3=CC=CC=C3)C(=O)N(CCC)C1=O |
| 密度 | 1.218g/cm3 |
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | ||||||||||||||||||||||||||||||
| 溶解度信息 | Ethanol: 4.5 mg/mL (14.41 mM), Sonication is recommended. DMSO: 8 mg/mL (25.61 mM), Sonication is recommended.  | ||||||||||||||||||||||||||||||
溶液配制表 | |||||||||||||||||||||||||||||||
Ethanol/DMSO
DMSO
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计算器
体内实验配液计算器
请在以下方框中输入您的动物实验信息后点击计算，可以得到母液配置方法和体内配方的制备方法：
比如您的给药剂量是10 mg/kg，每只动物体重20g，给药体积100 μL， 一共给药动物10只，您使用的配方为5%
DMSO + 30%PEG300 + 5%Tween 80 + 60%Saline/PBS/ddH2O， 那么您的工作液浓度为2mg/mL。 以上为“体内实验配液计算器”的使用方法举例，并不是具体某个化合物的推荐配制方式，请根据您的实验动物和给药方式选择适当的溶解方案。
剂量转换
对于不同动物的给药剂量换算，您也可以参考 更多
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