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ReFRAME 相关化合物库

ReFRAME 相关化合物库

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产品编号 L9230 ReFRAME Related Library
  库化合物信息   Excel SDF

2018年Jeff Janes 等人通过数据挖掘和文献查询,构建了ReFRAME 化合物库,在美国国家科学院院刊(PNAS)发表了关于ReFRAME 化合物库的应用和实用性;其中大部分已通过I 期临床研究具有临床安全性,ReFRAME 化合物库临床安全的独特性质将显著缩短候选药物进入临床的时间,降低失败风险,可高效应用于早期药物研发阶段的筛选以及先导化合物的发现。作者分享了ReFRAME 化合物库,旨在促进数据共享和药物发现机会。盖茨基金会和清华大学等创办的全球健康药物研发中心(GHDDI)也将ReFRAME 化合物库应用于抗COVID-19药物研发。

TargetMol 整理了ReFRAME 化合物库包含3274 种化合物,是药物再利用和抗COVID-19药物研发的有效工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 3274化合物的独特集合,可用于高通量筛选和高内涵筛选,是药物再利用和抗COVID-19药物研发的有效工具
  • 部分化合物已上市得到FDA、EMA、NMPA等权威部门审批,大部分已通过I期临床研究;
  • 通过结构多样性聚类分析,具有优良的结构多样性,包含2698个聚类簇(相似程度大于70%的为一簇),平均1.2个化合物一个簇;
  • 涵盖多个研究领域:肿瘤、心血管药物、抗炎/免疫、神经系统药物、呼吸系统药物等;
  • 靶点多样,包括5-HT Receptor、Sodium Channel、p38 MAPK、PI3K、MEK等;
  • 详细的说明书,化合物结构、靶点信息、适应症信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

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包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L9230)
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化合物库组成

Autophagy (338)
Apoptosis (322)
Antibacterial (254)
Antibiotic (224)
Endogenous Metabolite (197)
5-HT Receptor (129)
COX (116)
Dopamine Receptor (96)
Parasite (92)
Adrenergic Receptor (90)
HIV Protease (78)
AChR (72)
DNA/RNA Synthesis (72)
Antifungal (68)
Histamine Receptor (66)
Calcium Channel (64)
PDE (61)
Potassium Channel (61)
PI3K (58)
VEGFR (57)
Sodium Channel (54)
P450 (50)
Estrogen/progestogen Receptor (46)
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Estrogen Receptor/ERR (28)
c-Kit (28)
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NF-κB (26)
Mitophagy (25)
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p38 MAPK (24)
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LHRH (1)
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Protease (1)
Prolyl Endopeptidase (PREP) (1)
PKM (1)
PI4K (1)
PERK (1)
PD-1/PD-L1 (1)
PAFR (1)
PAD (1)
P2X Receptor (1)
MALT (1)
OXPHOS (1)
NPC1L1 (1)
NEDD8 (1)
NADPH-oxidase (1)
N-Acetylglucosaminyltransferase (1)
Motilin Receptor (1)
MNK (1)
Melanin-concentrating Hormone Receptor (MCHR) (1)
MAPK (1)
YAP (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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