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PCAF-IN-1是一种高选择性的PCAF(p300/CBP-associated factor)抑制剂,具有潜在的抗肿瘤、抗炎、抗心脏疾病作用。抑制PCAF可以减轻心肌梗死后的心脏重塑,减少M1型巨噬细胞的极化,减轻自身免疫性关节炎。
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PCAF-IN-1是一种高选择性的PCAF(p300/CBP-associated factor)抑制剂,具有潜在的抗肿瘤、抗炎、抗心脏疾病作用。抑制PCAF可以减轻心肌梗死后的心脏重塑,减少M1型巨噬细胞的极化,减轻自身免疫性关节炎。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
2 mg | ¥ 720 | 现货 | |
5 mg | ¥ 1,230 | 现货 | |
10 mg | ¥ 1,820 | 现货 | |
25 mg | ¥ 2,970 | 现货 | |
50 mg | ¥ 4,520 | 现货 | |
100 mg | ¥ 6,430 | 现货 | |
200 mg | ¥ 8,780 | 现货 |
产品描述 | PCAF-IN-1 is a highly selective PCAF (p300/CBP-associated factor) inhibitor with potential anti-tumor, anti-inflammatory, and anti-heart disease effects. Inhibition of PCAF attenuates cardiac remodeling after myocardial infarction, reduces polarization of M1-type macrophages, and attenuates autoimmune arthritis. |
体外活性 | 方法:PCAF-IN-1(10 μM,72 小时)处理肝细胞癌 (HePG-2)、乳腺癌 (MCF-7)、前列腺癌 (PC3) 和结直肠癌 (HCT-116),MTT 测定细胞活力。 结果:PCAF-IN-1对人类癌细胞系具有最强的抗肿瘤活性。[1]。 |
分子量 | 310.74 |
分子式 | C15H11ClN6 |
CAS No. | 2439194-86-0 |
Smiles | ClC=1C=CC(=CC1)C2=NN=C3C=4C=CC=CC4C(=NN)NN23 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
溶解度信息 | DMSO: 0.1 mg/mL (0.32 mM), Sonication and heating are recommended. |
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