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TargetMol | Compound Library

抗癌临床化合物库现货

Anti-Cancer Clinical Compound Library

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产品编号 L2120

尽管在过去的几十年中癌症的研究和治疗取得了巨大的成功,但癌症仍然是人类面临的巨大挑战,给患者身心健康带来巨大的痛苦。癌细胞具有许多显著不同的生物学特征,表现出无限的增殖潜能,维持自身生长信号的持续稳定,逃避应激信号(例如治疗药物)诱导的细胞凋亡,刺激血管生长,为肿瘤提供营养,同时逃避免疫系统防御和诱导局部慢性炎症,发挥其侵袭和转移能力,表现出异常的代谢活动,并通过突变和表观遗传机制显著改变全基因组的稳定性。

抗癌活性的药物是临床研究的热点之一,根据文献报道和有关公开资料,我们收集了2680 个具有抗癌活性或潜在抗癌活性的处于临床试验阶段的化合物,组成抗癌临床化合物库,可用于癌症相关研究及高通量高内涵筛选。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L2120

抗癌临床化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2680个具有抗癌活性小分子的独特集合,可用于高通量高内涵筛选;
  • 生物活性已经临床前实验证实,所有化合物均已进入临床实验阶段的抗癌化合物;
  • 包括肺癌、乳腺癌、白血病、淋巴瘤等15种癌症,是癌症相关研究的有效筛选工具;
  • 作用靶点涉及PI3K,HDAC, mTOR, CDK, JAK 等癌症相关靶点;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Apoptosis
Autophagy
Endogenous Metabolite
5-HT Receptor
Antibacterial
Adrenergic Receptor
DNA/RNA Synthesis
Dopamine Receptor
Antibiotic
VEGFR
COX
Histamine Receptor
Potassium Channel
Calcium Channel
EGFR
Sodium Channel
Parasite
PI3K
Cytochromes P450
CDK
Reactive Oxygen Species
FLT
HIV Protease
Glucocorticoid Receptor
Topoisomerase
PDGFR
JAK
FGFR
c-Kit
NF-κB
HDAC
c-Met/HGFR
mTOR
Microtubule Associated
PPAR
Virus Protease
Ferroptosis
AChR
Prostaglandin Receptor
SARS-CoV
Src
Dehydrogenase
Nucleoside Antimetabolite/Analog
Mitophagy
Akt
GABA Receptor
Tyrosine Kinases
Antifungal
Bcr-Abl
Estrogen Receptor/ERR
Estrogen/progestogen Receptor
iGluR
Influenza Virus
GPCR
Adenosine Receptor
Raf
Androgen Receptor
p38 MAPK
PARP
HSP
Caspase
Epigenetic Reader Domain
Bcl-2 Family
Ras
PDE
Interleukin
ERK
HSV
Aurora Kinase
TNF
Serotonin Transporter
P-gp
ALK
TRP/TRPV Channel
MEK
HIF/HIF Prolyl-Hydroxylase
HER
ATPase
c-RET
HBV
PKC
ROS
Opioid Receptor
c-Fms
MDM-2/p53
RAAS
Phosphatase
NMDAR
Norepinephrine
Trk receptor
Histone Methyltransferase
HCV Protease
DNA Alkylator/Crosslinker
Endothelin Receptor
STAT
Proton pump
E1/E2/E3 Enzyme
Mitochondrial Metabolism
MMP
AMPK
TAM Receptor
ROS Kinase
LPL Receptor
GSK-3
Chk
Retinoid Receptor
FAK
Progesterone Receptor
Gamma-secretase
Guanylate cyclase
CXCR
IGF-1R
SGLT
Reverse Transcriptase
HIF
p53
S1P Receptor
Carbonic Anhydrase
DNA-PK
JNK
Molecular Glues
DNA Alkylation
IL Receptor
TLR
Beta Amyloid
CFTR
Proteasome
Antioxidant
PKA
Antifolate
ROCK
Drug Metabolite
P2X Receptor
Vasopressin Receptor
GluR
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Nrf2
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ADC Cytotoxin
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GNRH Receptor
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PLK
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DHFR
P2Y Receptor
CSF-1R
IAP
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Lipoxygenase
Anti-infection
Kinesin
Monoamine Oxidase
NO Synthase
Mdm2
Integrin
MRP
MAO
IDO
BTK
Antifection
OX Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Sirtuin
Casein Kinase
IκB/IKK
Ligand for E3 Ligase
Cannabinoid Receptor
Neurokinin receptor
DNA Methyltransferase
Histone Demethylase
Serine Protease
Leukotriene Receptor
RIP kinase
Smo
PAK
Angiotensin-converting Enzyme (ACE)
DNA
Antiviral
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Sigma receptor
Tie-2
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FXR
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PERK
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MT Receptor
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transporter
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FKBP
ribosome
Melanocortin Receptor
PDK
Oxytocin Receptor
Adenosine Deaminase
Cuproptosis
Discoidin Domain Receptor (DDR)
NOD
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Protease-activated Receptor
NEDD8
Amino Acids and Derivatives
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Arginase
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TOPK
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Galectin
Cysteine Protease
IRE1
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LDL
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Hexokinase
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Thrombopoietin Receptor
OXPHOS
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Acyltransferase
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LPA Receptor
SGK
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p97
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Thyroid hormone receptor(THR)
Advanced Glycation End Products
MicroRNA
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NPC1L1
Hydrogenase
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MALT
Factor VIIa
DYRK
Necroptosis
MIF
GTPase
Factor Xa
OCT
Kisspeptin
N-Acetylglucosaminyltransferase
Hck
Liver X Receptor
Neurotensin Receptor
LIM Kinase
Glucokinase
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Myosin
PAFR
MTH1
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GlyT
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Thioredoxin
ACK1
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PI4K
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RXFP receptor
NADPH-oxidase
BMI-1
Imidazoline Receptor
Vitamin
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