规格

价格

库存

数量

1 mg

¥ 395

现货

5 mg

¥ 976

现货

10 mg

¥ 1,590

现货

25 mg

¥ 2,970

现货

50 mg

¥ 4,690

现货

100 mg

¥ 6,570

现货

200 mg

¥ 8,860

待询

1 mL x 10 mM (in DMSO)

¥ 912

现货

生物活性

产品描述	Saclofen is a sulfonic analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that acts as a competitive antagonist of the GABAB receptor (IC50: 7.8 μM).1 This compound can be used to determine the functional roles for the GABAB receptor as a mediator of slow inhibitory postsynaptic potentials in the brain.
靶点活性	GABAB:7.8 μM
体内活性	CCT241736 显著抑制了体内 MV4-11 人源 FLT3-ITD 阳性 AML 肿瘤异种移植物的生长，其生物标志物的调节和自由化合物暴露与双重 FLT3 和 Aurora 激酶目标的抑制一致。

化学信息

储存&溶解度

存储

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

溶解度信息

DMSO: 5.5 mg/mL (22.03 mM), Sonication is recommended.

溶液配制表

DMSO