- 全部删除
您的购物车当前为空
SKF38393 hydrobromide是SKF38393的盐形式。SKF38393是多巴胺D1受体激动剂,能够增加小鼠NAc中Shati/Nat8L mRNA的表达,在星形胶质细胞中增加了5-羟色胺和n -甲基- D -天冬氨酸诱导的运动相关破裂的频率;可以模拟多巴胺导致小鼠结肠运动的抑制;可促进蝗虫群居化

SKF38393 hydrobromide是SKF38393的盐形式。SKF38393是多巴胺D1受体激动剂,能够增加小鼠NAc中Shati/Nat8L mRNA的表达,在星形胶质细胞中增加了5-羟色胺和n -甲基- D -天冬氨酸诱导的运动相关破裂的频率;可以模拟多巴胺导致小鼠结肠运动的抑制;可促进蝗虫群居化
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 1 mg | ¥ 268 | In stock | |
| 5 mg | ¥ 615 | In stock | |
| 10 mg | ¥ 897 | In stock | |
| 25 mg | ¥ 1,864 | In stock | |
| 50 mg | ¥ 2,720 | In stock | |
| 100 mg | ¥ 3,980 | In stock | |
| 200 mg | ¥ 5,680 | In stock |
SKF38393 hydrobromide 相关产品
| 产品描述 | SKF38393 hydrobromide is the salt form of SKF38393.SKF38393 is a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice; increases the frequency of 5-hydroxytryptamine and n -methyl- D -aspartate-induced locomotion-associated ruptures in astrocytes; can mimic the dopamine-induced inhibition of colonic motility in mice; can promote locust swarming |
| 靶点活性 | D1 receptor:110 nM |
| 体外活性 | 方法:SKF38393 hydrobromide(0.001-10μM,48小时)处理MCF-7、MDA-MB231 和 MCF-10细胞,并通过 Alamar 蓝色染料试剂法测定细胞生长。分析光密度数据并确定 IC50 值。 |
| 体内活性 | 方法:为了评估多巴胺受体亚型在可卡因行为致敏启动中的作用,部分 D1 激动剂 SKF38393 hydrobromide (0.01-1.0 μg/侧)、D2/3 激动剂喹吡罗 (0.1-1.0 μg/侧) 或生理盐水在 3 天内每天一次输注到腹侧被盖区 (VTA) 或伏隔核壳中。 |
| 别名 | SKF 38393 hydrobromide |
| 分子量 | 336.22 |
| 分子式 | C16H18BrNO2 |
| CAS No. | 20012-10-6 |
| Smiles | Br.OC=1C=C2C(=CC1O)C(C=3C=CC=CC3)CNCC2 |
| 密度 | no data available |
| 存储 | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||||||||||||
| 溶解度信息 | H2O: 10 mg/mL (29.74 mM), Sonication is recommended. | |||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||
H2O
| ||||||||||||||||||||||||||
评论内容