Amelubant

Name: Amelubant
Brand: TargetMol
SKU: T14210
Rating: 4.5 (1 reviews)

还可以

产品编号 T14210Cas号 346735-24-8

别名 BIIL 284

Amelubant (BIIL 284) is a prodrug of active metabolites BIIL 260 and BIIL 315 with anti-inflammatory activity[1]. It is a potent, oral, long-acting LTB4 receptor antagonist that negligibly binds to the LTB4 receptor, exhibiting Kis of 221 nM and 230 nM in vital cells and membranes.

Amelubant

还可以

产品编号 T14210 别名 BIIL 284Cas号 346735-24-8

规格	价格	库存	数量
2 mg	¥ 3,420	5日内发货

大包装 & 定制

加入购物车

TargetMol 的所有产品仅用作科学研究或药证申报，不能被用于人体，我们不向个人提供产品和服务。请您遵守承诺用途，不得违反法律法规规定用于任何其他用途。

实验操作小课堂

常见问题解答

Amelubant 相关产品

产品介绍

生物活性

产品描述	Amelubant (BIIL 284) is a prodrug of active metabolites BIIL 260 and BIIL 315 with anti-inflammatory activity[1]. It is a potent, oral, long-acting LTB4 receptor antagonist that negligibly binds to the LTB4 receptor, exhibiting Kis of 221 nM and 230 nM in vital cells and membranes.
靶点活性	LTB4:221 nM （ki）（ in vital human granulocytes), LTB4:230 nM （ki）（ in cell membranes)
体外活性	Amelubant is a prodrug of active metabolites BIIL 260 and BIIL 315, which are reversible and competitive LTB4 receptor antagonists with Kis of 1.4 and 1.1 nM in cells, and 1.7 and 1.9 nM in membranes, respectively [1].
别名	BIIL 284