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抗寄生虫天然产物库

抗寄生虫天然产物库

产品编号 L6620 Antiparasitic Natural Product Library
  库化合物信息   Excel SDF

生活在宿主生物体身上或之内,并从宿主生物体获取食物或以宿主生物体为代价获取食物的生物体,被称为寄生虫。在世界范围内,特别是在热带和亚热带地区,寄生虫所引起的疾病一直是普遍存在的重大公共卫生问题。按照致病的虫种分类,人体寄生虫病主要可以分为原虫病、蠕虫病和节肢动物传播疾病。

天然产物长期以来一直被用于治疗各种寄生虫病,如巴贝西虫病、利什曼病、疟疾、锥虫病等等,并且对非靶标生物毒性低,是抗寄生虫药物先导化合物的重要来源。2015年度诺贝尔生理学颁给从青蒿植物中创造性的研究出抗疟新药的屠呦呦和从高效链霉菌中分离提取得到阿维菌素的大村智和威廉坎贝尔,以表彰他们在寄生虫病治疗研究方面做出的杰出贡献。

TargetMol 抗寄生虫天然产物库,精心整理收录了 253 个具有抗寄生虫活性的天然产物,可用于抗寄生虫新药研发和新靶点验证的多个领域。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 精心挑选253种具有抗寄生虫活性的天然产物,是抗寄生虫药物研发的有力工具;
  • 包含多种抗寄生虫活性天然产物,如抗疟原虫、抗利什曼原虫、抗丝虫病等;
  • 结构多样,包含萜类、生物碱、多酚等类别;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L6620)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Parasite (92)
Apoptosis (56)
Antibacterial (51)
Autophagy (40)
Antibiotic (33)
Endogenous Metabolite (30)
Antifungal (22)
NF-κB (16)
Reactive Oxygen Species (12)
AChR (10)
Ferroptosis (10)
Antifection (10)
Topoisomerase (9)
COX (9)
DNA/RNA Synthesis (8)
HIV Protease (8)
Influenza Virus (8)
p38 MAPK (8)
Caspase (6)
Antioxidant (6)
Potassium Channel (6)
AChE (6)
Anti-infection (5)
Sodium Channel (5)
PKC (5)
Calcium Channel (5)
IL Receptor (5)
Microtubule Associated (5)
TNF (4)
P450 (4)
SARS-CoV (4)
EGFR (4)
Akt (4)
PARP (4)
Mitochondrial Metabolism (4)
ATPase (4)
ribosome (4)
Virus Protease (4)
ROS (4)
Mitophagy (4)
JNK (4)
5-HT Receptor (4)
HSV (3)
Glucosidase (3)
BCL (3)
Dehydrogenase (3)
ERK (3)
GABA Receptor (3)
Nrf2 (3)
Phospholipase (3)
AMPK (3)
Beta Amyloid (3)
P-gp (2)
STAT (2)
GluR (2)
MMP (2)
Antiviral (2)
Lipoxygenase (2)
FAK (2)
Tyrosinase (2)
TGF-beta/Smad (2)
TLR (2)
HSP (2)
p53 (2)
Phosphatase (2)
MAO (2)
NOS (2)
Histamine Receptor (2)
Immunology/Inflammation related (2)
Estrogen Receptor/ERR (2)
HBV (2)
Dopamine Receptor (2)
VEGFR (2)
UGT (2)
TRP/TRPV Channel (2)
Estrogen/progestogen Receptor (2)
PI3K (2)
Gamma-secretase (2)
PKA (2)
ABC (1)
Fatty Acid Synthase (1)
HDAC (1)
PPAR (1)
IκB/IKK (1)
MRP (1)
Lipase (1)
Factor Xa (1)
Casein Kinase (1)
MEK (1)
NADPH (1)
DYRK (1)
Platelet aggregation (1)
Syk (1)
HCV Protease (1)
NOD (1)
Hydrogenase (1)
Transferase (1)
Carbonic Anhydrase (1)
HIF/HIF Prolyl-Hydroxylase (1)
Wnt/beta-catenin (1)
transporter (1)
RSV (1)
Androgen Receptor (1)
Opioid Receptor (1)
Monoamine Transporter (1)
CCR (1)
CXCR (1)
DNA gyrase (1)
Xanthine Oxidase (1)
Aurora Kinase (1)
NMDAR (1)
cAMP (1)
Drug Metabolite (1)
Epigenetic Reader Domain (1)
CaMK (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
GluCls (1)
mTOR (1)
MTH1 (1)
PAFR (1)
PDE (1)
IAP (1)
iGluR (1)
Adrenergic Receptor (1)
Prostaglandin Receptor (1)
Serine/threonin kinase (1)
Aminopeptidase (1)
Histone Acetyltransferase (1)
Chloride channel (1)
Serotonin Transporter (1)
Hedgehog/Smoothened (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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