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Jingzhaotoxin-XII (JzTx-XII) TFA,具有特异性地抑制Kv4.1通道的活性,其半抑制浓度(IC50)为0.363 μM。该化合物通过改变通道的门控行为来发挥作用。
Jingzhaotoxin-XII (JzTx-XII) TFA,具有特异性地抑制Kv4.1通道的活性,其半抑制浓度(IC50)为0.363 μM。该化合物通过改变通道的门控行为来发挥作用。
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 10 mg | 待询 | 待询 | |
| 50 mg | 待询 | 待询 |
Jingzhaotoxin-XII TFA 相关产品
| 产品描述 | Jingzhaotoxin-XII (JzTx-XII) TFA is a specific inhibitor of the Kv4.1 channel, exhibiting an IC50 of 0.363 μM. It interacts with the channel by altering gating behavior. |
| 别名 | JzTx-XII TFA |
| Sequence | Tyr-Cys-Gln-Lys-Trp-Met-Trp-Thr-Cys-Asp-Ser-Glu-Arg-Lys-Cys-Cys-Glu-Gly-Tyr-Val-Cys-Glu-Leu-Trp-Cys-Lys-Tyr-Asn-Leu-NH2 (Disulfide bridge: Cys2-Cys16,Cys9-Cys21,Cys15-Cys25) |
| Sequence Short | YCQKWMWTCDSERKCCEGYVCELWCKYNL-NH2 (Disulfide bridge: Cys2-Cys16,Cys9-Cys21,Cys15-Cys25) |
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
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