GSK2798745

Name: GSK2798745
Brand: TargetMol
SKU: T15434
Rating: 4.5 (1 reviews)

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产品编号 T15434Cas号 1419609-94-1

GSK2798745 is an orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker (IC50s: 1.8 and 1.6 nM for hTRPV4 and rTRPV4). It is used in research for the treatment of pulmonary edema associated with congestive heart failure.

GSK2798745

还可以

产品编号 T15434Cas号 1419609-94-1

规格	价格	库存
25 mg	¥ 17,200	3-6月
50 mg	¥ 22,800	3-6月
100 mg	¥ 29,500	3-6月

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TargetMol 的所有产品仅用作科学研究或药证申报，不能被用于人体，我们不向个人提供产品和服务。请您遵守承诺用途，不得违反法律法规规定用于任何其他用途。

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GSK2798745 相关产品

产品介绍

生物活性

产品描述	GSK2798745 is an orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker (IC50s: 1.8 and 1.6 nM for hTRPV4 and rTRPV4). It is used in research for the treatment of pulmonary edema associated with congestive heart failure.
靶点活性	TRPV4 (rat):1.6 nM, TRPV4 (human):1.8 nM

化学信息

分子量	460.53
分子式	C₂₅H₂₈N₆O₃
CAS No.	1419609-94-1
密度	1.35 g/cm3 (Predicted)

储存&溶解度

存储

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

溶解度信息

DMSO: 250 mg/mL (542.85 mM), Sonication is recommended.

溶液配制表

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.1714 mL	10.8571 mL	21.7141 mL	108.5706 mL
5 mM	0.4343 mL	2.1714 mL	4.3428 mL	21.7141 mL
10 mM	0.2171 mL	1.0857 mL	2.1714 mL	10.8571 mL
20 mM	0.1086 mL	0.5429 mL	1.0857 mL	5.4285 mL
50 mM	0.0434 mL	0.2171 mL	0.4343 mL	2.1714 mL
100 mM	0.0217 mL	0.1086 mL	0.2171 mL	1.0857 mL