购物车
  • TargetMol
    您的购物车当前为空
TargetMol | Compound Library

抗癌活性化合物库现货

Anti-Cancer Active Compound Library
Rating icon 很棒
货号 L2160

尽管在过去的几十年中癌症的研究和治疗取得了巨大的成功,但癌症仍然是人类面临的巨大挑战,给患者身心健康带来巨大的痛苦。癌细胞具有许多显著不同的生物学特征,表现出无限的增殖潜能,维持自身生长信号的持续稳定,逃避应激信号诱导的细胞凋亡,刺激血管生长,为肿瘤提供营养,同时逃避免疫系统防御和诱导局部慢性炎症,发挥其侵袭和转移能力;并且表现出异常的代谢活动,并通过突变和表观遗传机制显著改变全基因组的稳定性。

根据文献报道和有关公开资料,我们挑选了 4270 个具有已知抗癌活性的化合物组成抗癌活性库,可用于具体癌症的阳性对照及癌症机理的研究。希望我们在抗癌研究的路上,助您一臂之力!

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
资源下载
化合物库相关信息
Excel
SDF
联系我们获取更多批次信息

货号 L2160

抗癌活性化合物库

规格

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 4270种具有抗肿瘤活性的化合物的特有集合,用于高通量、高内涵筛选;
  • 是肿瘤发生机理研究、抗肿瘤药物筛选的有效工具;
  • 靶点含PI3K、HDAC、mTOR、CDK、Aurora Kinase、JAK等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS检测技术保证产品高纯度和高质量,减少假阳性发生概率。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

使用TargetMol产品
发表顶级期刊文献

引用更多关于TargetMol产品的科学文献吧!

查看更多

Library Customization | TargetMol 化合物库定制

Compound Library | TargetMol
您可以通过点击按钮
定制您专属的化合物!
联系专属定制

Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
Antibacterial
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
PI3K
EGFR
ROS
Ras
VEGFR
Akt
Antibiotic
Microtubule Associated
Parasite
mTOR
Topoisomerase
Epigenetic Reader Domain
Antifungal
Caspase
Reactive Oxygen Species
ERK
Bcl-2 Family
FLT
Dehydrogenase
STAT
Nucleoside Antimetabolite/Analog
COX
PDGFR
PARP
HDAC
Histone Methyltransferase
p38 MAPK
FGFR
Estrogen Receptor/ERR
c-Met/HGFR
TNF
Wnt/beta-catenin
HIV Protease
Cytochromes P450
c-Kit
Ferroptosis
Interleukin
JAK
Raf
MDM-2/p53
Src
Phosphatase
HSP
MMP
Antioxidant
Virus Protease
Influenza Virus
Estrogen/progestogen Receptor
Kras
PKC
Bcr-Abl
AMPK
NO Synthase
ALK
Aurora Kinase
Androgen Receptor
PPAR
JNK
Calcium Channel
E1/E2/E3 Enzyme
Nrf2
SARS-CoV
MEK
P-gp
FAK
DUB
HIF/HIF Prolyl-Hydroxylase
GSK-3
IL Receptor
TLR
PROTACs
MAPK
p53
HSV
IGF-1R
Mitophagy
TGF-beta/Smad
AChR
Antiviral
DNA Alkylator/Crosslinker
Drug Metabolite
Mitochondrial Metabolism
c-RET
Chk
Histone Demethylase
PDE
ATM/ATR
Sirtuin
Gamma-secretase
Potassium Channel
Proteasome
TAM Receptor
Lipoxygenase
Tyrosine Kinases
HER
Trk receptor
c-Fms
DNA-PK
Pim
Adrenergic Receptor
Molecular Glues
Histone Acetyltransferase
Sodium Channel
Cholinesterase (ChE)
5-HT Receptor
S6 Kinase
Mdm2
PERK
Casein Kinase
Retinoid Receptor
Hedgehog/Smoothened
Transferase
HIF
ROS Kinase
PLK
Integrin
Reductase
Smo
DNA Methyltransferase
GABA Receptor
PD-1/PD-L1
ADC Cytotoxin
Kinesin
Serine Protease
Anti-infection
IAP
Fatty Acid Synthase
Histamine Receptor
YAP
HBV
Aryl Hydrocarbon Receptor
CXCR
PKA
DNA Alkylation
TRP/TRPV Channel
HCV Protease
Glutathione Peroxidase
Tyrosinase
LPL Receptor
Antifolate
Phospholipase
Beta Amyloid
PDK
Dopamine Receptor
Antifection
Ligands for E3 Ligase
Indoleamine 2,3-Dioxygenase (IDO)
S1P Receptor
IDO
c-Myc
Isocitrate Dehydrogenase (IDH)
BTK
IκB/IKK
transporter
GPCR
Carbonic Anhydrase
DNA
Serine/threonin kinase
DHFR
CSF-1R
MAO
Aromatase
Prostaglandin Receptor
IKZF
Immunology/Inflammation related
Syk
ROCK
CaMK
Adenosine Receptor
DYRK
Rho
ATPase
NOS
OXPHOS
Glutaminase
Survivin
Cell Cycle Arrest
NADPH
AhR
Monoamine Oxidase
glycosidase
Monocarboxylate transporter
RIP kinase
BCRP
Glucosidase
IFNAR
Telomerase
Progesterone Receptor
Photosensitizer
Ephrin Receptor
Reverse Transcriptase
NOD
Cysteine Protease
STING
Wee1
Methionine Adenosyltransferase (MAT)
Amino Acids and Derivatives
MNK
Tie-2
Cholecystokinin Receptor
Acyltransferase
RANKL/RANK
Glucocorticoid Receptor
NOD-like Receptor (NLR)
GNRH Receptor
PAK
PAI-1
IRAK
iGluR
CCR
Proton pump
Opioid Receptor
GPX
P2X Receptor
Somatostatin
Discoidin Domain Receptor (DDR)
MicroRNA
RAAS
Bcl-6
NAMPT
ABC Transporter
Chloride channel
IRE1
Cannabinoid Receptor
PYK2
UGT
Aminopeptidase
HMG-CoA Reductase
p97
ROR
Ligands for Target Protein for PROTAC
Glucokinase
Angiotensin-converting Enzyme (ACE)
Orphan Receptor
Endothelin Receptor
Necroptosis
Lipid
PSMA
LPA Receptor
BMI-1
Thrombin
Liver X Receptor
ATG
GluR
Leukotriene Receptor
Pyroptosis
PKM
FOXO
DAPK
Galectin
MTH1
NMDAR
Hexokinase
Complement System
Myosin
Neurokinin receptor
GTPase
cAMP
MELK
GST
FAAH
p62
Hydroxylase
MALT
PTEN
CRM1
MRP
PAD
ASK
Protease-activated Receptor
Lipase
KLF
TOPK
Serotonin Transporter
Decarboxylase
Adenosine Deaminase
APC/C
GRK
Bombesin Receptor
ACK1
SGK
Factor Xa
Platelet aggregation
NEDD8
LTR
NR4A
Porcupine
CD73
ribosome
CRISPR/Cas9
MyD88
Arrestin
FXR
Xanthine Oxidase
KSP
Cadherin
MLK
MIF
Neurotensin Receptor
Adenylate cyclase
Thrombopoietin Receptor
Cuproptosis
PAFR
Haspin Kinase
GPCR19
RSV
Drug-Linker Conjugates for ADC
Protease
PI4K
Thyroid hormone receptor(THR)
FLAP
Beta-Secretase
Hck
Annexin A
Arp2/3 Complex
Stearoyl-CoA Desaturase (SCD)
HuR
FOXO3
CaSR
Gap Junction Protein
Lysosomal Autophagy
Factor VIIa
Vitamin
Adiponectin Receptor
ATP Citrate Lyase
E3 Ligase Ligand-Linker Conjugates
Hippo pathway
Sigma receptor
CFTR
RAR/RXR
DNA gyrase
Acetyl-CoA Carboxylase
FKBP
PARG(Poly(ADP-ribose) Glycohydrolase)
GlyT
PGE Synthase
Urea Transporter
Aquaporin
Apelin receptor
CYP19A1
Dynamin
P2Y Receptor
B7
DPP-4
HCAR
NEDD4-1
Tight Junction Protein
NPC1L1
Kisspeptin
LDLR
SIK
Thioredoxin
Glutathione reductase
Liposome
Advanced Glycation End Products
NUDIX hydrolase
BACE
OCT
Stemness kinase
Na-K-Cl cotransporter
Neuropeptide Y Receptor
SGLT
TMV
CAT
Y Box Binding Protein 1
Arginase
Na+/Ca2+ Exchanger
gp120/CD4
Vasopressin Receptor
Carboxypeptidase
Melanocortin Receptor
Oxytocin Receptor
GHSR
CD38
VDA
Target Protein Ligand-Linker Conjugates
LAG-3
PROTAC Linker
Transketolase
Melatonin Receptor
Amylase
Prolyl Endopeptidase (PREP)
FABP
LDL
Epoxide Hydrolase
LRRK2
Free radical scavengers
GluCls
RXFP receptor
NADPH-oxidase
Glyoxalase
Poly(ADP-ribose) Glycohydrolase (PARG)
Ferroportin
ADC Linker

Keywords