您的购物车当前为空
NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)

NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 25 mg | ¥ 10,600 | 6-8周 | |
| 50 mg | ¥ 13,800 | 6-8周 | |
| 100 mg | ¥ 17,500 | 6-8周 |
NRA-0160 相关产品
| 产品描述 | NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM) |
| 靶点活性 | α1-adrenoceptor (rat):237 nM (ki), D3 receptor:39 nM (ki), 5-HT2A receptor:180 nM (Ki, in rat), D4 receptor:0.48 nM (ki) |
| 体内活性 | NRA0160 dose-dependently and significantly reverses the effects of MAP on both A9 and Al0 dopamine neurons.?NRA0160 is slightly more potent in reversiig the effects of MAP on A10 (ED50 = 1.0 mg/kg) than on A9 dopamine neurons (ED50 = 1.3 mg/kg).?NRA0160 reverses the effect of AP0 on both A9 and A10 dopamine neurons.?ED50 values for the effects of NRA0160 on APO-induced inhibition of A9 and A10 dopamine neurons are 1.3 mg/kg and 0.5 mg/kg, respectively[2]. |
| 分子量 | 439.52 |
| 分子式 | C24H23F2N3OS |
| CAS No. | 204718-47-8 |
| 密度 | 1.297 g/cm3 (Predicted) |
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
评论内容