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Chromatin Modification Compound Library
染色质化学修饰是指对染色质的组成成分进行化学基团的添加或去除的反应过程,常见的染色质化学修饰方式有:甲基化-去甲基化、乙酰化-去乙酰化、磷酸化-去磷酸化,此外,还包括泛素化、ADP-核糖基化和二硫键形成等修饰方式。染色质中的组蛋白和DNA 是主要的化学修饰底物。目前,已在细胞中发现了一系列的染色质修饰酶类,这些酶不仅具有高度的位点特异性,而且对底物原有的修饰状态也有选择性。由于染色质化学修饰而导致某些基因沉默或异常表达,从而引起个体表型的改变,称为表型遗传修饰。 TargetMol 作为全球知名化合物库供应商,积极关注科研动态,为您提供大量染色质修饰相关的优质产品,致力于提供药物筛选领域的全流程的一站式服务。
Empty | 1477949-42-0 | 1815580-06-3 | 1450655-76-1 | 1628317-18-9 | 1857417-10-7 | 86361-55-9 | 937039-45-7 | 1346574-57-9 | 1206731-57-8 | 1913252-04-6 | Empty |
SantacruzaMate A | SKLB-23bb | CPI-169 racemate | MI-463 | MI-538 | Gnetol | Pimelic diphenylamide 106 | GSK126 | WT-161 | JQEZ5 | ||
Empty | 10356-76-0 | 1403254-99-8 | 149647-78-9 | 499-80-9 | 1628332-52-4 | 1872466-47-1 | 1857417-13-0 | 2361659-61-0 | 2463198-51-6 | 315698-07-8 | Empty |
5-Fluoro-2'-deoxycytidine | Tazemetostat | Vorinostat | lutidinic acid | GSK467 | CM-675 | MI-503 | AES-135 | HDAC-IN-40 | BRD 4354 | ||
Empty | 2098902-68-0 | 501-36-0 | 1423715-09-6 | 852475-26-4 | 1271738-62-5 | 946150-57-8 | 1883429-21-7 | 3565-26-2 | 1187075-34-8 | 1271738-59-0 | Empty |
KDM4D-IN-1 | Resveratrol | SP2509 | MC1568 | Menin-MLL inhibitor MI-2 | Remetinostat | BI-7273 | NSC 3852 | Resminostat hydrochloride | MI-3 | ||
Empty | 1001645-58-4 | 1093403-33-8 | 838-07-3 | 2196203-96-8 | 1259296-46-2 | 2102933-95-7 | 1620401-82-2 | 1396772-26-1 | 1146963-51-0 | 1357302-64-7 | Empty |
SRT1720 hydrochloride | SRT 2104 | 5-Methyl-2'-deoxycytidine | TH34 | MPI_5a | GSK-LSD1 dihydrochloride | UNC0379 | EPZ005687 | J-147 | OG-L002 | ||
Empty | 796-42-9 | 1403764-72-6 | 887686-02-4 | 849234-64-6 | 1271022-90-2 | 1314241-44-5 | 1105698-15-4 | 1869912-40-2 | 1636894-46-6 | 1431326-61-2 | Empty |
AS8351 | PFI-1 | OSS_128167 | BRD-6929 | BMS-911543 | UNC 669 | Salermide | AZD5153 6-Hydroxy-2-naphthoic acid | KA2507 | ORY1001 | ||
Empty | 1624117-53-8 | 1817802-18-8 | 1619994-68-1 | 199657-29-9 | 96017-59-3 | 1818-71-9 | 1184136-10-4 | 99873-43-5 | 440662-09-9 | 2126744-35-0 | Empty |
XY1 | MPT0B390 | GSK2801 | Givinostat hydrochloride | 2-hexyl-4-Pentynoic Acid | Crotonoside | UNC926 | Droxinostat | CeMMEC1 | SW-100 | ||
Empty | 1300031-52-0 | 2196-14-7 | 743420-02-2 | 1821-12-1 | 89412-79-3 | 1550053-02-5 | 1609389-52-7 | 1415800-43-9 | 652-37-9 | 1320288-17-2 | Empty |
GSK1324726A | 7,4'-Dihydroxyflavone | HDAC-IN-7 | 4-Phenylbutyric acid | Raddeanin A | BRD3308 | ACY-957 | UNC1215 | Acefylline | UNC0646 | ||
Empty | 1320288-19-4 | 1346572-63-1 | 537672-41-6 | 1619994-69-2 | 1260907-17-2 | 537034-17-6 | 535-96-6 | 1012054-59-9 | 2514-30-9 | 1252003-15-8 | Empty |
UNC 0631 | GSK503 | UF010 | Bromosporine | Molibresib | BML-210 | Marein | CUDC-101 | PBIT | Tubastatin A |