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TargetMol | Compound Library

DNA 损伤和修复分子库现货

DNA Damage & Repair Compound Library

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货号 L3900

癌细胞的耐药性是癌症治疗过程中面临的主要挑战,因此鉴定新的生物学靶标,并开发设计相应的药物成为重要策略,在各种潜在候选靶标中,癌细胞 DNA Damage & Repair 系统是重要的靶标。由于抗生素的滥用,细菌等微生物的耐药性越来越强,开发靶向微生物 DNA Damage & Repair 系统的药物迫在眉睫。

TargetMol DNA 损伤和修复分子库是1440 个与DNA 损伤和修复紧密相关的化合物集合,可用于DNA 损伤和修复相关研究的高通量筛选,高内涵筛选。

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货号 L3900

DNA 损伤和修复分子库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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产品描述

  • 1440个与DNA损伤和修复紧密相关的化合物集合,是高通量筛选,高内涵筛选的良好载体;
  • 涵盖与DNA损伤和修复相关的热门靶点,如HDAC、DNA/RNA Synthesis、Topoisomerase等;
  • 通过临床前研究和临床实验,生物活性和生物安全性得到保障;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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DNA/RNA Synthesis
Apoptosis
PPAR
HDAC
Nucleoside Antimetabolite/Analog
PARP
Topoisomerase
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Endogenous Metabolite
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