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TargetMol | Compound Library

疼痛相关化合物库现货

Pain-Related Compound Library
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货号 L2690

疼痛是一种与实际或潜在的组织损伤相关的不愉快的感觉和情绪情感体验,或与此相似的经历 ;作为六大生命体征之一,疼痛与呼吸、脉搏、血压、体温等同样重要,反映了身体的健康状态。疼痛按持续时间分为急性疼痛、慢性疼痛;按照病因分为伤害性疼痛和神经病理性疼痛;按感受系统分类表层疼痛、深层疼痛;还可根据来源分为内脏痛和体表痛。
疼痛的产生机制是一个复杂的过程,涉及多个层面,包括生理、心理和神经生物学方面,疼痛主要的机制包括:痛觉感受器的激活,痛觉感受器是分布在皮肤、内脏、骨骼肌和关节等部位的专门感知有害刺激的感觉神经末梢。致痛物质的释放:当组织损伤时,会释放多种致痛物质,如组胺、缓激肽、5-羟色胺、乙酰胆碱、前列腺素等,这些物质能激活痛觉感受器。此外还包括神经信号传导、中枢调控、心理因素等等
TargetMol收集了2780种疼痛相关活性化合物及靶向疼痛相关靶点的化合物,可用于疼痛相关研究。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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货号 L2690

疼痛相关化合物库

规格

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2780种疼痛相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
  • 结构多样,具有良好的细胞渗透性;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

5-HT Receptor
COX
Apoptosis
Calcium Channel
Potassium Channel
Histamine Receptor
Autophagy
Sodium Channel
GABA Receptor
Ras
AChR
TRP/TRPV Channel
Endogenous Metabolite
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ERK
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NF-κB
Prostaglandin Receptor
NMDAR
Opioid Receptor
Antibacterial
iGluR
Adrenergic Receptor
Raf
JNK
ROS
Parasite
MAPK
Akt
MEK
NO Synthase
TNF
KRas
Reactive Oxygen Species
Cytochromes P450
Serotonin Transporter
Caspase
S6 Kinase
Interleukin
PPAR
CDK
Lipoxygenase
Endothelin Receptor
Norepinephrine
Neurokinin receptor
Src
Drug Metabolite
Ferroptosis
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VEGFR
Bcl-2 Family
Antibiotic
PI3K
STAT
IL Receptor
Bradykinin Receptor
GluR
DNA/RNA Synthesis
EGFR
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PKC
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PKA
Wnt/beta-catenin
PGE Synthase
Cannabinoid Receptor
Sigma receptor
ATPase
NOS
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GSK-3
MMP
Anti-infection
Rho
PDE
Beta Amyloid
HIV Protease
P2X Receptor
TGF-beta/Smad
AMPK
Mitophagy
Cholinesterase (ChE)
Aurora Kinase
IGF-1R
SARS-CoV
PERK
PARP
Mitochondrial Metabolism
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Phospholipase
MLK
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FAAH
MNK
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FLT
Chloride channel
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IκB/IKK
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RAAS
TOPK
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Gamma-secretase
HSP
c-RET
CGRP Receptor
IRAK
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DYRK
Glutathione Peroxidase
Progesterone Receptor
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ABC Transporter
transporter
ASK
SGK
MDM-2/p53
Syk
LTR
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Lipase
Tie-2
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Immunology/Inflammation related
IAP
Myosin
UGT
LDL
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Antifection
PAK
cAMP
glycosidase
Epigenetic Reader Domain
Antiviral
c-Fms
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FOXO
Platelet aggregation
NOD
HIF/HIF Prolyl-Hydroxylase
PD-1/PD-L1
Transaminase
Amino Acids and Derivatives
Necroptosis
GTPase
Tyrosine Kinases
AAK1
FXR
Aryl Hydrocarbon Receptor
RIP kinase
GlyT
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MAGL
CCR
PTEN
Chk
DNA
Androgen Receptor
Beta-Secretase
Acyltransferase
STING
LRRK2
ALK
KLF
HMG-CoA Reductase
Microtubule Associated
AhR
NOD-like Receptor (NLR)
p53
Proteasome
Taste receptor
Integrin
MyD88
c-Met/HGFR
LPL Receptor
MIF
Melatonin Receptor
OCT
c-Myc
GNRH Receptor
Pim
Cell Cycle Arrest
PYK2
CSF-1R
Adenylate cyclase
GRK
AAK1 (AP2 associated kinase 1)
DNA Alkylation
Stearoyl-CoA Desaturase (SCD)
Angiotensin-converting Enzyme (ACE)
OX Receptor
Epoxide Hydrolase
Lipid
Survivin
GPCR19
Free radical scavengers
Sirtuin
PAI-1
Pyroptosis
RSV
GST
Gap Junction Protein
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NADPH-oxidase
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CFTR
BTK
Melanin-concentrating Hormone Receptor (MCHR)
Apelin receptor
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Monocarboxylate transporter
RAR/RXR
ASBT
Y Box Binding Protein 1
Arrestin
BACE
gp120/CD4
N-Acetylglucosaminyltransferase
CaSR
Cholecystokinin Receptor
ASCT
Antifolate
Nucleoside Antimetabolite/Analog
Cysteine Protease
Liver X Receptor
LIM Kinase
Glucokinase
NR4A
IDO
Prolyl Endopeptidase (PREP)
Annexin A
FLAP
Glucagon Receptor
MT Receptor
DNA gyrase
Na-K-Cl cotransporter
Anion Exchanger
PROTAC Linker
Vasopressin Receptor
ACK1
CXCR
Cadherin
Indoleamine 2,3-Dioxygenase (IDO)
BCRP
OXPHOS
MRGPR
Aminopeptidase
Urea Transporter
Ephrin Receptor
GluCls
HuR
MELK
Hippo pathway
Carboxypeptidase
GPX
Retinoid Receptor
Aromatase
Melanocortin Receptor
PI4K
PDK
RXFP receptor
DAPK
BMI-1
ROS Kinase
Imidazoline Receptor
S1P Receptor
HER
Kinesin
PKM
Sodium-dependent phosphate transporter

Keywords