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TargetMol | Compound Library

抗糖尿病库现货

Anti-Diabetic Compound Library

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产品编号 L1900

糖尿病是一种以高血糖为特征的代谢性疾病,长期的高血糖会导致全身各种组织功能障碍,如果出现并发症,糖尿病会对生活质量产生重大影响,并可能降低预期寿命,目前仍然无法治愈糖尿病,只能通过饮食调节和药物辅助治疗进行病情控制。 TargetMol 抗糖尿病库包含了 800 个糖尿病相关活性化合物,是研究糖尿病的优良工具和药物筛选的极佳载体。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L1900

抗糖尿病库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 800种生物活性小分子化合物;
  • 靶点包括SGLT、PPAR、DPP-4、OC receptor、AMPK等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库定制

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Library Customization | TargetMol 化合物库组成

PPAR
Autophagy
Apoptosis
AMPK
mTOR
NF-κB
Endogenous Metabolite
IGF-1R
JNK
PI3K
Antibacterial
Glucagon Receptor
COX
GSK-3
DPP-4
Akt
SGLT
Potassium Channel
Glucosidase
Proteasome
Antibiotic
CDK
GPCR
STAT
Antioxidant
Ferroptosis
p38 MAPK
Parasite
Phosphatase
TNF
Influenza Virus
Reductase
Sirtuin
Cytochromes P450
DNA-PK
Mitophagy
Dehydrogenase
ERK
Glucokinase
IL Receptor
PDE
Reactive Oxygen Species
Src
transporter
S6 Kinase
Antifungal
MMP
PKC
Prostaglandin Receptor
Adrenergic Receptor
ALK
EGFR
FLT
Lipoxygenase
NO Synthase
Adenosine Receptor
ATM/ATR
Calcium Channel
FGFR
Interleukin
IκB/IKK
TRP/TRPV Channel
VEGFR
Virus Protease
AChR
ATPase
Bcl-2 Family
Beta Amyloid
Cannabinoid Receptor
Caspase
DNA/RNA Synthesis
HDAC
HIF/HIF Prolyl-Hydroxylase
HIV Protease
Mitochondrial Metabolism
Nrf2
p53
ROS
SARS-CoV
Tyrosinase
Wnt/beta-catenin
Aurora Kinase
Cholinesterase (ChE)
c-Met/HGFR
FAK
Glucocorticoid Receptor
HSV
JAK
MEK
NADPH
PDGFR
Sodium Channel
5-HT Receptor
ABC Transporter
Antifection
Casein Kinase
CCR
CETP
Drug Metabolite
Fatty Acid Synthase
GABA Receptor
HIF
Histamine Receptor
MAPK
NADPH-oxidase
NOD
PDK
Phosphorylase
PKA
ROCK
Serine Protease
SIK
Thrombin
Transferase
Trk receptor
Tyrosine Kinases
Androgen Receptor
BACE
Bcr-Abl
Bombesin Receptor
Carbonic Anhydrase
CFTR
Chk
c-RET
DNA
E1/E2/E3 Enzyme
Epigenetic Reader Domain
Epoxide Hydrolase
FXR
Glutathione Peroxidase
HBV
Leukotriene Receptor
Liver X Receptor
MAO
MLK
Norepinephrine
NOS
Opioid Receptor
PARP
PERK
P-gp
Phospholipase
PYK2
Raf
Retinoid Receptor
Stearoyl-CoA Desaturase (SCD)
Syk
Topoisomerase
ACK1
Acyltransferase
Advanced Glycation End Products
Amylase
Annexin A
Anti-infection
Antiviral
Aromatase
Arrestin
Aryl Hydrocarbon Receptor
ATP Citrate Lyase
Beta-Secretase
Bradykinin Receptor
CaMK
CaSR
Cell Cycle Arrest
c-Fms
Chloride channel
c-Kit
CXCR
Cysteine Protease
DNA Alkylation
Dopamine Receptor
DYRK
Estrogen Receptor/ERR
Estrogen/progestogen Receptor
FAAH
FLAP
FOXO1
Free radical scavengers
GluR
GPCR19
GRK
GTPase
Hexokinase
Hippo pathway
Histone Methyltransferase
HMG-CoA Reductase
Immunology/Inflammation related
Integrin
IRAK
LDL
LPL Receptor
LRRK2
LTR
MNK
Monoamine Oxidase
Neurotensin Receptor
NOD-like Receptor (NLR)
NPC1L1
PAI-1
PAK
PI4K
PKM
PROTAC Linker
Proton pump
Pyroptosis
RAAS
Reverse Transcriptase
Rho
S1P Receptor
Serotonin Transporter
SGK
Sigma receptor
Telomerase
TGF-beta/Smad
Tie-2
TLR
YAP
ADC Cytotoxin
IGF-2R
BTK
PGC-1α

Keywords