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TargetMol | Compound Library

抗糖尿病库现货

Anti-Diabetic Compound Library

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产品编号 L1900

糖尿病是一种以高血糖为特征的代谢性疾病,长期的高血糖会导致全身各种组织功能障碍,如果出现并发症,糖尿病会对生活质量产生重大影响,并可能降低预期寿命,目前仍然无法治愈糖尿病,只能通过饮食调节和药物辅助治疗进行病情控制。

TargetMol 抗糖尿病库包含了 800 个糖尿病相关活性化合物,是研究糖尿病的优良工具和药物筛选的极佳载体。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L1900

抗糖尿病库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 800种生物活性小分子化合物;
  • 靶点包括SGLT、PPAR、DPP-4、OC receptor、AMPK等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

PPAR
Autophagy
Apoptosis
AMPK
Endogenous Metabolite
NF-κB
mTOR
Antibacterial
IGF-1R
JNK
PI3K
Proteasome
DPP-4
COX
Akt
GSK-3
Glucagon Receptor
Glucosidase
Antibiotic
Reactive Oxygen Species
SGLT
Potassium Channel
GPCR
Ferroptosis
Parasite
p38 MAPK
Antifungal
STAT
TNF
Antioxidant
Phosphatase
ERK
CDK
Mitophagy
Cytochromes P450
Sirtuin
Dehydrogenase
Reductase
Influenza Virus
DNA-PK
Src
Glucokinase
PDE
transporter
NO Synthase
Caspase
PKC
IL Receptor
S6 Kinase
MMP
DNA/RNA Synthesis
Prostaglandin Receptor
Bcl-2 Family
HIV Protease
Virus Protease
Calcium Channel
TRP/TRPV Channel
Adrenergic Receptor
Mitochondrial Metabolism
Lipoxygenase
EGFR
ALK
IκB/IKK
Beta Amyloid
FLT
ATPase
Adenosine Receptor
Wnt/beta-catenin
VEGFR
ROS
HSV
Nrf2
ATM/ATR
FGFR
AChR
HIF/HIF Prolyl-Hydroxylase
NADPH
Cholinesterase (ChE)
Aurora Kinase
Interleukin
SARS-CoV
HDAC
Cannabinoid Receptor
MDM-2/p53
Tyrosinase
p53
Glucocorticoid Receptor
SIK
Fatty Acid Synthase
PDGFR
Stearoyl-CoA Desaturase (SCD)
Sodium Channel
FAK
Transferase
MTP
c-Met/HGFR
BACE
Histamine Receptor
PKA
Tyrosine Kinases
PARP
Serine Protease
ROCK
Topoisomerase
Drug Metabolite
Phosphorylase
ABC Transporter
Antifection
Opioid Receptor
JAK
CCR
MAPK
Casein Kinase
PDK
GABA Receptor
5-HT Receptor
HIF
MEK
NADPH-oxidase
NOD
Thrombin
Chloride channel
Proton pump
NOS
Carbonic Anhydrase
PERK
Glutathione Peroxidase
c-Myc
HBV
Liver X Receptor
Leukotriene Receptor
FXR
PYK2
Amylase
MAO
E1/E2/E3 Enzyme
Bcr-Abl
Raf
Bombesin Receptor
Chk
Epigenetic Reader Domain
Norepinephrine
DNA
Androgen Receptor
ATP Citrate Lyase
Beta-Secretase
Acyltransferase
P-gp
Trk receptor
Pyroptosis
FKBP
Retinoid Receptor
Phospholipase
FOXO
c-RET
Syk
Anti-infection
Ras
NOD-like Receptor (NLR)
CFTR
MLK
Apelin receptor
Advanced Glycation End Products
NPC1L1
ASBT
Dopamine Receptor
Histone Methyltransferase
Integrin
Amino Acids and Derivatives
Estrogen/progestogen Receptor
YAP
LPL Receptor
LTR
Arrestin
DYRK
RAAS
MIF
Tie-2
GTPase
CaSR
Estrogen Receptor/ERR
Photosensitizer
Rho
Serotonin Transporter
Cell Cycle Arrest
Cysteine Protease
Neurotensin Receptor
RANKL/RANK
Aryl Hydrocarbon Receptor
Immunology/Inflammation related
Prolyl Endopeptidase (PREP)
Annexin A
FLAP
LDL
GRK
GlyT
Hexokinase
PROTAC Linker
DNA Alkylation
PAK
FAAH
ACK1
Bradykinin Receptor
CXCR
PTEN
Angiotensin-converting Enzyme (ACE)
Epoxide Hydrolase
cAMP
GluR
glycosidase
CaMK
Telomerase
TGF-beta/Smad
Lipid
MNK
Antiviral
HSP
TLR
LRRK2
Free radical scavengers
GPCR19
Urea Transporter
Histone Acetyltransferase
PAI-1
Hippo pathway
Reverse Transcriptase
c-Fms
Aromatase
PI4K
CGRP Receptor
SGK
c-Kit
IRAK
HMG-CoA Reductase
Sigma receptor
Microtubule Associated
ROS Kinase
Monoamine Oxidase
S1P Receptor
PKM
ADC Cytotoxin
IGF-2R
BTK
PGC-1α

Keywords