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TargetMol | Compound Library

FDA上市及药典收录分子库现货

FDA-Approved & Pharmacopeia Drug Library

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产品编号 L1010

传统的药物开发涉及从头确认和验证新分子实体,这是一个耗时且成本高昂的过程,随着对药物安全性及有效性的要求不断提高,开发新药的成本还将持续上涨。由于时间和成本大幅降低,近年来药物功能重定位受到越来越多关注,高内涵筛选、新的生物标志物发现和生物信息学的快速发展为基于靶点或细胞的药物重定位创造了机会。

上市药物都具有已知的和良好表征的生物活性、安全性和生物利用度,这些特征可以显著加速药物开发和优化,从上市药物中筛出的苗头化合物将为后续的药物优化计划提供有利的线索。此外,由于活性明确,靶点已知,很多科学家会从上市药物库中选择可以用于细胞诱导分化的小分子,通过单一或几个小分子的联合作用,选择出将各种体细胞诱导成为诱导多能干细胞、神经前体细胞、心肌细胞等,甚至还有使用小分子组合在体内完成诱导分化的成功尝试。

TargetMol FDA 上市及药典收录分子库收集了3280 个FDA、EMA、PMDA、NMPA 等多个国家药监局批准上市的药物以及USP、EP、BP、JP、CP 等药典收录的药物分子,可用于老药新用及细胞诱导。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L1010

FDA上市及药典收录分子库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 3280个上市及药典分子集合,可用于高通量筛选和高内涵筛选;
  • 所有化合物得到FDA、EMA、CFDA等权威部门审批或收录在USP、EP,BP、JP、CP等药典文献中;
  • 老药新用、细胞诱导的有效工具;
  • 涵盖多个研究领域:肿瘤、心血管药物、抗炎/免疫、神经系统药物、呼吸系统药物等;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • 结构多样,药效显著,可渗透细胞;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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