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TargetMol | Tags 蛋白酶体

Prolyl Endopeptidase (PREP)

脯氨酰内肽酶(PE),是一种在人类中由PREP基因编码的酶。脯氨酰内肽酶是一种大型的细胞质酶,属于一类独特的丝氨酸肽酶。该酶参与肽激素和神经肽的成熟和降解。

Y-29794 Tosylate
T35233143984-17-2
Y-29794 Tosylate (Y-29794) 是一种具有口服活性、有效且特异性的非肽脯氨酰内肽酶 (PPCE) 抑制剂。
  • ¥ 392
In stock
规格
数量
Linderene acetate
TN444226146-28-1
Linderene acetate 是一种脯氨酸肽链内切酶抑制剂,分离自Lindera strychnifolia 中。
  • ¥ 1230
In stock
规格
数量
Z-Pro-Pro-CHO
T78619108708-25-4
Z-Pro-Pro-CHO为一种有效的脯氨酰寡肽酶抑制剂,其具有针对人类及曼氏血吸虫脯氨酰寡肽酶的较低半抑制浓度(IC50),分别为0.16 μM和0.01 μM。
  • 待询
8-10周
规格
数量
Z-Pro-Pro-aldehyde-dimethyl acetal
T80106170116-63-9
Z-Pro-Pro-aldehyde-dimethyl acetal 是一种高效的脯氨酸内肽酶(PRE P)抑制剂,其IC50值为12 nM。该化合物在衰老过程和神经退行性疾病,诸如阿尔茨海默病中认知功能障碍的研究中具有重要作用。
  • 待询
规格
数量