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细胞周期化合物库

细胞周期化合物库

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产品编号 L8100 Cell Cycle Compound Library
  库化合物信息   Excel SDF

细胞周期(cell cycle)是指增殖细胞从一次分裂结束到下一次分裂结束所经历的全过程,分为间期与分裂期两个阶段,间期又分为DNA 合成前期(G1期)、DNA 合成期(S 期)与DNA 合成后期(G2期),分裂期也称为M 期。细胞周期相关化合物依赖于不同的作用机制来调控细胞周期的正常进展。这些化合物中的一些干扰CDK /细胞周期蛋白复合物,使细胞停留在G2 / M 期边界,还有一些化合物影响CaMKII 磷酸化,诱导G1期停滞。其它作用机制包括干扰RNA 功能和抑制蛋白质合成。许多这些化合物由于它们中断细胞周期而诱导细胞凋亡,可用于抗肿瘤药的筛选。 TargetMol 细胞周期化合物库是695 个细胞周期相关的小分子化合物的独特集合,用于细胞周期相关的研究及药物的筛选,可用于高通量、高内涵筛选。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 695种细胞周期相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括CDK、ROCK、Aurora Kinase、ATM/ATR、DNA-PK、DNA/RNA Synthesis等;
  • 是研究细胞周期及相关疾病的有效工具,例如癌症、心血管疾病、炎症、神经退行性疾病等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L8100)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

DNA/RNA Synthesis (188)
CDK (143)
Apoptosis (143)
Ferroptosis (94)
Autophagy (94)
Nucleoside Antimetabolite/Analog (42)
Antibacterial (41)
Aurora Kinase (41)
Endogenous Metabolite (39)
Antibiotic (36)
DUB (33)
ROCK (31)
Serine/threonin kinase (29)
PLK (22)
Chk (19)
FLT (19)
Ras (16)
Antifolate (16)
c-Myc (15)
GSK-3 (15)
Influenza Virus (15)
Parasite (14)
Dehydrogenase (14)
PKC (14)
Src (14)
IRE1 (13)
Rho (13)
VEGFR (13)
DHFR (12)
HSV (12)
PKA (11)
Reactive Oxygen Species (11)
HIV Protease (10)
PDGFR (10)
JAK (10)
SARS-CoV (10)
PD-1/PD-L1 (10)
Nrf2 (9)
Antifungal (9)
DYRK (9)
DNA Alkylator/Crosslinker (9)
Akt (8)
FGFR (8)
Topoisomerase (8)
ERK (8)
Bcr-Abl (8)
Mitophagy (8)
NF-κB (7)
Lipoxygenase (7)
c-Kit (7)
Epigenetic Reader Domain (7)
c-RET (7)
Casein Kinase (7)
S6 Kinase (7)
APC (6)
IκB/IKK (6)
Virus Protease (6)
STAT (6)
Antioxidant (6)
PPAR (6)
MEK (5)
HMG-CoA Reductase (5)
p53 (5)
COX (5)
p38 MAPK (5)
Raf (5)
Trk receptor (5)
LIM Kinase (5)
BMI-1 (5)
EGFR (5)
Sodium Channel (4)
Proteasome (4)
SGK (4)
Tyrosine Kinases (4)
Serine Protease (4)
ROS (4)
HBV (4)
DPP-4 (4)
PI3K (4)
cell cycle arrest (4)
JNK (4)
IGF-1R (3)
LRRK2 (3)
AChR (3)
KSP (3)
Kinesin (3)
5-HT Receptor (3)
PDK (3)
DNA Methyltransferase (3)
Wnt/beta-catenin (3)
Wee1 (3)
ATPase (3)
BCL (3)
TGF-beta/Smad (3)
Calcium Channel (3)
HIF/HIF Prolyl-Hydroxylase (3)
DNA Alkylation (3)
c-Met/HGFR (3)
Drug Metabolite (3)
Reverse Transcriptase (3)
GluR (3)
Glutathione Peroxidase (3)
GPX (3)
HCV Protease (3)
Mitochondrial Metabolism (3)
ribosome (2)
Syk (2)
PYK2 (2)
TAM Receptor (2)
P450 (2)
TRP/TRPV Channel (2)
NADPH (2)
mTOR (2)
MTH1 (2)
Interleukin (2)
Histone Demethylase (2)
Arginase (2)
Caspase (2)
Haspin Kinase (2)
Histone Acetyltransferase (2)
DNA-PK (2)
GRK (2)
iGluR (2)
cholecystokinin (2)
ATM/ATR (2)
Indoleamine 2,3-Dioxygenase (IDO) (2)
Carboxypeptidase (2)
Carbonic Anhydrase (2)
KLF (2)
DNA (2)
Antifection (2)
AMPK (2)
Amino Acids and Derivatives (2)
FAK (2)
MAPK (2)
DNA gyrase (2)
CXCR (1)
Cysteine Protease (1)
RSV (1)
c-Fms (1)
Sigma receptor (1)
Sirtuin (1)
CRISPR/Cas9 (1)
MLK (1)
CaMK (1)
BTK (1)
Telomerase (1)
Beta Amyloid (1)
Tie-2 (1)
TNF (1)
TOPK (1)
Aryl Hydrocarbon Receptor (1)
Tyrosinase (1)
Antiviral (1)
UGT (1)
VDAC (1)
Adenosine Receptor (1)
Xanthine Oxidase (1)
RIP kinase (1)
GABA Receptor (1)
Dopamine Receptor (1)
PAI-1 (1)
Microtubule Associated (1)
Myosin (1)
MAO (1)
NADPH-oxidase (1)
lysosomal autophagy (1)
NMDAR (1)
NO Synthase (1)
NOD-like Receptor (NLR) (1)
IRAK (1)
OCT (1)
Opioid Receptor (1)
P2Y Receptor (1)
IL Receptor (1)
HSP (1)
Histone Methyltransferase (1)
E1/E2/E3 Enzyme (1)
Potassium Channel (1)
Free radical scavengers (1)
MNK (1)
Glucokinase (1)
Proton pump (1)
Glutathione reductase (1)
GPR (1)
GST (1)
Histamine Receptor (1)
Pim (1)
HIF (1)
Phospholipase (1)
Phosphatase (1)
P-gp (1)
PERK (1)
YAP (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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