CCK-B Receptor Antagonist 2

Name: CCK-B Receptor Antagonist 2
Brand: TargetMol
SKU: T10707
Rating: 4.5 (1 reviews)

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产品编号 T10707Cas号 155412-88-7

CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM).

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CCK-B Receptor Antagonist 2

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产品编号 T10707Cas号 155412-88-7

CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM).

规格	价格	库存
2 mg	¥ 3,190	5日内发货
5 mg	¥ 3,730	5日内发货
25 mg	¥ 10,600	6-8周
50 mg	¥ 13,800	6-8周
100 mg	¥ 17,500	6-8周
1 mL x 10 mM (in DMSO)	¥ 4,120	5日内发货

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产品介绍

生物活性

产品描述	CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM).
靶点活性	Gastrin/CCK-A:1.82 μM , Gastrin/CCK-B:0.43 nM
体内活性	CCK-B Receptor Antagonist 2 (0.1 μmol/kg; i.v.) has an inhibition effect on pentagastrin-induced gastric acid secretion in anesthetized rats (ED50: 8.3 nmol/kg).

化学信息

分子量	484.55
分子式	C₂₇H₂₈N₆O₃
CAS No.	155412-88-7
密度	1.29 g/cm3 (Predicted)

储存&溶解度

存储

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

溶解度信息

DMSO: 250 mg/mL (515.94 mM), Sonication is recommended.

溶液配制表

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.0638 mL	10.3189 mL	20.6377 mL	103.1885 mL
5 mM	0.4128 mL	2.0638 mL	4.1275 mL	20.6377 mL
10 mM	0.2064 mL	1.0319 mL	2.0638 mL	10.3189 mL
20 mM	0.1032 mL	0.5159 mL	1.0319 mL	5.1594 mL
50 mM	0.0413 mL	0.2064 mL	0.4128 mL	2.0638 mL
100 mM	0.0206 mL	0.1032 mL	0.2064 mL	1.0319 mL