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临床失败化合物库

Name: 临床失败化合物库
Brand: TargetMol
SKU: L3420

很棒

产品编号 L3420

TargetMol临床失败化合物库汇集了1332种来自ClinicalTrials数据库中TERMINATED或WITHDRAWN的临床试验所涉及的药物分子。尽管这些药物未能在其原始适应症上取得成功，但它们已经经历了不同程度的人体研究，积累了宝贵的安全性和初步疗效数据。每一个化合物都附带详细的靶点信息、活性描述以及适应症等信息临床失败化合物库的药物具有较好的安全性和生物利用度，是进行老药新用的重要资源，可以大大提高药物研发的成功率，同时缩短研发周期并节约成本。

TargetMol 的所有产品和服务仅用于科学研究，不能被用于人体，我们也不向个人提供产品和服务。

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化合物库相关信息

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产品编号 L3420

临床失败化合物库

规格

1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)

询价 & 定制

产品描述

1332个临床失败化合物的独特集合，可用于高通量筛选和高内涵筛选；
涵盖多个研究领域：肿瘤、心血管药物、神经系统药物、呼吸系统药物等；
结构多样，药效显著，可渗透细胞；
详细的说明书，化合物结构、靶点信息、IC50值、活性描述等；
NMR、HPLC/LCMS等多种检测技术保证产品结构正确，纯度高，减少假阳性。

包装和储存

可选用DMSO耐受的96/384孔板或2D 条形码编码管；
干粉蓝冰运输，DMSO溶液干冰运输；
排布：96孔板：1st & 12th 空白对照，384孔板：1st & 2nd & 23th & 24th空白对照。

使用TargetMol产品
发表顶级期刊文献

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SCI 文献

文件下载

化合物库操作手册 (635 KB) Targetmol化合物库目录 (60.2 MB)

化合物库定制

您可以通过点击按钮
定制您专属的化合物！

联系专属定制

化合物库组成

Autophagy

Apoptosis

Antibacterial

Antibiotic

5-HT Receptor

Adrenergic Receptor

Dopamine Receptor

Endogenous Metabolite

HIV Protease

DNA/RNA Synthesis

Histamine Receptor

AChR

VEGFR

Parasite

FLT

Potassium Channel

Sodium Channel

c-Kit

PDGFR

EGFR

Calcium Channel

Antifungal

PI3K

COX

Dehydrogenase

JAK

SARS-CoV

Topoisomerase

Cytochromes P450

Influenza Virus

Microtubule Associated

Src

Ferroptosis

FGFR

Serotonin Transporter

PDE

c-Met/HGFR

RAAS

PPAR

Bcr-Abl

Epigenetic Reader Domain

mTOR

Mitophagy

Nucleoside Antimetabolite/Analog

CDK

HSP

Estrogen/progestogen Receptor

PKC

Glucocorticoid Receptor

Reactive Oxygen Species

HDAC

Opioid Receptor

Norepinephrine

NF-κB

HER

Proteasome

Phosphatase

HBV

Tyrosine Kinases

MAO

Endothelin Receptor

Aurora Kinase

Antiviral

Prostaglandin Receptor

Reverse Transcriptase

HCV Protease

PARP

Raf

NMDAR

Androgen Receptor

Akt

c-Fms

ribosome

GABA Receptor

Progesterone Receptor

iGluR

Vasopressin Receptor

GPR

c-RET

Neurokinin receptor

TAM Receptor

Thrombin

Proton pump

HSV

Trk receptor

Nrf2

ALK

Beta Amyloid

Retinoid Receptor

Phospholipase

TNF

Monoamine Oxidase

ATPase

Adenosine Receptor

Virus Protease

IAP

CSF-1R

Gamma-secretase

ROS

CXCR

Indoleamine 2,3-Dioxygenase (IDO)

P-gp

Hydroxylase

HMG-CoA Reductase

S1P Receptor

Carbonic Anhydrase

DHFR

LPL Receptor

Antioxidant

DNA Alkylator/Crosslinker

Factor Xa

Estrogen Receptor/ERR

Serine Protease

Antifolate

FXR

Caspase

TRP/TRPV Channel

ERK

ROCK

E1/E2/E3 Enzyme

Guanylate cyclase

DPP-4

Hedgehog/Smoothened

CCR

MMP

GluR

TLR

Ephrin Receptor

Bcl-2 Family

STAT

PLK

MEK

Cannabinoid Receptor

Syk

ADC Cytotoxin

P2Y Receptor

BACE

Histone Demethylase

MRP

GNRH Receptor

P2X Receptor

Mitochondrial Metabolism

Antifection

Molecular Glues

Smo

DNA Alkylation

IL Receptor

IGF-1R

CaMK

Interleukin

SGLT

Beta-Secretase

Ligand for E3 Ligase

HIF

DNA Methyltransferase

S6 Kinase

HIF/HIF Prolyl-Hydroxylase

ROS Kinase

Thyroid hormone receptor(THR)

Transferase

Histone Methyltransferase

Integrin

CETP

GSK-3

Kisspeptin

Glucokinase

Aryl Hydrocarbon Receptor

IDO

RIP kinase

GlyT

PAK

OX Receptor

DNA

Aminopeptidase

transporter

Decarboxylase

RSV

ATM/ATR

GST

AMPK

Oxytocin Receptor

GHSR

NADPH-oxidase

AhR

Imidazoline Receptor

p53

PD-1/PD-L1

NO Synthase

BTK

Mdm2

NOS

ROR

NEDD8

CRM1

p38 MAPK

Ligands for Target Protein for PROTAC

Reductase

IFNAR

Glutathione Peroxidase

Melatonin Receptor

c-Myc

CaSR

PKA

Pim

Rho

Serine/threonin kinase

Leukotriene Receptor

Myosin

IRE1

Drug Metabolite

MT Receptor

DNA gyrase

ABC Transporter

Integrase

Fatty Acid Synthase

Thrombopoietin Receptor

Lipoxygenase

TGF-beta/Smad

Wee1

Acyltransferase

GPCR19

GluCls

CRFR

Casein Kinase

IκB/IKK

Aromatase

Adenosine Deaminase

IRAK

Ras

Sigma receptor

p97

FAK

NOD-like Receptor (NLR)

Advanced Glycation End Products

NPC1L1

DNA-PK

Amino Acids and Derivatives

DprE1

YAP

Cell wall

NADPH

Lipase

JNK

Tie-2

gp120/CD4

VDA

Cholecystokinin Receptor

Wnt/beta-catenin

Hck

Cysteine Protease

Liver X Receptor

NAMPT

Glutaminase

SIK

FLAP

PAFR

LDL

Glucagon Receptor

Na-K-Cl cotransporter

Hexokinase

Monoamine Transporter

Isocitrate Dehydrogenase (IDH)

Thioredoxin

FAAH

Bradykinin Receptor

Cholinesterase (ChE)

Somatostatin

Chk

Xanthine Oxidase

KSP

DUB

ATP Citrate Lyase

PGE Synthase

MAPK

MNK

STING

Sirtuin

Histone Acetyltransferase

PAI-1

Pyroptosis

Methionine Adenosyltransferase (MAT)

Hippo pathway

Acetyl-CoA Carboxylase

GPX

LPA Receptor

PI4K

KLF

PDK

Aquaporin

Complement System

Discoidin Domain Receptor (DDR)

Gap Junction Protein

NOD

Tyrosinase

MLK

Kinesin

Vitamin

化合物库信息

Empty	99755-59-6	99009-20-8	98-96-4	987-78-0	98769-84-7	98717-15-8	985-12-6	98319-26-7	980-71-2	97-77-8	Empty
Empty	Rotigotine-	Pyrazoloacridine	Pyrazinamide	Citicoline	Reboxetine mesylate	Ropivacaine hydrochloride	Drotaverine hydrochloride	Finasteride	Brompheniramine maleate	Disulfiram	Empty
Empty	97657-92-6	96187-53-0	960404-48-2	96036-03-2	96020-91-6	960203-27-4	958852-01-2	95809-78-2	957054-30-7	956905-27-4	Empty
Empty	Latrepirdine dihydrochloride	Brequinar	Dapagliflozin ((2S)-1,2-propanediol, hydrate)	Meropenem	Eflornithine hydrochloride hydrate	Vortioxetine hydrobromide	GSK1059615	Devimistat	Pictilisib	PF-04217903	Empty
Empty	956483-03-7	95635-56-6	95635-55-5	956104-40-8	955365-80-7	954126-98-8	953769-46-5	953428-73-4	950769-58-1	95058-81-4	Empty
Empty	FV-100	Ranolazine dihydrochloride	Ranolazine	Apalutamide	Adavosertib	Danirixin	Sotuletinib	JNJ-39393406	Quizartinib	Gemcitabine	Empty
Empty	947331-05-7	945755-56-6	945635-15-4	945531-77-1	94497-51-5	944396-07-0	943540-75-8	943319-70-8	942123-43-5	94-16-6	Empty
Empty	Allisartan Isoproxil	XL019	Deferitazole	Ezutromid	Tamibarotene	Buparlisib	JNJ-38877605	Ponatinib	Inarigivir soproxil	Aminohippurate sodium	Empty
Empty	93957-55-2	937272-79-2	937174-76-0	936563-96-1	936539-80-9	936500-94-6	936091-26-8	935888-69-0	935881-37-1	935840-31-6	Empty
Empty	Fluvastatin sodium	Pacritinib	GSK-690693	Ibrutinib	Betrixaban maleate	Elinogrel	Fedratinib	Oprozomib	AR42	PF-03654746	Empty
Empty	935666-88-9	935283-04-8	93265-81-7	929016-96-6	928659-17-0	92823-03-5	928037-13-2	926927-61-9	92-62-6	925206-65-1	Empty
Empty	AZD-1480	Linzagolix	Ropidoxuridine	Pracinostat	Triazavirin	Flomoxef sodium	Golvatinib	Motolimod	Proflavine	RRX-001	Empty
Empty	923564-51-6	923359-38-0	923288-95-3	923288-90-8	923262-96-8	923032-37-5	920113-03-7	918639-08-4	918407-35-9	916151-99-0	Empty
Empty	Navitoclax	SAR407899	Nilotinib hydrochloride	Nilotinib monohydrochloride monohydrate	SAR407899 hydrochloride	Refametinib	Riviciclib hydrochloride	Bosutinib hydrate	Avoralstat	APTO-253	Empty
Empty	915942-22-2	915769-50-5	915385-81-8	915020-55-2	915019-65-7	914453-95-5	91374-20-8	912999-49-6	911714-45-9	91161-71-6	Empty
Empty	Neratinib maleate	Dovitinib lactate hydrate	Opaganib	BGT226	Dactolisib	Atosiban acetate	Ropinirole hydrochloride	Onalespib	SP-420	Terbinafine	Empty

Keywords

FailedClinicalTrialsCompoundLibrary

临床失败化合物库

产品编号 L3420

规格

产品描述

包装和储存

使用TargetMol产品 发表顶级期刊文献

SCI 文献

文件下载

化合物库定制

化合物库组成

化合物库信息

Keywords

使用TargetMol产品
发表顶级期刊文献