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- 1332个临床失败化合物的独特集合，可用于高通量筛选和高内涵筛选；
- 涵盖多个研究领域：肿瘤、心血管药物、神经系统药物、呼吸系统药物等；
- 结构多样，药效显著，可渗透细胞；
- 详细的说明书，化合物结构、靶点信息、IC50值、活性描述等；
- NMR、HPLC/LCMS等多种检测技术保证产品结构正确，纯度高，减少假阳性。
临床失败化合物库
很棒TargetMol临床失败化合物库汇集了1332种来自ClinicalTrials数据库中TERMINATED或WITHDRAWN的临床试验所涉及的药物分子。尽管这些药物未能在其原始适应症上取得成功，但它们已经经历了不同程度的人体研究，积累了宝贵的安全性和初步疗效数据。每一个化合物都附带详细的靶点信息、活性描述以及适应症等信息 临床失败化合物库的药物具有较好的安全性和生物利用度，是进行老药新用的重要资源，可以大大提高药物研发的成功率，同时缩短研发周期并节约成本。
TargetMol 的所有产品和服务仅用于科学研究，不能被用于人体，我们也不向个人提供产品和服务。
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化合物库相关信息
Excel
SDF
联系我们获取更多批次信息产品编号 L3420
临床失败化合物库规格
- 1 mg
- 30 μL x 10 mM (in DMSO)
- 50 μL x 10 mM (in DMSO)
- 100 μL x 10 mM (in DMSO)
- 250 μL x 10 mM (in DMSO)
询价 & 定制
产品描述
包装和储存
- 可选用DMSO耐受的96/384孔板或2D 条形码编码管；
- 干粉蓝冰运输，DMSO溶液干冰运输；
- 排布：96孔板：1st & 12th 空白对照，384孔板：1st & 2nd & 23th & 24th空白对照。
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化合物库组成
Autophagy
Apoptosis
Antibacterial
Antibiotic
5-HT Receptor
Adrenergic Receptor
Dopamine Receptor
Endogenous Metabolite
HIV Protease
DNA/RNA Synthesis
Histamine Receptor
AChR
VEGFR
Parasite
FLT
Potassium Channel
Sodium Channel
c-Kit
PDGFR
EGFR
Calcium Channel
Antifungal
PI3K
COX
Dehydrogenase
JAK
SARS-CoV
Topoisomerase
Cytochromes P450
Influenza Virus
Microtubule Associated
Src
Ferroptosis
FGFR
Serotonin Transporter
PDE
c-Met/HGFR
RAAS
PPAR
Bcr-Abl
Epigenetic Reader Domain
mTOR
Mitophagy
Nucleoside Antimetabolite/Analog
CDK
HSP
Estrogen/progestogen Receptor
PKC
Glucocorticoid Receptor
Opioid Receptor
Reactive Oxygen Species
HDAC
Norepinephrine
NF-κB
HER
Proteasome
Phosphatase
HBV
Tyrosine Kinases
MAO
Endothelin Receptor
Aurora Kinase
Antiviral
Prostaglandin Receptor
Reverse Transcriptase
HCV Protease
PARP
Raf
NMDAR
Androgen Receptor
Akt
c-Fms
ribosome
GABA Receptor
Progesterone Receptor
iGluR
Vasopressin Receptor
GPR
c-RET
Neurokinin receptor
TAM Receptor
Thrombin
Proton pump
HSV
Trk receptor
Nrf2
ALK
Beta Amyloid
Retinoid Receptor
Phospholipase
TNF
Monoamine Oxidase
ATPase
Adenosine Receptor
Virus Protease
IAP
CSF-1R
Gamma-secretase
ROS
CXCR
Indoleamine 2,3-Dioxygenase (IDO)
P-gp
Hydroxylase
HMG-CoA Reductase
S1P Receptor
Carbonic Anhydrase
DHFR
Antioxidant
LPL Receptor
DNA Alkylator/Crosslinker
Factor Xa
Estrogen Receptor/ERR
Serine Protease
Antifolate
FXR
Caspase
TRP/TRPV Channel
ERK
ROCK
E1/E2/E3 Enzyme
Guanylate cyclase
DPP-4
Hedgehog/Smoothened
CCR
MMP
GluR
TLR
Ephrin Receptor
Bcl-2 Family
STAT
PLK
MEK
Cannabinoid Receptor
Syk
ADC Cytotoxin
P2Y Receptor
BACE
Histone Demethylase
GNRH Receptor
MRP
P2X Receptor
Mitochondrial Metabolism
Antifection
Molecular Glues
Smo
DNA Alkylation
IL Receptor
IGF-1R
CaMK
Interleukin
SGLT
Beta-Secretase
Ligand for E3 Ligase
HIF
DNA Methyltransferase
S6 Kinase
HIF/HIF Prolyl-Hydroxylase
ROS Kinase
Thyroid hormone receptor(THR)
Transferase
Histone Methyltransferase
Integrin
CETP
GSK-3
Kisspeptin
Glucokinase
Aryl Hydrocarbon Receptor
IDO
RIP kinase
GlyT
PAK
OX Receptor
DNA
Aminopeptidase
transporter
Decarboxylase
RSV
ATM/ATR
GST
AMPK
Oxytocin Receptor
GHSR
NADPH-oxidase
AhR
Imidazoline Receptor
p53
PD-1/PD-L1
NO Synthase
BTK
Mdm2
NOS
ROR
NEDD8
CRM1
p38 MAPK
Ligands for Target Protein for PROTAC
IFNAR
Reductase
Glutathione Peroxidase
Melatonin Receptor
c-Myc
CaSR
PKA
Pim
Rho
Serine/threonin kinase
Leukotriene Receptor
IRE1
Myosin
Drug Metabolite
MT Receptor
DNA gyrase
ABC Transporter
Integrase
Fatty Acid Synthase
Thrombopoietin Receptor
Lipoxygenase
TGF-beta/Smad
Wee1
Acyltransferase
GPCR19
GluCls
CRFR
Casein Kinase
IκB/IKK
Aromatase
Adenosine Deaminase
IRAK
Ras
Sigma receptor
p97
FAK
NOD-like Receptor (NLR)
Advanced Glycation End Products
NPC1L1
DNA-PK
DprE1
Amino Acids and Derivatives
YAP
Cell wall
NADPH
Lipase
JNK
gp120/CD4
Tie-2
VDA
Cholecystokinin Receptor
Wnt/beta-catenin
Hck
Liver X Receptor
Cysteine Protease
NAMPT
Glutaminase
SIK
FLAP
PAFR
LDL
Glucagon Receptor
Na-K-Cl cotransporter
Hexokinase
Monoamine Transporter
Isocitrate Dehydrogenase (IDH)
Thioredoxin
FAAH
Bradykinin Receptor
Cholinesterase (ChE)
Somatostatin
Chk
Xanthine Oxidase
KSP
DUB
ATP Citrate Lyase
PGE Synthase
MAPK
MNK
STING
Sirtuin
Histone Acetyltransferase
PAI-1
Pyroptosis
Methionine Adenosyltransferase (MAT)
Hippo pathway
Acetyl-CoA Carboxylase
GPX
LPA Receptor
KLF
PI4K
PDK
Aquaporin
Complement System
Discoidin Domain Receptor (DDR)
Gap Junction Protein
NOD
Tyrosinase
MLK
Kinesin
Vitamin
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