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活性脂质化合物库

活性脂质化合物库

产品编号 L7000 Bioactive Lipid Compound Library
  库化合物信息   Excel SDF

研究表明,多种脂质分子能够调节组织的脂肪酸构成或诱导细胞信号通路,具有促进身体健康的作用。除了某些短链或中链脂肪酸以外,多不饱和脂肪酸(PUFA)是重要的生物活性脂质分子,PUFA 大部分来源于植物油,是合成细胞激素(二十烷类化合物)及其他调节人体健康的信号分子的重要前体物质。PUFA 的益处与它们的构型有关,顺式异构体是主要的生物活性形式,能够增加膜的流动性,促进细胞之间的通讯,维持正常的稳态,阻止代谢疾病的发展。

TargetMol 为您提供大量活性脂质相关化合物,L7000 包含385 个脂质相关的小分子化合物抑制剂,充分满足您的科研需求;

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 385种生物活性小分子化合物,用于高通量、高内涵筛选;
  • 靶点包括GPCR、 HDAC、PPAR、DNA Alkylating、EGFR等;?
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L7000)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Endogenous Metabolite (91)
Autophagy (82)
Apoptosis (53)
PDE (48)
COX (25)
PPAR (20)
Estrogen/progestogen Receptor (19)
Antibacterial (18)
Phospholipase (17)
MAO (15)
Ferroptosis (13)
TRP/TRPV Channel (11)
Antifungal (10)
HMG-CoA Reductase (10)
P450 (10)
Lipoxygenase (10)
Prostaglandin Receptor (10)
HDAC (9)
Thrombin (9)
Mitophagy (9)
HIV Protease (9)
Antibiotic (8)
Adenosine Receptor (8)
FXR (8)
Cannabinoid Receptor (8)
Estrogen Receptor/ERR (8)
NF-κB (8)
Monoamine Oxidase (8)
Glucocorticoid Receptor (8)
Potassium Channel (7)
Retinoid Receptor (7)
Lipase (7)
Reactive Oxygen Species (7)
PI3K (7)
Virus Protease (6)
Fatty Acid Synthase (6)
TNF (6)
Factor Xa (6)
AhR (6)
Lipid (6)
Parasite (5)
Aryl Hydrocarbon Receptor (5)
Casein Kinase (5)
Adrenergic Receptor (5)
Sirtuin (5)
Calcium Channel (5)
Progesterone Receptor (5)
Dehydrogenase (5)
AChR (5)
p38 MAPK (4)
GABA Receptor (4)
Influenza Virus (4)
PKC (4)
CETP (4)
Histamine Receptor (4)
GPR (4)
Nrf2 (4)
FAAH (3)
PLK (3)
Akt (3)
HIF (3)
5-HT Receptor (3)
DNA/RNA Synthesis (3)
IκB/IKK (3)
Androgen Receptor (3)
GPCR19 (3)
Sodium Channel (3)
p53 (3)
Antioxidant (3)
Phosphatase (3)
Liver X Receptor (3)
Glutathione Peroxidase (2)
MMP (2)
Acyltransferase (2)
AChE (2)
RSV (2)
ERK (2)
Histone Demethylase (2)
LPA Receptor (2)
DNA-PK (2)
CaMK (2)
DNA (2)
LTR (2)
LPL Receptor (2)
mTOR (2)
GSK-3 (2)
PAK (2)
TGF-beta/Smad (2)
Chloride channel (2)
Caspase (2)
Leukotriene Receptor (2)
LDL (2)
CDK (2)
PARP (2)
Mitochondrial Metabolism (2)
ROS (2)
Opioid Receptor (2)
BCL (2)
MRP (2)
Mdm2 (2)
HIF/HIF Prolyl-Hydroxylase (1)
PKM (1)
PAI-1 (1)
ALK (1)
S1P Receptor (1)
MLK (1)
MEK (1)
FAK (1)
Microtubule Associated (1)
ATM/ATR (1)
Acetyl-CoA Carboxylase (1)
Tyrosinase (1)
c-RET (1)
Ras (1)
NOD (1)
AMPK (1)
NADPH-oxidase (1)
Platelet aggregation (1)
Hydroxylase (1)
STAT (1)
Proteasome (1)
Histone Acetyltransferase (1)
NADPH (1)
iGluR (1)
VEGFR (1)
Cysteine Protease (1)
Nucleoside Antimetabolite/Analog (1)
Wnt/beta-catenin (1)
Tyrosine Kinases (1)
HBV (1)
PKA (1)
ABC (1)
Melatonin Receptor (1)
DYRK (1)
Topoisomerase (1)
Reductase (1)
DNA Alkylator/Crosslinker (1)
c-Met/HGFR (1)
Src (1)
ROR (1)
Dopamine Receptor (1)
Monocarboxylate transporter (1)
Transferase (1)
NOS (1)
ATPase (1)
IAP (1)
Annexin A (1)
SARS-CoV (1)
IL Receptor (1)
HSP (1)
P-gp (1)
MNK (1)
PGE Synthase (1)
EGFR (1)
Epigenetic Reader Domain (1)
GluR (1)
Epoxide Hydrolase (1)
Xanthine Oxidase (1)
PAD (1)
HSV (1)
RIP kinase (1)
Hedgehog/Smoothened (1)
PDGFR (1)
Smo (1)
Guanylate cyclase (1)
NMDAR (1)
P2X Receptor (1)
Phosphorylase (1)
Drug Metabolite (1)
Gamma-secretase (1)
UGT (1)
NO Synthase (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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