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TargetMol | Compound Library

天然多酚类化合物库现货

Polyphenolic Natural Product Library
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货号 L6100

天然多酚类化合物具有抗氧化、抗癌、抗诱变和抗炎等多种生物活性,能够阻滞细胞周期,诱导细胞凋亡,抑制细胞粘附、迁移、增殖和分化,在癌症预防和治疗中发挥重要作用。来自药草和膳食植物的酚类化合物包括酚酸、类黄酮、单宁、芪类、类姜黄素、香豆素、木脂素、醌等,其特征在于存在大量的苯酚结构单元,这些酚结构的存在决定了每一个化合物独特的物理、化学和生物特性。

天然多酚类化合物库是825 个天然多酚化合物的独特集合,是筛选抗癌药物的理想工具,可用于高通量和高内涵筛选。

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货号 L6100

天然多酚类化合物库

规格

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 825 种天然多酚化合物,用于高通量筛选和高内涵筛选;
  • 靶点包括 JAK、AMPK、CYP 等;
  • 详细的化合物信息,包括结构、靶点、IC50 值和生物活性描述;
  • 结构多样,具有药物活性和细胞通透性;
  • NMR、HPLC/LCMS 等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
NF-κB
Antibacterial
ROS
Autophagy
Antioxidant
Endogenous Metabolite
Reactive Oxygen Species
COX
Akt
Antifungal
p38 MAPK
NO Synthase
Cytochromes P450
TNF
ERK
HIV Protease
PI3K
Tyrosinase
DNA/RNA Synthesis
Influenza Virus
Interleukin
Caspase
Glucosidase
AMPK
Anti-infection
Nrf2
Antibiotic
Parasite
Bcl-2 Family
glycosidase
MMP
PPAR
JNK
STAT
Virus Protease
Cholinesterase (ChE)
IL Receptor
Estrogen Receptor/ERR
PKC
Lipoxygenase
Wnt/beta-catenin
Phosphatase
Ferroptosis
GABA Receptor
HSV
Reductase
Immunology/Inflammation related
mTOR
TLR
Antifection
Calcium Channel
HBV
Xanthine Oxidase
5-HT Receptor
HIF/HIF Prolyl-Hydroxylase
PARP
PDE
Estrogen/progestogen Receptor
Drug Metabolite
SARS-CoV
Dehydrogenase
transporter
Beta Amyloid
MAO
EGFR
NOS
Topoisomerase
Mitophagy
CDK
TGF-beta/Smad
TRP/TRPV Channel
Adrenergic Receptor
Monoamine Oxidase
HDAC
P-gp
Androgen Receptor
GSK-3
PKA
JAK
IκB/IKK
AChR
ATPase
IGF-1R
p53
UGT
Phospholipase
SGLT
Antiviral
NOD-like Receptor (NLR)
Angiotensin-converting Enzyme (ACE)
MAPK
Ras
GPCR
NOD
Carbonic Anhydrase
PERK
Sirtuin
Amylase
Aryl Hydrocarbon Receptor
Prostaglandin Receptor
Free radical scavengers
Dopamine Receptor
Microtubule Associated
RAAS
Epigenetic Reader Domain
Transferase
Reverse Transcriptase
Sodium Channel
IAP
Casein Kinase
HCV Protease
LDL
Fatty Acid Synthase
Integrin
CaMK
MEK
Lipase
VEGFR
Gamma-secretase
Mitochondrial Metabolism
Potassium Channel
Adenosine Receptor
c-Myc
cAMP
Histone Acetyltransferase
GST
Aromatase
MDM-2/p53
Platelet aggregation
PD-1/PD-L1
Src
NR4A
PDGFR
DNA
Hydroxylase
Chloride channel
Glutathione Peroxidase
PTEN
Cannabinoid Receptor
HMG-CoA Reductase
FAK
Proteasome
Histamine Receptor
Hedgehog/Smoothened
Beta-Secretase
Acyltransferase
ATM/ATR
FOXO
ADC Cytotoxin
IFNAR
BACE
Pim
RANKL/RANK
Bombesin Receptor
Lipid
S6 Kinase
AhR
Trk receptor
Syk
FOXO3
CAT
Arginase
c-Met/HGFR
CaSR
Liver X Receptor
Ephrin Receptor
AIM2
Melanocortin Receptor
HIF
ROS Kinase
stilbene oxidase
CD38
Histone Demethylase
Tyrosine Kinases
ATG
iGluR
ABC Transporter
Monoamine Transporter
FAAH
CCR
p62
Proton pump
Monocarboxylate transporter
MyD88
Arrestin
Serine/threonin kinase
Cysteine Protease
FXR
Leukotriene Receptor
Opioid Receptor
CXCR
Cadherin
Norepinephrine
Pyroptosis
Acetyl-CoA Carboxylase
Retinoid Receptor
CGRP Receptor
NADPH-oxidase
MLK
PKM
Histone Methyltransferase
Adenylate cyclase
RIP kinase
Bcr-Abl
Aurora Kinase
Thrombopoietin Receptor
PGE Synthase
Aminopeptidase
Urea Transporter
FGFR
Serotonin Transporter
Decarboxylase
Adenosine Deaminase
Advanced Glycation End Products
Cell wall
Necroptosis
OCT
Telomerase
PSMA
hCE
Dynamin
Serine Protease
Cell Cycle Arrest
Glucokinase
MTH1
NMDAR
DPP-4
HCAR
Chk
OAT
RSV
Protease
PLK

Keywords