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TargetMol | Compound Library

抗胰腺癌化合物库现货

Anti-Pancreatic Cancer Compound Library

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产品编号 L2192

随着医学技术的进步,大部分癌症的生存率都在提高,例如乳腺癌,结直肠癌等肿瘤,近几十年来,生存率得到了大幅度的提升。但是,有一个例外,那就是胰腺癌,胰腺癌是一种发病隐匿,进展迅速,治疗效果和预后极差的消化道恶性肿瘤。胰腺癌的生存率一直停滞不前,胰腺癌的五年生存率只有5%至10%,绝大部分患者在诊断胰腺癌半年内死亡,由于生存率低,死亡率高,胰腺癌称为癌中之王。

为了满足胰腺癌研究客户的需求,TargeMol 收集了 2508 种与胰腺癌相关的化合物,作用于 KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等胰腺癌相关靶点,助力胰腺癌治疗药物的开发。

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产品编号 L2192

抗胰腺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品特点 产品特点

  • 2508种与胰腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 靶点含KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
EGFR
CDK
COX
VEGFR
Ras
Akt
PPAR
Wnt/beta-catenin
mTOR
JAK
ERK
HDAC
PARP
STAT
Endogenous Metabolite
Src
p38 MAPK
GSK-3
AMPK
Antibacterial
FGFR
Raf
ROS
c-Met/HGFR
PDGFR
MDM-2/p53
FLT
TGF-beta/Smad
Caspase
Parasite
Kras
p53
JNK
c-Kit
MEK
Reactive Oxygen Species
TNF
MMP
Potassium Channel
DNA/RNA Synthesis
IGF-1R
S6 Kinase
HIF/HIF Prolyl-Hydroxylase
Tyrosine Kinases
Bcr-Abl
DNA-PK
Interleukin
Ferroptosis
Bcl-2 Family
ATM/ATR
MAPK
Cytochromes P450
Aurora Kinase
ALK
NO Synthase
HER
Antibiotic
HIV Protease
Influenza Virus
Mitophagy
c-RET
Gamma-secretase
IL Receptor
Mdm2
STING
Antifungal
PDK
PD-1/PD-L1
HIF
Hedgehog/Smoothened
Pim
PKC
E1/E2/E3 Enzyme
Dehydrogenase
Calcium Channel
Prostaglandin Receptor
Virus Protease
Lipoxygenase
Nrf2
Beta Amyloid
FAK
PKA
Casein Kinase
IκB/IKK
PI4K
Topoisomerase
Trk receptor
c-Fms
Epigenetic Reader Domain
PDE
Chk
NOS
Phosphatase
HSV
Rho
TAM Receptor
TLR
Tyrosinase
Mitochondrial Metabolism
Adrenergic Receptor
Sirtuin
GABA Receptor
Sodium Channel
HCV Protease
PTEN
P-gp
ROCK
Anti-infection
PERK
DYRK
c-Myc
Tie-2
SIK
Smo
HSP
PLK
Syk
5-HT Receptor
Antioxidant
Drug Metabolite
PGE Synthase
Microtubule Associated
Adenosine Receptor
Ephrin Receptor
Integrin
AChR
Aryl Hydrocarbon Receptor
MLK
ATPase
Antifection
GPCR
Histone Acetyltransferase
MELK
Proteasome
CSF-1R
Glucosidase
SARS-CoV
Cannabinoid Receptor
Serine Protease
TRP/TRPV Channel
CaMK
Antiviral
transporter
SGK
IAP
RIP kinase
BTK
IRAK
ROS Kinase
Estrogen Receptor/ERR
Serine/threonin kinase
IFNAR
NOD-like Receptor (NLR)
Carbonic Anhydrase
glycosidase
Estrogen/progestogen Receptor
PYK2
GTPase
Reductase
Histamine Receptor
Cholecystokinin Receptor
Chloride channel
Proton pump
DNA Alkylator/Crosslinker
LDL
Opioid Receptor
Retinoid Receptor
Transferase
HBV
CCR
Cholinesterase (ChE)
Histone Methyltransferase
Survivin
cAMP
Reverse Transcriptase
NOD
RAAS
DNA Alkylation
Decarboxylase
Phospholipase
Glutathione Peroxidase
Leukotriene Receptor
OXPHOS
LRRK2
Free radical scavengers
FKBP
NMDAR
Angiotensin-converting Enzyme (ACE)
DUB
MNK
BACE
NADPH
Hck
Glucocorticoid Receptor
DNA Methyltransferase
Histone Demethylase
Nucleoside Antimetabolite/Analog
ATP Citrate Lyase
Porcupine
Hippo pathway
Dopamine Receptor
MRP
UGT
Fatty Acid Synthase
Androgen Receptor
Discoidin Domain Receptor (DDR)
Progesterone Receptor
PAK
Aromatase
Gap Junction Protein
Myosin
Beta-Secretase
Acyltransferase
FXR
Prolyl Endopeptidase (PREP)
Pyroptosis
NADPH-oxidase
Cell Cycle Arrest
Glucokinase
Immunology/Inflammation related
RSV
S1P Receptor
ADC Cytotoxin
RANKL/RANK
Lipid
iGluR
ABC Transporter
Monoamine Transporter
FAAH
GluR
CFTR
DAPK
Kinesin
Y Box Binding Protein 1
Arginase
Na+/Ca2+ Exchanger
gp120/CD4
ASCT
Liver X Receptor
AIM2
PAI-1
Melanin-concentrating Hormone Receptor (MCHR)
NPC1L1
DHFR
TOPK
FLAP
Thioredoxin
Adenosine Deaminase
RAR/RXR
MyD88
Cysteine Protease
IRE1
FABP
Guanylate cyclase
Epoxide Hydrolase
Cadherin
PKM
MicroRNA
ROR
Amino Acids and Derivatives
PAFR
Haspin Kinase
Hexokinase
DPP-4
YAP
OCT
Na-K-Cl cotransporter
ACK1
hCE
LPA Receptor
BMI-1
Thrombin
Monoamine Oxidase
CD38
LTR
VDA
NR4A
DNA
CRISPR/Cas9
Hydroxylase
Sigma receptor
Adenylyl Cyclase
LPL Receptor
MIF
PAD
Thrombopoietin Receptor
BCRP
Aminopeptidase
ASK
Methionine Adenosyltransferase (MAT)
p97

Keywords