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TargetMol | Compound Library

抗胰腺癌化合物库现货

Anti-Pancreatic Cancer Compound Library
Rating icon 很棒
货号 L2192

随着医学技术的进步,大部分癌症的生存率都在提高,例如乳腺癌,结直肠癌等肿瘤,近几十年来,生存率得到了大幅度的提升。但是,有一个例外,那就是胰腺癌,胰腺癌是一种发病隐匿,进展迅速,治疗效果和预后极差的消化道恶性肿瘤。胰腺癌的生存率一直停滞不前,胰腺癌的五年生存率只有5%至10%,绝大部分患者在诊断胰腺癌半年内死亡,由于生存率低,死亡率高,胰腺癌称为癌中之王。

为了满足胰腺癌研究客户的需求,TargeMol 收集了 2508 种与胰腺癌相关的化合物,作用于 KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等胰腺癌相关靶点,助力胰腺癌治疗药物的开发。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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货号 L2192

抗胰腺癌化合物库

规格

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品特点 产品特点

  • 2508种与胰腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 靶点含KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
EGFR
CDK
COX
VEGFR
Ras
Akt
PPAR
Wnt/beta-catenin
mTOR
JAK
ERK
STAT
HDAC
PARP
Src
Endogenous Metabolite
p38 MAPK
GSK-3
Antibacterial
AMPK
FGFR
Raf
ROS
PDGFR
c-Met/HGFR
MDM-2/p53
FLT
Caspase
TGF-beta/Smad
Parasite
Kras
p53
JNK
c-Kit
MEK
MMP
Reactive Oxygen Species
TNF
Potassium Channel
DNA/RNA Synthesis
IGF-1R
S6 Kinase
HIF/HIF Prolyl-Hydroxylase
Tyrosine Kinases
Bcr-Abl
DNA-PK
Interleukin
MAPK
Bcl-2 Family
ATM/ATR
Cytochromes P450
Ferroptosis
ALK
Aurora Kinase
HER
NO Synthase
Antibiotic
HIV Protease
Influenza Virus
Mitophagy
Gamma-secretase
Mdm2
c-RET
PDK
Antifungal
IL Receptor
STING
PD-1/PD-L1
Pim
PKC
E1/E2/E3 Enzyme
Hedgehog/Smoothened
Dehydrogenase
HIF
Virus Protease
Calcium Channel
Beta Amyloid
Prostaglandin Receptor
Nrf2
Lipoxygenase
FAK
Casein Kinase
PKA
PI4K
IκB/IKK
Topoisomerase
c-Fms
Trk receptor
PDE
Epigenetic Reader Domain
Chk
NOS
Phosphatase
HSV
Tyrosinase
Adrenergic Receptor
Anti-infection
Sirtuin
TLR
Rho
TAM Receptor
ROCK
Mitochondrial Metabolism
HCV Protease
PTEN
P-gp
GABA Receptor
Sodium Channel
5-HT Receptor
PLK
Syk
Antioxidant
PERK
DYRK
c-Myc
Drug Metabolite
PGE Synthase
Microtubule Associated
Tie-2
SIK
Smo
HSP
IAP
Aryl Hydrocarbon Receptor
MLK
Adenosine Receptor
Ephrin Receptor
Antifection
Integrin
AChR
TRP/TRPV Channel
CaMK
Antiviral
SGK
Serine Protease
ATPase
Cannabinoid Receptor
GPCR
Histone Acetyltransferase
MELK
RIP kinase
Proteasome
CSF-1R
Glucosidase
SARS-CoV
BTK
IFNAR
transporter
NOD-like Receptor (NLR)
Carbonic Anhydrase
glycosidase
Serine/threonin kinase
IRAK
ROS Kinase
Estrogen/progestogen Receptor
PYK2
Survivin
Estrogen Receptor/ERR
Transferase
Hck
HBV
CCR
Cholinesterase (ChE)
Chloride channel
Proton pump
DNA Alkylator/Crosslinker
Opioid Receptor
Retinoid Receptor
GTPase
Histone Methyltransferase
Reductase
Histamine Receptor
Cholecystokinin Receptor
BACE
NADPH
Glucocorticoid Receptor
DNA Methyltransferase
NMDAR
Angiotensin-converting Enzyme (ACE)
DUB
MNK
Histone Demethylase
Nucleoside Antimetabolite/Analog
ATP Citrate Lyase
Porcupine
Hippo pathway
Glutathione Peroxidase
Leukotriene Receptor
LDL
OXPHOS
LRRK2
Free radical scavengers
FKBP
cAMP
Reverse Transcriptase
NOD
Dopamine Receptor
MRP
UGT
Fatty Acid Synthase
Androgen Receptor
Discoidin Domain Receptor (DDR)
RAAS
DNA Alkylation
Decarboxylase
Phospholipase
ADC Cytotoxin
RANKL/RANK
Lipid
Cell Cycle Arrest
Glucokinase
Immunology/Inflammation related
RSV
S1P Receptor
iGluR
ABC Transporter
Monoamine Transporter
FAAH
GluR
CFTR
FXR
Prolyl Endopeptidase (PREP)
Pyroptosis
NADPH-oxidase
Progesterone Receptor
PAK
Aromatase
Gap Junction Protein
Aminopeptidase
DAPK
Kinesin
Beta-Secretase
Acyltransferase
YAP
OCT
Na-K-Cl cotransporter
ACK1
hCE
LPA Receptor
BMI-1
Thrombin
Monoamine Oxidase
MicroRNA
ROR
Amino Acids and Derivatives
PAFR
Haspin Kinase
Hexokinase
DPP-4
CD38
LTR
VDA
NR4A
DNA
Hydroxylase
Sigma receptor
RAR/RXR
MyD88
Cysteine Protease
IRE1
FABP
Guanylate cyclase
Epoxide Hydrolase
Cadherin
PKM
Y Box Binding Protein 1
Arginase
Na+/Ca2+ Exchanger
gp120/CD4
ASCT
Liver X Receptor
AIM2
PAI-1
LPL Receptor
MIF
Glutaminase
Adenylate cyclase
PAD
Thrombopoietin Receptor
BCRP
ASK
Methionine Adenosyltransferase (MAT)
p97
Melanin-concentrating Hormone Receptor (MCHR)
NPC1L1
DHFR
TOPK
Myosin
FLAP
Thioredoxin
Adenosine Deaminase

Keywords