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TargetMol | Compound Library

抗胰腺癌化合物库现货

Anti-Pancreatic Cancer Compound Library

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产品编号 L2192

随着医学技术的进步,大部分癌症的生存率都在提高,例如乳腺癌,结直肠癌等肿瘤,近几十年来,生存率得到了大幅度的提升。但是,有一个例外,那就是胰腺癌,胰腺癌是一种发病隐匿,进展迅速,治疗效果和预后极差的消化道恶性肿瘤。胰腺癌的生存率一直停滞不前,胰腺癌的五年生存率只有5%至10%,绝大部分患者在诊断胰腺癌半年内死亡,由于生存率低,死亡率高,胰腺癌称为癌中之王。

为了满足胰腺癌研究客户的需求,TargeMol 收集了 2508 种与胰腺癌相关的化合物,作用于 KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等胰腺癌相关靶点,助力胰腺癌治疗药物的开发。

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产品编号 L2192

抗胰腺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品特点 产品特点

  • 2508种与胰腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 靶点含KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
EGFR
CDK
COX
VEGFR
Ras
PPAR
Akt
Wnt/beta-catenin
mTOR
JAK
PARP
HDAC
ERK
STAT
Endogenous Metabolite
Src
GSK-3
AMPK
Antibacterial
FGFR
p38 MAPK
c-Met/HGFR
Raf
PDGFR
MDM-2/p53
FLT
TGF-beta/Smad
Kras
Parasite
p53
Caspase
c-Kit
JNK
Reactive Oxygen Species
MEK
MMP
Potassium Channel
TNF
S6 Kinase
IGF-1R
Tyrosine Kinases
HIF/HIF Prolyl-Hydroxylase
DNA-PK
Bcr-Abl
DNA/RNA Synthesis
ATM/ATR
Ferroptosis
Cytochromes P450
Aurora Kinase
MAPK
ALK
Bcl-2 Family
HER
HIV Protease
Antibiotic
Mitophagy
IL Receptor
Influenza Virus
c-RET
Mdm2
Antifungal
Gamma-secretase
Interleukin
PDK
STING
Pim
E1/E2/E3 Enzyme
HIF
PKC
Hedgehog/Smoothened
PD-1/PD-L1
Dehydrogenase
Virus Protease
Lipoxygenase
NO Synthase
PKA
Calcium Channel
Casein Kinase
Prostaglandin Receptor
IκB/IKK
PI4K
FAK
Topoisomerase
Beta Amyloid
Nrf2
c-Fms
Epigenetic Reader Domain
Trk receptor
PDE
Chk
NOS
Phosphatase
Tyrosinase
Rho
ROS
HSV
Sirtuin
Anti-infection
TAM Receptor
HCV Protease
ROCK
Mitochondrial Metabolism
PTEN
GABA Receptor
Antioxidant
DYRK
PERK
Tie-2
Adrenergic Receptor
SIK
Drug Metabolite
Smo
PGE Synthase
P-gp
5-HT Receptor
Syk
Sodium Channel
Microtubule Associated
ATPase
c-Myc
Aryl Hydrocarbon Receptor
Antifection
HSP
TLR
Ephrin Receptor
GPCR
Proteasome
Integrin
TRP/TRPV Channel
IAP
CSF-1R
Glucosidase
Antiviral
Histone Acetyltransferase
transporter
MELK
PLK
SGK
Cannabinoid Receptor
AChR
MLK
BTK
Carbonic Anhydrase
Estrogen/progestogen Receptor
Adenosine Receptor
Serine/threonin kinase
PYK2
RIP kinase
SARS-CoV
IRAK
ROS Kinase
Chloride channel
Proton pump
Transferase
Histone Methyltransferase
DNA Alkylator/Crosslinker
IFNAR
Histamine Receptor
GTPase
Estrogen Receptor/ERR
HBV
Cholecystokinin Receptor
Serine Protease
LDL
Opioid Receptor
CCR
Cholinesterase (ChE)
Retinoid Receptor
NOD-like Receptor (NLR)
Reductase
BACE
Histone Demethylase
NADPH
RAAS
Glutathione Peroxidase
MRP
Hck
Nucleoside Antimetabolite/Analog
Leukotriene Receptor
Glucocorticoid Receptor
NMDAR
DNA Alkylation
Angiotensin-converting Enzyme (ACE)
cAMP
CaMK
DUB
Androgen Receptor
ATP Citrate Lyase
OXPHOS
MNK
Survivin
Porcupine
LRRK2
Free radical scavengers
Decarboxylase
Hippo pathway
FKBP
Reverse Transcriptase
Phospholipase
Discoidin Domain Receptor (DDR)
DNA Methyltransferase
NOD
Dopamine Receptor
ADC Cytotoxin
Progesterone Receptor
Cell Cycle Arrest
FXR
Glucokinase
Immunology/Inflammation related
iGluR
Prolyl Endopeptidase (PREP)
Myosin
UGT
ABC Transporter
Fatty Acid Synthase
PAK
FAAH
GluR
Lipid
Beta-Secretase
Acyltransferase
Aminopeptidase
Pyroptosis
RSV
Aromatase
Gap Junction Protein
DAPK
NADPH-oxidase
CFTR
S1P Receptor
Melanin-concentrating Hormone Receptor (MCHR)
Adenylyl Cyclase
MicroRNA
NPC1L1
RAR/RXR
CD38
DHFR
ROR
Amino Acids and Derivatives
MyD88
Y Box Binding Protein 1
YAP
Arginase
LPL Receptor
LTR
Na+/Ca2+ Exchanger
gp120/CD4
MIF
TOPK
VDA
OCT
ASCT
Cysteine Protease
Liver X Receptor
NR4A
RANKL/RANK
IRE1
FLAP
PAFR
Haspin Kinase
Na-K-Cl cotransporter
Monoamine Transporter
Hexokinase
Guanylate cyclase
DPP-4
Thioredoxin
ACK1
PAD
Epoxide Hydrolase
Thrombopoietin Receptor
DNA
BCRP
AIM2
ASK
hCE
PAI-1
Methionine Adenosyltransferase (MAT)
LPA Receptor
CRISPR/Cas9
Hydroxylase
Adenosine Deaminase
BMI-1
Sigma receptor
Thrombin
p97
Kinesin
PKM
Monoamine Oxidase

Keywords