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TargetMol | Compound Library

抗胰腺癌化合物库现货

Anti-Pancreatic Cancer Compound Library

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产品编号 L2192

随着医学技术的进步,大部分癌症的生存率都在提高,例如乳腺癌,结直肠癌等肿瘤,近几十年来,生存率得到了大幅度的提升。但是,有一个例外,那就是胰腺癌,胰腺癌是一种发病隐匿,进展迅速,治疗效果和预后极差的消化道恶性肿瘤。胰腺癌的生存率一直停滞不前,胰腺癌的五年生存率只有5%至10%,绝大部分患者在诊断胰腺癌半年内死亡,由于生存率低,死亡率高,胰腺癌称为癌中之王。 为了满足胰腺癌研究客户的需求,TargeMol 收集了 2508 种与胰腺癌相关的化合物,作用于 KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等胰腺癌相关靶点,助力胰腺癌治疗药物的开发。

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产品编号 L2192

抗胰腺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品特点 产品特点

  • 2508种与胰腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 靶点含KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
EGFR
CDK
COX
VEGFR
Ras
PPAR
Wnt/beta-catenin
mTOR
Akt
JAK
HDAC
PARP
ERK
STAT
Endogenous Metabolite
Src
GSK-3
AMPK
Antibacterial
FGFR
p38 MAPK
c-Met/HGFR
Raf
PDGFR
MDM-2/p53
FLT
TGF-beta/Smad
Kras
Parasite
p53
c-Kit
Caspase
Reactive Oxygen Species
MEK
MMP
Potassium Channel
JNK
TNF
S6 Kinase
IGF-1R
Tyrosine Kinases
Bcr-Abl
DNA-PK
HIF/HIF Prolyl-Hydroxylase
ATM/ATR
DNA/RNA Synthesis
Ferroptosis
MAPK
ALK
Cytochromes P450
Aurora Kinase
HER
HIV Protease
Bcl-2 Family
Antibiotic
Mitophagy
IL Receptor
Influenza Virus
c-RET
Antifungal
Gamma-secretase
Mdm2
PDK
STING
E1/E2/E3 Enzyme
HIF
Pim
Hedgehog/Smoothened
PD-1/PD-L1
PKC
Virus Protease
Interleukin
Dehydrogenase
Lipoxygenase
Casein Kinase
PKA
Calcium Channel
NO Synthase
PI4K
FAK
IκB/IKK
Prostaglandin Receptor
Topoisomerase
Beta Amyloid
c-Fms
Nrf2
Trk receptor
Epigenetic Reader Domain
Chk
PDE
NOS
Phosphatase
Tyrosinase
ROS
Sirtuin
TAM Receptor
Rho
Anti-infection
Mitochondrial Metabolism
HSV
GABA Receptor
HCV Protease
PTEN
ROCK
Syk
Drug Metabolite
PGE Synthase
Microtubule Associated
Antioxidant
PERK
Tie-2
SIK
Smo
DYRK
Sodium Channel
P-gp
Adrenergic Receptor
5-HT Receptor
Antifection
ATPase
HSP
c-Myc
Aryl Hydrocarbon Receptor
TLR
PLK
Proteasome
Integrin
CSF-1R
Glucosidase
AChR
GPCR
Ephrin Receptor
Histone Acetyltransferase
MELK
Cannabinoid Receptor
MLK
TRP/TRPV Channel
Antiviral
transporter
SGK
BTK
Estrogen/progestogen Receptor
PYK2
RIP kinase
Carbonic Anhydrase
IAP
SARS-CoV
Adenosine Receptor
IRAK
ROS Kinase
Serine/threonin kinase
Serine Protease
HBV
CCR
Cholinesterase (ChE)
Histamine Receptor
Estrogen Receptor/ERR
Cholecystokinin Receptor
GTPase
Chloride channel
Proton pump
DNA Alkylator/Crosslinker
LDL
Opioid Receptor
Retinoid Receptor
IFNAR
NOD-like Receptor (NLR)
NMDAR
Angiotensin-converting Enzyme (ACE)
DUB
MNK
Histone Methyltransferase
MRP
Androgen Receptor
Discoidin Domain Receptor (DDR)
Nucleoside Antimetabolite/Analog
ATP Citrate Lyase
Porcupine
Hippo pathway
Reductase
RAAS
DNA Alkylation
Decarboxylase
Phospholipase
cAMP
Reverse Transcriptase
NOD
Glutathione Peroxidase
Leukotriene Receptor
OXPHOS
LRRK2
Free radical scavengers
FKBP
Transferase
BACE
NADPH
Hck
Glucocorticoid Receptor
CaMK
DNA Methyltransferase
Cell Cycle Arrest
Glucokinase
Immunology/Inflammation related
RSV
S1P Receptor
Dopamine Receptor
UGT
Fatty Acid Synthase
Survivin
Aminopeptidase
DAPK
Histone Demethylase
iGluR
ABC Transporter
FAAH
GluR
CFTR
Myosin
Beta-Secretase
Acyltransferase
Progesterone Receptor
PAK
Aromatase
Gap Junction Protein
FXR
Prolyl Endopeptidase (PREP)
Pyroptosis
NADPH-oxidase
ADC Cytotoxin
Lipid
MicroRNA
ROR
Amino Acids and Derivatives
PAFR
Haspin Kinase
Hexokinase
DPP-4
Adenylyl Cyclase
LPL Receptor
MIF
PAD
Thrombopoietin Receptor
BCRP
ASK
Methionine Adenosyltransferase (MAT)
p97
Kinesin
CD38
LTR
VDA
NR4A
Monoamine Transporter
DNA
CRISPR/Cas9
Hydroxylase
Sigma receptor
Melanin-concentrating Hormone Receptor (MCHR)
NPC1L1
DHFR
TOPK
FLAP
Thioredoxin
Adenosine Deaminase
Y Box Binding Protein 1
Arginase
Na+/Ca2+ Exchanger
gp120/CD4
ASCT
Liver X Receptor
AIM2
PAI-1
RAR/RXR
MyD88
Cysteine Protease
IRE1
Guanylate cyclase
Epoxide Hydrolase
PKM
YAP
OCT
RANKL/RANK
Na-K-Cl cotransporter
ACK1
hCE
LPA Receptor
BMI-1
Thrombin
Monoamine Oxidase

Keywords