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TargetMol | Compound Library

抗胰腺癌化合物库现货

Anti-Pancreatic Cancer Compound Library

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产品编号 L2192

随着医学技术的进步,大部分癌症的生存率都在提高,例如乳腺癌,结直肠癌等肿瘤,近几十年来,生存率得到了大幅度的提升。但是,有一个例外,那就是胰腺癌,胰腺癌是一种发病隐匿,进展迅速,治疗效果和预后极差的消化道恶性肿瘤。胰腺癌的生存率一直停滞不前,胰腺癌的五年生存率只有5%至10%,绝大部分患者在诊断胰腺癌半年内死亡,由于生存率低,死亡率高,胰腺癌称为癌中之王。

为了满足胰腺癌研究客户的需求,TargeMol 收集了 2508 种与胰腺癌相关的化合物,作用于 KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等胰腺癌相关靶点,助力胰腺癌治疗药物的开发。

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产品编号 L2192

抗胰腺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品特点 产品特点

  • 2508种与胰腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 靶点含KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
EGFR
CDK
COX
VEGFR
Ras
Akt
PPAR
Wnt/beta-catenin
mTOR
JAK
ERK
STAT
HDAC
PARP
Src
Endogenous Metabolite
p38 MAPK
GSK-3
Antibacterial
AMPK
FGFR
Raf
ROS
c-Met/HGFR
PDGFR
MDM-2/p53
FLT
Caspase
TGF-beta/Smad
Parasite
Kras
p53
JNK
c-Kit
MEK
Reactive Oxygen Species
MMP
TNF
DNA/RNA Synthesis
Potassium Channel
IGF-1R
S6 Kinase
Tyrosine Kinases
Bcr-Abl
HIF/HIF Prolyl-Hydroxylase
DNA-PK
Interleukin
Bcl-2 Family
MAPK
ATM/ATR
Ferroptosis
Cytochromes P450
Aurora Kinase
ALK
HIV Protease
HER
NO Synthase
Antibiotic
Mitophagy
Influenza Virus
Gamma-secretase
IL Receptor
c-RET
Mdm2
Antifungal
STING
PDK
PD-1/PD-L1
Pim
PKC
E1/E2/E3 Enzyme
Hedgehog/Smoothened
HIF
Dehydrogenase
Virus Protease
Calcium Channel
Prostaglandin Receptor
Lipoxygenase
Nrf2
Beta Amyloid
FAK
PKA
Casein Kinase
IκB/IKK
PI4K
Topoisomerase
c-Fms
PDE
Epigenetic Reader Domain
Trk receptor
NOS
Chk
Phosphatase
HSV
Tyrosinase
Rho
Adrenergic Receptor
Mitochondrial Metabolism
TLR
Sirtuin
Anti-infection
TAM Receptor
HCV Protease
PERK
ROCK
PTEN
P-gp
GABA Receptor
Sodium Channel
Antioxidant
DYRK
Tie-2
c-Myc
SIK
Drug Metabolite
Smo
PGE Synthase
HSP
5-HT Receptor
PLK
Syk
Microtubule Associated
ATPase
Integrin
Adenosine Receptor
Aryl Hydrocarbon Receptor
IAP
Antifection
Ephrin Receptor
AChR
MLK
GPCR
Proteasome
Serine Protease
TRP/TRPV Channel
CSF-1R
RIP kinase
Glucosidase
CaMK
Antiviral
SARS-CoV
Histone Acetyltransferase
transporter
MELK
SGK
Cannabinoid Receptor
BTK
Carbonic Anhydrase
Estrogen/progestogen Receptor
IFNAR
Estrogen Receptor/ERR
Serine/threonin kinase
PYK2
glycosidase
Survivin
IRAK
ROS Kinase
NOD-like Receptor (NLR)
Chloride channel
Proton pump
Transferase
Histone Methyltransferase
DNA Alkylator/Crosslinker
Reductase
Histamine Receptor
GTPase
HBV
Cholecystokinin Receptor
Hck
LDL
Opioid Receptor
CCR
Cholinesterase (ChE)
Retinoid Receptor
Dopamine Receptor
BACE
Histone Demethylase
NADPH
RAAS
Glutathione Peroxidase
MRP
Nucleoside Antimetabolite/Analog
Leukotriene Receptor
Glucocorticoid Receptor
UGT
NMDAR
Fatty Acid Synthase
DNA Alkylation
Angiotensin-converting Enzyme (ACE)
cAMP
DUB
Androgen Receptor
ATP Citrate Lyase
OXPHOS
MNK
Porcupine
LRRK2
Free radical scavengers
Decarboxylase
Hippo pathway
FKBP
Reverse Transcriptase
Phospholipase
Discoidin Domain Receptor (DDR)
DNA Methyltransferase
NOD
ADC Cytotoxin
Progesterone Receptor
Cell Cycle Arrest
FXR
Glucokinase
RANKL/RANK
Immunology/Inflammation related
iGluR
Prolyl Endopeptidase (PREP)
Myosin
ABC Transporter
Monoamine Transporter
PAK
FAAH
GluR
Lipid
Beta-Secretase
Acyltransferase
Aminopeptidase
Pyroptosis
RSV
Aromatase
Gap Junction Protein
DAPK
NADPH-oxidase
CFTR
Kinesin
S1P Receptor
Melanin-concentrating Hormone Receptor (MCHR)
MicroRNA
Adenylyl Cyclase
NPC1L1
RAR/RXR
CD38
DHFR
ROR
Amino Acids and Derivatives
MyD88
Y Box Binding Protein 1
YAP
Arginase
LPL Receptor
LTR
Na+/Ca2+ Exchanger
gp120/CD4
MIF
TOPK
VDA
OCT
ASCT
Cysteine Protease
Liver X Receptor
NR4A
IRE1
FLAP
PAFR
Haspin Kinase
FABP
Na-K-Cl cotransporter
Hexokinase
Guanylate cyclase
DPP-4
Thioredoxin
ACK1
PAD
Epoxide Hydrolase
Cadherin
Thrombopoietin Receptor
DNA
BCRP
AIM2
ASK
hCE
PAI-1
Methionine Adenosyltransferase (MAT)
LPA Receptor
CRISPR/Cas9
Hydroxylase
Adenosine Deaminase
BMI-1
Sigma receptor
Thrombin
p97
PKM
Monoamine Oxidase

Keywords