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抗心血管疾病化合物库

抗心血管疾病化合物库

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产品编号 L5400 Anti-Cardiovascular Disease Compound Library
  库化合物信息   Excel SDF

心血管疾病泛指由于动脉粥样硬化、高脂血症、血液黏稠、高血压等所导致的心脏、大脑及全身组织发生的缺血性或出血性疾病,例如心绞痛、心肌梗塞、中风等,是全球死亡的首要原因。不同类型疾病的发病机制不同,各种抗氧化、抗高血脂、抗缺血、抑制血小板聚集和抗炎物质都具有降低心血管疾病风险的作用。某些天然产物具有抑制粘附分子、细胞因子和趋化因子基因表达,抑制血小板功能,增强内皮细胞一氧化氮释放,抑制平滑肌活化的作用,这些化合物都是心血管疾病药物筛选中的重要工具。

TargetMol 抗心血管疾病化合物库是由 1428 个心血管疾病相关的化合物组成的综合筛选库,用于心血管疾病的相关研究和高通量高内涵筛选。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 1428种心血管疾病相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括膜转运体、离子通道等心血管疾病相关靶点;
  • 大部分产品是经FDA、EMA或NMPA批准上市的药物,是研究心血管相关疾病的有效工具;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L5400)
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客户使用化合物库发表的文献

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化合物库组成

Autophagy (162)
VEGFR (157)
Calcium Channel (152)
Apoptosis (150)
Adrenergic Receptor (141)
COX (96)
Endogenous Metabolite (91)
Sodium Channel (85)
PDE (75)
PDGFR (58)
TNF (57)
5-HT Receptor (48)
TGF-beta/Smad (48)
Antibacterial (46)
RAAS (45)
AChR (43)
Potassium Channel (42)
Dopamine Receptor (40)
c-Kit (39)
FLT (37)
FGFR (37)
NF-κB (36)
IL Receptor (35)
Reactive Oxygen Species (32)
PARP (29)
CDK (26)
MMP (25)
Histamine Receptor (25)
PPAR (22)
Parasite (22)
PKC (21)
JAK (20)
ALK (20)
Ferroptosis (18)
Antibiotic (18)
c-Met/HGFR (18)
IGF-1R (18)
EGFR (17)
c-RET (16)
ATPase (16)
Src (16)
Carbonic Anhydrase (16)
P450 (16)
p38 MAPK (16)
Prostaglandin Receptor (15)
Mitophagy (15)
Adenosine Receptor (15)
Thrombin (15)
HIV Protease (15)
Norepinephrine (14)
HMG-CoA Reductase (14)
Antifungal (14)
Endothelin Receptor (13)
NO Synthase (13)
DNA/RNA Synthesis (13)
Influenza Virus (13)
ERK (12)
Raf (11)
Akt (11)
Histone Acetyltransferase (11)
Rho (10)
P-gp (10)
Glucocorticoid Receptor (10)
Tyrosine Kinases (10)
BACE (10)
Beta Amyloid (9)
Antioxidant (9)
AMPK (9)
Drug Metabolite (9)
Serotonin Transporter (9)
GABA Receptor (9)
Aurora Kinase (8)
STAT (8)
iGluR (8)
P2Y Receptor (8)
ROS (8)
Bcr-Abl (8)
Proton pump (8)
Interleukin (8)
Guanylate cyclase (8)
MEK (8)
Beta-Secretase (8)
CaMK (8)
ROCK (7)
Virus Protease (7)
Topoisomerase (7)
GSK-3 (7)
HIF/HIF Prolyl-Hydroxylase (7)
TAM Receptor (7)
NMDAR (7)
Phospholipase (7)
PI3K (7)
MRP (7)
TRP/TRPV Channel (7)
PKA (7)
Ras (7)
HDAC (6)
c-Fms (6)
Factor Xa (6)
Trk receptor (6)
IκB/IKK (6)
Nrf2 (6)
Caspase (6)
Dehydrogenase (6)
Tyrosinase (6)
Acetyl-CoA Carboxylase (6)
mTOR (5)
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Monoamine Oxidase (4)
Epigenetic Reader Domain (4)
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MAO (4)
BCL (4)
Serine Protease (4)
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RSV (4)
Chk (4)
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Estrogen/progestogen Receptor (4)
PGE Synthase (3)
PDK (3)
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MLK (3)
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transporter (2)
Protease-activated Receptor (2)
Sirtuin (2)
Antifection (2)
PYK2 (2)
Androgen Receptor (2)
DHFR (2)
RIP kinase (2)
Gap Junction Protein (2)
LRRK2 (2)
Xanthine Oxidase (2)
NADPH-oxidase (2)
HBV (2)
Na+/Ca2+ Exchanger (2)
Na-K-Cl cotransporter (2)
Myosin (2)
Integrin (2)
Monoamine Transporter (2)
IRE1 (2)
HCV Protease (2)
LDL (2)
PAFR (2)
MAPK (2)
Lipid (2)
Vasopressin Receptor (1)
BTK (1)
ACK (1)
VDAC (1)
Sigma receptor (1)
IRAK (1)
BCRP (1)
ATP Citrate Lyase (1)
ASK (1)
Aryl Hydrocarbon Receptor (1)
Adiponectin receptor (1)
Melanocortin Receptor (1)
UGT (1)
Thrombopoietin Receptor (1)
Isocitrate Dehydrogenase (IDH) (1)
Anion Exchanger (1)
N-Acetylglucosaminyltransferase (1)
Amylase (1)
TOPK (1)
Aminopeptidase (1)
Transferase (1)
Adenylyl cyclase (1)
Ligands for Target Protein for PROTAC (1)
Lipase (1)
Antiviral (1)
PAI-1 (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
GPCR19 (1)
NPC1L1 (1)
DNA-PK (1)
Hedgehog/Smoothened (1)
PKM (1)
HCN Channel (1)
DprE1 (1)
Phosphatase (1)
DNA gyrase (1)
FAAH (1)
GlyT (1)
Glucokinase (1)
Free radical scavengers (1)
PAD (1)
Gamma-secretase (1)
Progesterone Receptor (1)
Histone Methyltransferase (1)
cell cycle arrest (1)
Reductase (1)
CRISPR/Cas9 (1)
ROR (1)
Immunology/Inflammation related (1)
CXCR (1)
Cysteine Protease (1)
Retinoid Receptor (1)
Decarboxylase (1)
HSP (1)
Neurokinin receptor (1)
Discoidin Domain Receptor (DDR) (1)
DNA (1)
Pyroptosis (1)
IFNAR (1)
IAP (1)
PLK (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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