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TargetMol | Compound Library

抗心血管疾病化合物库现货

Anti-Cardiovascular Disease Compound Library

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产品编号 L5400

心血管疾病泛指由于动脉粥样硬化、高脂血症、血液黏稠、高血压等所导致的心脏、大脑及全身组织发生的缺血性或出血性疾病,例如心绞痛、心肌梗塞、中风等,是全球死亡的首要原因。不同类型疾病的发病机制不同,各种抗氧化、抗高血脂、抗缺血、抑制血小板聚集和抗炎物质都具有降低心血管疾病风险的作用。某些天然产物具有抑制粘附分子、细胞因子和趋化因子基因表达,抑制血小板功能,增强内皮细胞一氧化氮释放,抑制平滑肌活化的作用,这些化合物都是心血管疾病药物筛选中的重要工具。 TargetMol 抗心血管疾病化合物库是由 1793 个心血管疾病相关的化合物组成的综合筛选库,用于心血管疾病的相关研究和高通量高内涵筛选。

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产品编号 L5400

抗心血管疾病化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 1793种心血管疾病相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括膜转运体、离子通道等心血管疾病相关靶点;
  • 大部分产品是经FDA、EMA或NMPA批准上市的药物,是研究心血管相关疾病的有效工具;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Adrenergic Receptor
Calcium Channel
PDE
Apoptosis
Autophagy
VEGFR
COX
Sodium Channel
Endogenous Metabolite
Potassium Channel
5-HT Receptor
AChR
RAAS
PDGFR
Dopamine Receptor
TNF
Antibacterial
NF-κB
IL Receptor
Histone Acetyltransferase
FGFR
c-Kit
FLT
PARP
Histamine Receptor
PPAR
CDK
Parasite
HMG-CoA Reductase
BACE
EGFR
Antioxidant
Adenosine Receptor
Factor Xa
PKC
Reactive Oxygen Species
Epigenetic Reader Domain
Cytochromes P450
Carbonic Anhydrase
JAK
IGF-1R
ATPase
Antibiotic
Src
p38 MAPK
c-Met/HGFR
Mitophagy
c-RET
Thrombin
Antifungal
Influenza Virus
ERK
Norepinephrine
P2Y Receptor
Phospholipase
HIV Protease
Ferroptosis
Glucocorticoid Receptor
Akt
Beta-Secretase
PI3K
TRP/TRPV Channel
Drug Metabolite
DNA/RNA Synthesis
P-gp
ROS
Guanylate cyclase
Lipoxygenase
CaMK
Prostaglandin Receptor
Beta Amyloid
HDAC
GABA Receptor
NO Synthase
MRP
PKA
Raf
Nrf2
STAT
Proteasome
Integrin
GSK-3
Tyrosine Kinases
ROCK
iGluR
Bcr-Abl
NMDAR
Aurora Kinase
Acetyl-CoA Carboxylase
MEK
Proton pump
Dehydrogenase
CETP
Virus Protease
Serotonin Transporter
Serine/threonin kinase
MAO
Topoisomerase
Angiotensin-converting Enzyme (ACE)
Interleukin
SARS-CoV
c-Fms
AMPK
Hydroxylase
NOD
Tyrosinase
Chloride channel
NADPH
Serine Protease
Caspase
LDL
P2X Receptor
Mitochondrial Metabolism
GluR
Acyltransferase
Trk receptor
IκB/IKK
TAM Receptor
HIF/HIF Prolyl-Hydroxylase
Monoamine Oxidase
NOS
Glutathione Peroxidase
Wnt/beta-catenin
Nucleoside Antimetabolite/Analog
Liver X Receptor
Opioid Receptor
DPP-4
HSV
Cholinesterase (ChE)
Chk
Epoxide Hydrolase
PGE Synthase
Ephrin Receptor
Neprilysin
HIF
Anti-infection
Sigma receptor
Protease-activated Receptor
NOD-like Receptor (NLR)
Imidazoline Receptor
p53
Thyroid hormone receptor(THR)
Estrogen/progestogen Receptor
Arginase
DNA Alkylator/Crosslinker
Na+/Ca2+ Exchanger
JNK
Tie-2
FXR
CSF-1R
Myosin
Na-K-Cl cotransporter
HCN Channel
Fatty Acid Synthase
Endothelin Receptor
cAMP
mTOR
TLR
Bcl-2 Family
transporter
ALK
RSV
Reverse Transcriptase
PDK
Platelet aggregation
Syk
NADPH-oxidase
S6 Kinase
Microtubule Associated
FAK
GPCR
Adenylyl Cyclase
Transferase
DHFR
ROR
Histone Methyltransferase
Amino Acids and Derivatives
LTR
Histone Demethylase
Estrogen Receptor/ERR
HBV
Rho
Antifolate
Leukotriene Receptor
PYK2
Amylase
Immunology/Inflammation related
UGT
ABC Transporter
Antifection
Monoamine Transporter
DNA Alkylation
FAAH
Xanthine Oxidase
DNA
Androgen Receptor
TGF-beta/Smad
MAPK
Aminopeptidase
Sirtuin
PAI-1
SGK
Gap Junction Protein
DNA Methyltransferase
AhR
Monocarboxylate transporter
NPC1L1
DNA-PK
HCV Protease
DprE1
YAP
Reductase
IFNAR
Lipase
PERK
TOPK
Phosphatase
Progesterone Receptor
N-Acetylglucosaminyltransferase
VDAC
Cell Cycle Arrest
Cysteine Protease
Neurotensin Receptor
Glucokinase
Aryl Hydrocarbon Receptor
IAP
IRE1
Annexin A
FLAP
RIP kinase
Adiponectin Receptor
PAFR
Gamma-secretase
GRK
DNA gyrase
GlyT
Glucosidase
Anion Exchanger
Isocitrate Dehydrogenase (IDH)
CCR
ACK1
Vasopressin Receptor
MMP
Thrombopoietin Receptor
Indoleamine 2,3-Dioxygenase (IDO)
ATP Citrate Lyase
Lipid
BCRP
OAT
Antiviral
HSP
Decarboxylase
ASK
Casein Kinase
GST
Retinoid Receptor
Aromatase
CRISPR/Cas9
RXFP receptor
PLK
Cannabinoid Receptor
Discoidin Domain Receptor (DDR)
IRAK
Ras
p97
CFTR
MLK
PKM
HER
S1P Receptor
ADC Cytotoxin
Sodium-dependent phosphate transporter
Vitamin
BTK

Supporting Files | TargetMol 化合物库信息

Empty99899-45-399755-59-699-66-199599-78-799522-79-999-50-399429-64-899254-95-298769-84-7987-65-5Empty
SM-2470Rotigotine-Valproic AcidE 0747PranidipineProtocatechuic acidEthyl 4-chloro-2-oxo-1,2-dihydroquinoline-3-carboxylateMcN5691Reboxetine mesylateATP disodium salt
Empty98717-15-898625-26-4985-12-698410-36-797657-92-697240-79-4969-33-596847-55-196843-99-196480-44-3Empty
Ropivacaine hydrochloride(S)-(-)-Bay-K-8644Drotaverine hydrochloridePalatrigineLatrepirdine dihydrochlorideTopiramateCyproheptadine hydrochlorideDextromilnacipranT-0509Bisaramil hydrochloride
Empty964-52-396441-14-496087-21-795853-92-295635-56-695635-55-5955371-66-1955272-06-795445-79-7953778-63-7Empty
Moxisylyte hydrochlorideLabetalone hydrochlorideStylopine hydrochlorideCGS 15435Ranolazine dihydrochlorideRanolazineVK-II-36GKT136901FPL-62129TTA-A2
Empty953778-58-0952021-60-295153-31-4951151-97-6949912-58-7948-60-7947620-48-6947331-05-7945755-56-6945619-74-9Empty
SuvecaltamidePF 477736PerindoprilatJNJ-38158471RemodelinPterine-6-carboxylic acidLotamilastAllisartan IsoproxilXL019OPHIOPOGONIN D
Empty945614-12-0944261-79-4944241-52-5943319-70-8942655-44-994-25-794238-00-3942206-85-1941678-49-594-09-7Empty
PexmetinibA-803467CarbodenafilPonatinibJK-P3ButambenGardenia yellowGSK1016790ARuxolitinibBenzocaine
Empty940954-41-694-07-593957-54-1937782-05-3936623-90-4936539-80-9936500-94-6936091-26-8934353-76-1934240-30-9Empty
BI-1935SynephrineFluvastatinDifamilastSacubitril/ValsartanBetrixaban maleateElinogrelFedratinibENMD-2076Raxatrigine
Empty93392-97-393379-54-5932749-62-793035-32-6929915-58-292953-10-1928037-13-2927880-90-892-78-4927691-21-2Empty
KT-362 free base(S)-(-)-AtenololHistone Acetyltransferase Inhibitor IITamolarizineDG051Clofilium tosylateGolvatinibRAF265Naphthol AS-EPQ-10
Empty92532-23-5923981-14-0923359-38-0923262-96-892302-55-192134-98-0920509-32-6919351-41-091-75-891-64-5Empty
REV 5901ACentanafadine hydrochlorideSAR407899SAR407899 hydrochlorideDevapamilFosphenytoin disodiumResmetiromAZD1283AntazolineCoumarin

Keywords