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TargetMol | Compound Library

抗心血管疾病化合物库现货

Anti-Cardiovascular Disease Compound Library
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货号 L5400

心血管疾病泛指由于动脉粥样硬化、高脂血症、血液黏稠、高血压等所导致的心脏、大脑及全身组织发生的缺血性或出血性疾病,例如心绞痛、心肌梗塞、中风等,是全球死亡的首要原因。不同类型疾病的发病机制不同,各种抗氧化、抗高血脂、抗缺血、抑制血小板聚集和抗炎物质都具有降低心血管疾病风险的作用。某些天然产物具有抑制粘附分子、细胞因子和趋化因子基因表达,抑制血小板功能,增强内皮细胞一氧化氮释放,抑制平滑肌活化的作用,这些化合物都是心血管疾病药物筛选中的重要工具。

TargetMol 抗心血管疾病化合物库是由 1793 个心血管疾病相关的化合物组成的综合筛选库,用于心血管疾病的相关研究和高通量高内涵筛选。

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货号 L5400

抗心血管疾病化合物库

规格

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 1793种心血管疾病相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括膜转运体、离子通道等心血管疾病相关靶点;
  • 大部分产品是经FDA、EMA或NMPA批准上市的药物,是研究心血管相关疾病的有效工具;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Adrenergic Receptor
Apoptosis
Calcium Channel
PDE
Autophagy
VEGFR
Endogenous Metabolite
COX
Sodium Channel
Potassium Channel
NF-κB
Antibacterial
5-HT Receptor
TNF
AChR
ROS
PDGFR
RAAS
Dopamine Receptor
Parasite
Angiotensin-converting Enzyme (ACE)
FGFR
c-Kit
IL Receptor
p38 MAPK
Histamine Receptor
Interleukin
PARP
Histone Acetyltransferase
FLT
Reactive Oxygen Species
PPAR
Drug Metabolite
ERK
Akt
CDK
NO Synthase
Cytochromes P450
HMG-CoA Reductase
EGFR
PKC
Adenosine Receptor
Factor Xa
DNA/RNA Synthesis
Antifungal
JAK
Epigenetic Reader Domain
BACE
Antioxidant
PI3K
Antibiotic
Influenza Virus
Carbonic Anhydrase
IGF-1R
Prostaglandin Receptor
Src
Ferroptosis
c-Met/HGFR
Mitophagy
ATPase
Caspase
Norepinephrine
HIV Protease
JNK
Beta-Secretase
c-RET
TRP/TRPV Channel
Thrombin
Nrf2
PKA
Phospholipase
Glucocorticoid Receptor
STAT
NOD-like Receptor (NLR)
P2Y Receptor
SARS-CoV
CaMK
Beta Amyloid
Wnt/beta-catenin
iGluR
Cholinesterase (ChE)
HDAC
P-gp
GABA Receptor
GSK-3
Lipoxygenase
Mitochondrial Metabolism
Proteasome
Integrin
AMPK
Raf
Virus Protease
Guanylate cyclase
MRP
MEK
Anti-infection
Monoamine Oxidase
NMDAR
c-Fms
Bcr-Abl
Dehydrogenase
ROCK
Tyrosine Kinases
Hydroxylase
Tyrosinase
Serine Protease
Serotonin Transporter
LDLR
Aurora Kinase
NADPH
Proton pump
Glutathione Peroxidase
Serine/threonin kinase
Topoisomerase
Acetyl-CoA Carboxylase
Liver X Receptor
MAO
NOD
MMP
Tie-2
IκB/IKK
Microtubule Associated
CETP
PERK
Nucleoside Antimetabolite/Analog
HSV
GluR
mTOR
Chloride channel
FXR
LDL
Opioid Receptor
TLR
Na+/Ca2+ Exchanger
Amino Acids and Derivatives
Trk receptor
HIF/HIF Prolyl-Hydroxylase
TGF-beta/Smad
Acyltransferase
TAM Receptor
P2X Receptor
Fatty Acid Synthase
FAK
Sigma receptor
Imidazoline Receptor
NOS
Epoxide Hydrolase
GPCR
cAMP
Ephrin Receptor
Bcl-2 Family
HIF
DPP-4
Chk
MAPK
RSV
Ras
Myosin
HSP
Neprilysin
PGE Synthase
Protease-activated Receptor
Na-K-Cl cotransporter
Lipid
transporter
S6 Kinase
ABC Transporter
Sirtuin
MTP
DNA Alkylator/Crosslinker
Leukotriene Receptor
NADPH-oxidase
p53
Arginase
HCN Channel
PAI-1
ALK
Reverse Transcriptase
MDM-2/p53
Platelet aggregation
Immunology/Inflammation related
Syk
Thyroid hormone receptor(THR)
Reductase
Estrogen Receptor/ERR
CSF-1R
Endothelin Receptor
Histone Methyltransferase
RIP kinase
UGT
Androgen Receptor
Vitamin
Transferase
IFNAR
Necroptosis
Annexin A
PDK
SGK
DNA Methyltransferase
AhR
Factor VIIa
LTR
Histone Demethylase
Monoamine Transporter
FAAH
CCR
glycosidase
DNA
Casein Kinase
CFTR
Monocarboxylate transporter
Phosphatase
Amylase
Prolyl Endopeptidase (PREP)
Xanthine Oxidase
OXPHOS
FKBP
MLK
Rho
Gap Junction Protein
IRAK
ROR
Gamma-secretase
GPCR19
DHFR
Glucosidase
DNA Alkylation
Estrogen/progestogen Receptor
LPL Receptor
Antifolate
PYK2
Adenylate cyclase
Antifection
Thrombopoietin Receptor
Aminopeptidase
ASK
PGC-1α
YAP
OCT
IDO
GRK
Arp2/3 Complex
ACK1
SGLT
Antiviral
N-Acetylglucosaminyltransferase
HBV
VDAC
IAP
Photosystem (PS)
Adiponectin Receptor
Anion Exchanger
ATP Citrate Lyase
Kras
CRISPR/Cas9
HER
HCV Protease
DprE1
Cysteine Protease
Aryl Hydrocarbon Receptor
IRE1
DNA gyrase
CXCR
STING
LRRK2
Retinoid Receptor
RXFP receptor
Cannabinoid Receptor
PKM
Progesterone Receptor
CaSR
Isocitrate Dehydrogenase (IDH)
Vasopressin Receptor
AIM2
GST
Aromatase
ROS Kinase
Lipase
Cell Cycle Arrest
Glucokinase
PAFR
OAT
PLK
Tight Junction Protein
S1P Receptor
NPC1L1
DNA-PK
TOPK
FLAP
Hedgehog/Smoothened
Decarboxylase
MIF
Neurotensin Receptor
GlyT
Indoleamine 2,3-Dioxygenase (IDO)
BCRP
Cuproptosis
Discoidin Domain Receptor (DDR)
p97
ADC Cytotoxin
Sodium-dependent phosphate transporter
BTK

Keywords