规格

价格

库存

数量

1 mg

¥ 1,790

现货

5 mg

¥ 3,880

现货

10 mg

¥ 5,530

现货

25 mg

¥ 8,280

现货

50 mg

¥ 10,900

现货

100 mg

¥ 14,800

现货

1 mL x 10 mM (in DMSO)

¥ 3,830

现货

生物活性

产品描述	EPZ-719 is a selective and orally available SETD2 inhibitor (IC50 = 0.005 μM), with anti-cancer activity, and can be used for hematological malignancies.
靶点活性	SETD2:0.005 μM
体内活性	EPZ-719(14 天)在KMS34和KMS11细胞中能够抑制细胞的增殖，IC50值分别为0.025 μM、0.211μM[1]。
别名	EPZ719, EPZ 719

化学信息

分子量	450.57
分子式	C₂₂H₃₁FN₄O₃S
CAS No.	2697176-16-0
Smiles	FC1=C2C(NC(C(N[C@H]3C[C@H](CCC3)N4C[C@@H](N(S(C)(=O)=O)C)CC4)=O)=C2)=C(C)C=C1
密度	1.33 g/cm3 (Predicted)
颜色	White
物理性状	Solid

储存&溶解度

存储

store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

溶解度信息

DMSO: 40 mg/mL (88.78 mM), Sonication is recommended.

溶液配制表

DMSO