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PPI抑制剂库

PPI抑制剂库

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产品编号 L9400 PPI Inhibitor Library
  库化合物信息   Excel SDF

蛋白-蛋白相互作用(PPI)在生物过程中扮有非常重要的角色,是生物信息调控的主要实现方式,并且与人类疾病息息相关。在传统药物的作用中,药物靶标通常为酶或受体,而蛋白-蛋白相互作用为我们展示了一类新的、重要的疾病治疗切入点。目前,作用于蛋白-蛋白相互作用小分子抑制剂的研究已经取得了一些进展,其中有的化合物已被应用于临床研究。同时随着越来越多的蛋白-蛋白复合物晶体结构的解析,将为新型小分子抑制剂的发现奠定基础。

TaregtMol PPI 抑制剂库收集了 490 种已知活性的 PPI 相关的抑制剂,可以用于蛋白-蛋白相互作用相关的研究。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 490种已知活性的PPI相关的抑制剂,可用于高通量、高内涵筛选;
  • 作用靶点包含PD-1/PD-L1、Bcl-2、BET bromodomain、BRD4 bromodomain等;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/ LCMS多重检测,保证产品结构准确,纯度高,保障实验顺利进行。

化合物库定制

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包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L9400)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Epigenetic Reader Domain (111)
Apoptosis (78)
BCL (72)
Autophagy (38)
Nrf2 (34)
p53 (25)
Mdm2 (23)
HIV Protease (23)
E1/E2/E3 Enzyme (22)
Histone Methyltransferase (16)
Caspase (15)
PD-1/PD-L1 (14)
IAP (13)
NF-κB (12)
Ferroptosis (11)
Endogenous Metabolite (11)
RIP kinase (10)
Ras (9)
Wnt/beta-catenin (9)
DNA/RNA Synthesis (9)
PARP (8)
Histone Acetyltransferase (8)
Microtubule Associated (7)
p38 MAPK (7)
c-Myc (6)
COX (6)
STAT (6)
Sirtuin (6)
Akt (5)
TNF (5)
Antibacterial (5)
Parasite (5)
CDK (5)
Raf (5)
Rho (5)
IL Receptor (4)
Integrin (4)
JNK (4)
ERK (4)
PROTACs (4)
Dehydrogenase (4)
Ligand for E3 Ligase (4)
NMDAR (3)
Reactive Oxygen Species (3)
mTOR (3)
Sodium Channel (3)
Mitophagy (3)
PPAR (3)
Ligands for Target Protein for PROTAC (3)
PKC (3)
PI3K (3)
HIF/HIF Prolyl-Hydroxylase (3)
HSP (3)
PERK (3)
P-gp (3)
YAP (3)
HIF (3)
CXCR (3)
Carboxypeptidase (2)
Estrogen/progestogen Receptor (2)
Dopamine Receptor (2)
DNA-PK (2)
DNA Alkylator/Crosslinker (2)
PDE (2)
Phosphatase (2)
PLK (2)
Calcium Channel (2)
GABA Receptor (2)
Reverse Transcriptase (2)
Aryl Hydrocarbon Receptor (2)
Antioxidant (2)
Antifungal (2)
Src (2)
Antibiotic (2)
TLR (2)
Virus Protease (2)
NEDD8 (2)
5-HT Receptor (2)
Influenza Virus (2)
HDAC (2)
GSK-3 (2)
Lipoxygenase (2)
iGluR (2)
Integrase (2)
GTPase (2)
JAK (2)
IFNAR (2)
IκB/IKK (2)
IGF-1R (1)
ATPase (1)
Retinoid Receptor (1)
SARS-CoV (1)
ATTECs (1)
Beta Amyloid (1)
RAAS (1)
Proton pump (1)
Prostaglandin Receptor (1)
ROS (1)
Liver X Receptor (1)
Serine/threonin kinase (1)
Topoisomerase (1)
AhR (1)
Hedgehog/Smoothened (1)
VEGFR (1)
UGT (1)
Tyrosinase (1)
transporter (1)
Androgen Receptor (1)
Serotonin Transporter (1)
Thrombin (1)
TGF-beta/Smad (1)
STING (1)
HCV Protease (1)
HMG-CoA Reductase (1)
Smo (1)
GPCR19 (1)
Anti-infection (1)
CCR (1)
Potassium Channel (1)
Neurokinin receptor (1)
Gamma-secretase (1)
Mitochondrial Metabolism (1)
FXR (1)
MLK (1)
MMP (1)
MNK (1)
Molecular Glues (1)
Monoamine Oxidase (1)
Monoamine Transporter (1)
FAK (1)
MyD88 (1)
Myosin (1)
NADPH (1)
Glucokinase (1)
Neurotensin Receptor (1)
MAO (1)
DNA (1)
Chloride channel (1)
Glutathione Peroxidase (1)
Cysteine Protease (1)
PDK (1)
Interleukin (1)
Discoidin Domain Receptor (DDR) (1)
DNA Methyltransferase (1)
AChE (1)
Histamine Receptor (1)
GluR (1)
Ephrin Receptor (1)
NPC1L1 (1)
NO Synthase (1)
Estrogen Receptor/ERR (1)
P450 (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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