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Carbocisteine
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很棒纯度: 99.93%
货号 T3612Cas号 2387-59-9
别名 羧甲司坦, S-Carboxymethyl-L-cysteine, Mucodyne, Carbocysteine, Broncodeterge
Carbocisteine (Mucodyne) 常被用作具有粘液溶解和祛痰作用的抗感染鼻喷雾剂。
其他形式的 “Carbocisteine”:
Carbocisteine
一键复制产品信息 很棒纯度: 99.93%
货号 T3612 别名 羧甲司坦, S-Carboxymethyl-L-cysteine, Mucodyne, Carbocysteine, BroncodetergeCas号 2387-59-9
Carbocisteine (Mucodyne) 常被用作具有粘液溶解和祛痰作用的抗感染鼻喷雾剂。
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 500 mg | ¥ 119 | 现货 | |
| 1 g | ¥ 197 | 现货 | |
| 5 g | ¥ 458 | 现货 |
库存状态实时更新，以官网显示为准，现货产品可直接加购物车下单
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产品介绍
Carbocisteine AI Summary
Carbocisteine exhibits a diverse range of pharmacological activities. It acts as an inhibitor of the Eg5 protein by inhibiting ATP hydrolysis with an IC50 greater than 63,000 nM, and demonstrates cytotoxic activity against HeLa cells with an IC50 greater than 50,000 nM. In terms of enzyme inhibition, the compound shows no activity against human recombinant UGT1A6 and UGT1A9 enzymes.
Moderate liver toxicity is observed, indicated by elevated ALT or AST serum activity during clinical trials, although it does not cause acute liver toxicity or other specific forms of severe liver damage. Besides its weak antiviral activity against SARS-CoV-2, with a notable inhibition rate of 0.3% at 10 µM concentrations for 48 hours in Caco-2 cells and varied inhibition percentages in VERO-6 cells and 3CL-Pro protease assays, the compound also demonstrates potential inhibition of HDAC6, with enzymatic assay inhibition percentages of 17.77% and 12.71% using different substrates.
Moreover, Carbocisteine shows significant binding affinities and modulatory activities toward various neurotransmitter receptors and enzymes. This includes binding to ADRB1, ADRB2, SLC6A3, CHRNA4, HTR2C, DRD2, ADORA1, ADORA3, among others, and displaying agonistic activity at OPRM1 and DRD1 receptors, while acting antagonistically at CHRM2, HTR1A, ADRA1A, NR1I2, HTR2A, HTR2B, CNR1, rat Ar receptors, and inhibiting enzymes like PDE4D, PDE3A, MAOA, and Ptgs1.
These interactions suggest that Carbocisteine has potential bioactivity related to neurotransmitter modulation, enzyme inhibition, and antiviral effects, warranting further research into its pharmacological applications..
Note: Summary generated by AI. Data source: ChEMBL 
生物活性
化学信息
储存&溶解度
| 产品描述 | Carbocisteine (Mucodyne) is commonly used as an anti-infective nasal spray with mucolytic and expectorant effects. |
| 别名 | 羧甲司坦, S-Carboxymethyl-L-cysteine, Mucodyne, Carbocysteine, Broncodeterge |
| 分子量 | 179.19 |
| 分子式 | C5H9NO4S |
| CAS No. | 2387-59-9 |
| Smiles | N[C@@H](CSCC(O)=O)C(O)=O |
| 密度 | 1.514 g/cm3 |
| 存储 | keep away from direct sunlight | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||
| 溶解度信息 | DMSO: < 1 mg/mL (insoluble or slightly soluble)  H2O: 1 mg/mL (5.58 mM), Sonication is recommended. | |||||||||||||||
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计算器
体内实验配液计算器
请在以下方框中输入您的动物实验信息后点击计算，可以得到母液配置方法和体内配方的制备方法：
比如您的给药剂量是10 mg/kg，每只动物体重20 g，给药体积100 μL， 一共给药动物10只，您使用的配方为 10% DMSO + 40% PEG300 + 5% Tween 80 + 45% Saline / PBS / ddH2O， 那么您的工作液浓度为2 mg/mL。
母液配置方法：2 mg 药物溶于 100 μL DMSO （ 母液浓度为 20 mg/mL ）, 如您需要配置的浓度超过该产品的溶解度，请先与我们联系。
体内配方的制备方法： 取 100 μL DMSO 母液， 添加 400 μL PEG300 混匀澄清， 再加 50 μL Tween 80, 混匀澄清, 再加 450 μL Saline / PBS / ddH2O 混匀澄清
以上为“体内实验配液计算器”的使用方法举例，并不是具体某个化合物的推荐配制方式，请根据您的实验动物和给药方式选择适当的溶解方案。
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