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抗代谢疾病化合物库

抗代谢疾病化合物库

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产品编号 L5200 Anti-Metabolism Disease Compound Library
  库化合物信息   Excel SDF

代谢是指一组负责将碳水化合物、脂类和蛋白质转化为能量的生化反应,是维持内环境稳态的一个基本过程。代谢领域研究的重点是调节代谢的基本生物学机制及其在肥胖、糖尿病、心血管疾病和癌症等疾病中的作用。TargetMol 是全球知名的化合物库供应商,积极关注科研动态,为您提供大量代谢疾病研究相关的优质产品,为您的研究或相关药物筛选提供支持。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 1558个代谢疾病相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括CYP、FAAH、IDO、MAO 等代谢相关热门靶点;是研究细胞代谢及相关疾病的有效工具,例如糖尿病、肥胖、高甘油三酯血脂、高胆固醇血症等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L5200)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Autophagy (241)
Apoptosis (189)
P450 (157)
Endogenous Metabolite (128)
Dehydrogenase (85)
AMPK (81)
Antibacterial (80)
PDE (77)
PPAR (72)
PI3K (55)
Antibiotic (51)
COX (49)
Glucocorticoid Receptor (39)
MAO (37)
Reactive Oxygen Species (37)
HSP (35)
HIV Protease (34)
Ferroptosis (32)
mTOR (32)
Parasite (31)
Potassium Channel (31)
FAAH (28)
Carbonic Anhydrase (27)
Akt (27)
NF-κB (27)
Lipoxygenase (26)
Calcium Channel (25)
Proteasome (25)
Antifungal (24)
Phosphatase (24)
Mitophagy (24)
GSK-3 (24)
Retinoid Receptor (23)
Phospholipase (23)
Influenza Virus (22)
RAAS (22)
DNA/RNA Synthesis (22)
Casein Kinase (21)
HIF/HIF Prolyl-Hydroxylase (20)
Mitochondrial Metabolism (20)
Monoamine Oxidase (20)
FXR (19)
DPP-4 (18)
NADPH (17)
Glucosidase (17)
ROCK (17)
5-HT Receptor (16)
CDK (16)
Transferase (16)
AChR (15)
Adrenergic Receptor (15)
HMG-CoA Reductase (15)
SARS-CoV (14)
GPR (14)
AhR (13)
HCV Protease (13)
Indoleamine 2,3-Dioxygenase (IDO) (13)
Reductase (13)
Sodium Channel (12)
PKA (12)
Adenosine Receptor (12)
IL Receptor (12)
Virus Protease (12)
Prostaglandin Receptor (12)
ATM/ATR (12)
ERK (11)
HIF (11)
MMP (11)
PARP (11)
Fatty Acid Synthase (11)
GABA Receptor (11)
HBV (11)
Glucokinase (11)
DHFR (11)
TNF (11)
Lipase (11)
SGLT (11)
Histamine Receptor (11)
S6 Kinase (11)
DNA-PK (11)
Wnt/beta-catenin (10)
transporter (10)
PKC (10)
Tyrosinase (10)
ROR (10)
Aryl Hydrocarbon Receptor (9)
ROS (9)
Cannabinoid Receptor (9)
Hydroxylase (9)
Caspase (9)
Serine Protease (9)
Liver X Receptor (9)
Estrogen/progestogen Receptor (9)
Estrogen Receptor/ERR (9)
PDK (8)
Glutathione Peroxidase (8)
Xanthine Oxidase (8)
NO Synthase (8)
ATPase (8)
Reverse Transcriptase (8)
HSV (8)
Dopamine Receptor (8)
Isocitrate Dehydrogenase (IDH) (8)
IκB/IKK (8)
Thrombin (8)
Interleukin (8)
JNK (8)
STAT (8)
NAMPT (8)
Factor Xa (8)
AChE (8)
Antifolate (8)
Nrf2 (7)
Stearoyl-CoA Desaturase (SCD) (7)
HDAC (7)
Cysteine Protease (7)
UGT (7)
PAI-1 (7)
Glucagon Receptor (7)
Lipid (7)
Topoisomerase (7)
IDO (7)
PKM (7)
Acyltransferase (6)
TRP/TRPV Channel (6)
Opioid Receptor (6)
P-gp (6)
Phosphorylase (6)
Neprilysin (6)
Sirtuin (6)
VEGFR (6)
Aminopeptidase (6)
Src (6)
BCL (5)
iGluR (5)
Beta Amyloid (5)
Microtubule Associated (5)
MEK (5)
SGK (5)
Androgen Receptor (5)
p38 MAPK (5)
c-Met/HGFR (5)
Chloride channel (5)
CETP (5)
FLT (5)
Serine/threonin kinase (4)
JAK (4)
CCR (4)
GluR (4)
NOS (4)
Aurora Kinase (4)
CAT (4)
Anti-infection (4)
Norepinephrine (4)
DNA (4)
CaMK (4)
Leukotriene Receptor (4)
ribosome (4)
LDL (4)
TGF-beta/Smad (4)
ATP Citrate Lyase (4)
GPCR19 (4)
RSV (4)
IGF-1R (3)
Carboxypeptidase (3)
Acetyl-CoA Carboxylase (3)
OAT (3)
Decarboxylase (3)
Thyroid hormone receptor(THR) (3)
Adiponectin receptor (3)
Hexokinase (3)
SIK (3)
Annexin A (3)
TAM Receptor (3)
P2Y Receptor (3)
Antioxidant (3)
ABC (3)
Integrin (3)
Drug Metabolite (3)
Antifection (3)
FGFR (3)
BACE (3)
c-RET (3)
PERK (3)
NADPH-oxidase (3)
Ras (3)
NPC1L1 (3)
MRP (3)
Vasopressin Receptor (3)
Endothelin Receptor (3)
Histone Demethylase (2)
Sigma receptor (2)
Trk receptor (2)
ASK (2)
Amino Acids and Derivatives (2)
LTR (2)
ALK (2)
Histone Methyltransferase (2)
ROS Kinase (2)
CFTR (2)
GST (2)
MLK (2)
p53 (2)
Proton pump (2)
Progesterone Receptor (2)
Chk (2)
Antiviral (2)
Nucleoside Antimetabolite/Analog (2)
Gap Junction Protein (2)
PDGFR (2)
EGFR (2)
E1/E2/E3 Enzyme (2)
Hedgehog/Smoothened (2)
Syk (2)
PAK (2)
Glutaminase (2)
cell cycle arrest (2)
Adenosine deaminase (2)
c-Kit (2)
Epigenetic Reader Domain (2)
MAPK (2)
Rho (2)
PGC-1α (2)
Tyrosine Kinases (2)
OX Receptor (2)
Epoxide Hydrolase (2)
Neurokinin receptor (2)
HER (1)
BMI-1 (1)
Complement System (1)
c-Fms (1)
CRISPR/Cas9 (1)
Aromatase (1)
cholecystokinin (1)
LPA Receptor (1)
PI4K (1)
DNA Methyltransferase (1)
Platelet aggregation (1)
DNA Alkylation (1)
MELK (1)
IFNAR (1)
IAP (1)
Serotonin Transporter (1)
Pim (1)
VDAC (1)
N-Acetylglucosaminyltransferase (1)
CaSR (1)
Galectin (1)
Melatonin Receptor (1)
Tie-2 (1)
RAR/RXR  (1)
DYRK (1)
aconitase (1)
DNA Alkylator/Crosslinker (1)
Immunology/Inflammation related (1)
LPL Receptor (1)
Arginase (1)
YAP (1)
DprE1 (1)
stilbene oxidase (1)
Hydrogenase (1)
Monocarboxylate transporter (1)
Transaminase (1)
GSNOR (1)
Adenylyl cyclase (1)
Mdm2 (1)
advanced glycation end products (1)
CSF-1R (1)
FLAP (1)
Pyroptosis (1)
Bradykinin Receptor (1)
hCE (1)
GluCls (1)
Free radical scavengers (1)
LRRK2 (1)
TLR (1)
Glutathione reductase (1)
PGE Synthase (1)
Beta-Secretase (1)
BCRP (1)
Telomerase (1)
PAD (1)
CXCR (1)
Thioredoxin (1)
RIP kinase (1)
Bombesin Receptor (1)
MAGL (1)
PROTAC Linker (1)
Smo (1)
Guanylate cyclase (1)
Anion Exchanger (1)
Monoamine Transporter (1)
DNA gyrase (1)
NMDAR (1)
MT Receptor (1)
GRK (1)
FABP (1)
Bcr-Abl (1)
S1P Receptor (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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