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TargetMol | Compound Library

抗代谢疾病化合物库现货

Anti-Metabolism Disease Compound Library

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产品编号 L5200

代谢是指一组负责将碳水化合物、脂类和蛋白质转化为能量的生化反应,是维持内环境稳态的一个基本过程。代谢领域研究的重点是调节代谢的基本生物学机制及其在肥胖、糖尿病、心血管疾病和癌症等疾病中的作用。TargetMol 是全球知名的化合物库供应商,积极关注科研动态,为您提供大量代谢疾病研究相关的优质产品,为您的研究或相关药物筛选提供支持。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L5200

抗代谢疾病化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 1544个代谢疾病相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括CYP、FAAH、IDO、MAO 等代谢相关热门靶点;是研究细胞代谢及相关疾病的有效工具,例如糖尿病、肥胖、高甘油三酯血脂、高胆固醇血症等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

Autophagy
Apoptosis
Cytochromes P450
Endogenous Metabolite
Dehydrogenase
Antibacterial
AMPK
PDE
PPAR
PI3K
COX
Antibiotic
mTOR
Glucocorticoid Receptor
MAO
NF-κB
HSP
HIV Protease
Reactive Oxygen Species
Potassium Channel
Ferroptosis
Parasite
FAAH
Carbonic Anhydrase
Antifungal
GSK-3
Lipoxygenase
Proteasome
Akt
RAAS
Mitophagy
Calcium Channel
DNA/RNA Synthesis
Influenza Virus
Phosphatase
Casein Kinase
Retinoid Receptor
HIF/HIF Prolyl-Hydroxylase
Monoamine Oxidase
FXR
Mitochondrial Metabolism
Phospholipase
Glucagon Receptor
DPP-4
NADPH
ROCK
Glucosidase
Transferase
CDK
5-HT Receptor
Adrenergic Receptor
GPCR
SARS-CoV
AChR
HMG-CoA Reductase
IL Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Sodium Channel
DNA-PK
Reductase
Virus Protease
ATM/ATR
TNF
AhR
HCV Protease
Adenosine Receptor
Lipase
Histamine Receptor
PKA
HBV
PARP
Glucokinase
ERK
Fatty Acid Synthase
SGLT
Prostaglandin Receptor
transporter
GABA Receptor
HIF
S6 Kinase
DHFR
ROR
JNK
Wnt/beta-catenin
PKC
MMP
Tyrosinase
Estrogen/progestogen Receptor
Estrogen Receptor/ERR
Caspase
Aryl Hydrocarbon Receptor
ROS
Hydroxylase
Cannabinoid Receptor
ATPase
Glutathione Peroxidase
Factor Xa
Serine Protease
Antifolate
NAMPT
Isocitrate Dehydrogenase (IDH)
Stearoyl-CoA Desaturase (SCD)
HSV
Xanthine Oxidase
Interleukin
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IκB/IKK
Reverse Transcriptase
STAT
PDK
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Liver X Receptor
TRP/TRPV Channel
IDO
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Nrf2
PAI-1
HDAC
Thrombin
NO Synthase
Src
p38 MAPK
VEGFR
Opioid Receptor
IGF-1R
Acyltransferase
Aminopeptidase
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PKM
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c-Met/HGFR
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ATP Citrate Lyase
GPCR19
RSV
FGFR
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P2Y Receptor
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SIK
Annexin A
E1/E2/E3 Enzyme
Adiponectin Receptor
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Antifection
Hexokinase
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Endothelin Receptor
Epigenetic Reader Domain
CaMK
Androgen Receptor
EGFR
OAT
Decarboxylase
ALK
Acetyl-CoA Carboxylase
Carboxypeptidase
ribosome
c-RET
NADPH-oxidase
Ras
TAM Receptor
ADC Cytotoxin
NPC1L1
Amino Acids and Derivatives
Histone Demethylase
Progesterone Receptor
Tyrosine Kinases
Rho
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PAK
OX Receptor
Chk
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MAPK
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Trk receptor
ASK
Adenosine Deaminase
Gap Junction Protein
Neurokinin receptor
Syk
c-Kit
Sigma receptor
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CFTR
MLK
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Mdm2
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GSNOR
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stilbene oxidase
Hydrogenase
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LTR
IFNAR
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DYRK
Tie-2
Melatonin Receptor
Galectin
N-Acetylglucosaminyltransferase
CaSR
Cholecystokinin Receptor
Pim
Serotonin Transporter
CSF-1R
IAP
Immunology/Inflammation related
FLAP
RIP kinase
Bcr-Abl
FABP
GRK
MT Receptor
NMDAR
DNA gyrase
Monoamine Transporter
Anion Exchanger
Guanylate cyclase
Smo
PROTAC Linker
MAGL
DNA Alkylation
Thioredoxin
Bombesin Receptor
Bradykinin Receptor
CXCR
Telomerase
BCRP
Beta-Secretase
PGE Synthase
Glutathione reductase
TLR
LRRK2
Free radical scavengers
GluCls
hCE
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GST
c-Fms
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LPA Receptor
PI4K
CRISPR/Cas9
Complement System
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DNA Methyltransferase
BMI-1
NOD
S1P Receptor
PGC-1α

Keywords