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TargetMol | Compound Library

抗癌天然产物库现货

Anti-Tumor Natural Product Library

Rating icon 很棒
产品编号 L6700

癌症是严重危害人类健康的疾病, 从天然产物中寻找预防和治疗恶性肿瘤的活性成分始终是国内外肿瘤药物开发的热门领域,众多药物化学家们一直在致力于天然抗瘤药物的开发。随着对肿瘤发生、恶变的分子机制研究不断深入,人们以肿瘤发生发展过程中相关酶、受体为作用靶点, 筛选出一系列新的有潜在抗癌活性的天然先导化合物。据权威机构统计,从1981年至今,99种小分子抗癌药物中的79种是以天然产物为基础研制成功的,例如紫杉烷类、喜树碱类和长春碱类等热门抗肿瘤药物。天然产物是一个巨大的药物开发宝库,天然产物的研究与开发历来是人类寻找新药以及向疾病作斗争的重要手段。借助天然产物的结构先导、修饰和改造也促进了合成药物的迅速发展。

TargetMol 精心筛选1812 种来源于植物、动物或微生物的具有已知或潜在抗肿瘤活性天然产物,性价比高,能够为您提供肿瘤药物开发、天然先导化合物筛选等研究的有力工具。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L6700

抗癌天然产物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 1812种已知活性天然产物的独特集合,是肿瘤药物开发、抗癌先导化合物筛选等领域的有力工具,可用于HTS和HCS。
  • 全部产品活性已知:提供产品的生物学信息和药物学信息,为筛选提供理论方向和研究基础;
  • 来源清晰:精选来自动物、植物、微生物的已知活性天然产物;更具体到植物种属,并标注准确英文名与拉丁名,方便您的后期研究确证。
  • 信息全面:从化合物结构到溶解度,从信号通路、作用靶点到生物活性信息均有详细描述。
  • 性价比高:剔除了价格昂贵但成药性差的天然产物,让您用更少的成本得到更多高品质的天然产物。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Endogenous Metabolite
Autophagy
NF-κB
Antibacterial
COX
Reactive Oxygen Species
Antioxidant
Antibiotic
P450
TNF
Parasite
Antifungal
DNA/RNA Synthesis
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NO Synthase
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Microtubule Associated
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Immunology/Inflammation related
Dopamine Receptor
Nucleoside Antimetabolite/Analog
mTOR
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CDK
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PKA
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transporter
HCV Protease
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cell cycle arrest
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ROR
Arginase
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PAI-1
ALK
CRISPR/Cas9
PLK
FLT
NADPH-oxidase
cholecystokinin
Thrombin
ROS Kinase
CFTR
PD-1/PD-L1

Supporting Files | TargetMol 化合物库信息

Empty99-93-499-66-199353-00-199-32-199-24-1989-51-5989-30-0989-23-198891-44-2987-78-0Empty
4-HydroxyacetophenoneValproic AcidMethyl rosmarinateChelidonic acidMethyl gallate(-)-Epigallocatechin Gallate3-Epiursolic acidDeoxylimoninPseudolaric acid A-O-β-D-glucopyranosideCiticoline
Empty987-65-598665-15-798474-78-398474-74-9981-15-797938-30-297792-45-597682-44-597-65-497-59-6Empty
ATP disodium saltGanoderic acid FPseudoginsenoside RT5Pseudoginsenoside RT1AilanthoneSophoraflavanone GLappaconitine hydrobromideIrinotecanItaconic acidAllantoin
Empty97-54-197540-22-297-53-0973-67-197230-47-297230-46-197207-47-1970-74-1970-73-096990-18-0Empty
IsoeugenolS-Adenosyl-L-methionine disulfate tosylateEugenol5,6,7-TRIMETHOXYFLAVONEPicfeltarraenin IAPicfeltarraenin IBMeisoindigo(-)-Epigallocatechin(+)-GallocatechinMomordin Ic
Empty96574-01-5961-29-596087-21-795975-55-6959-23-9957-66-495311-94-795258-14-395041-90-094987-08-3Empty
Salvianolic acid AIsoliquiritigeninStylopine hydrochlorideGuggulsterone4'-MethoxychalconeIsolinderalactoneLucideric acid AYadanziolide AErianinGypenoside XLIX
Empty94805-82-094705-70-194-62-294596-28-894-53-194487-74-894-41-794356-22-694-13-394105-90-5Empty
GlycycoumarinGypenoside XLVIPiperineSenkyunolide IPiperonylic acidAngelic anhydrideChalconeRhapontigenin 3'-O-glucosidePropylparaben(±)-Equol
Empty94-07-5938-55-693772-31-793-35-693-29-893-15-293-07-292-61-591-64-591531-30-5Empty
Synephrine6-(Dimethylamino)purineNeogambogic acidUmbelliferoneIsoeugenol acetateMethyl eugenolVeratric acidScopoletinCoumarinAntineoplaston A10
Empty91432-48-391421-43-191421-42-090985-77-690-80-2906-33-2905954-18-9905954-17-890-47-190-33-5Empty
Ascamycin9-amino-CPTRubitecanGinsenoside Ra3D-(+)-Glucono-1,5-lactoneNeochlorogenic acidIsopsoralenosidePsoralenosideXanthone4-Methylumbelliferone
Empty90332-63-190-24-490-18-69008-22-490-05-189919-62-089-82-789595-71-189590-95-489-57-6Empty
10-Deacetyl-7-xylosyl paclitaxelXanthoxylinQuercetagetinLaminaranGuaiacol3,5-O-Dicaffeoylquinic acidPulegoneChamaejasmenin Bmogroside IV5-Aminosalicylic Acid

Keywords