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FASN-IN-3 是脂肪酸合酶抑制剂。


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FASN-IN-3 是脂肪酸合酶抑制剂。
| 规格 | 价格 | 库存 | 数量 | 
|---|---|---|---|
| 1 mg | ¥ 417  | In stock | |
| 5 mg | ¥ 973  | In stock | |
| 10 mg | ¥ 1,380  | In stock | |
| 25 mg | ¥ 2,290  | In stock | |
| 50 mg | ¥ 3,120  | In stock | |
| 100 mg | ¥ 4,130  | In stock | |
| 200 mg | ¥ 5,570  | In stock | |
| 1 mL x 10 mM (in DMSO) | ¥ 833  | In stock | 
FASN-IN-3 相关产品
| 产品描述 | FASN-IN-3 is an inhibitor of fatty acid synthase (FASN).  | 
| 体外活性 | 对单核细胞而言,FASN-IN-3处理后,由LTA刺激引起的IL-1 beta水平降低,然而在LPS刺激后仅轻微降低。在细胞培养中,人类PBMC与单核细胞会用脂多糖(LPS,一种Toll 4受体激动剂)或脂壁酸(LTA,一种Toll 2受体激动剂)进行刺激。无论是LPS或LTA联合DMSO(即FASN-IN-3的溶剂)的刺激,均会导致IL-1 beta的分泌。而FASN-IN-1对PBMC的处理—PBMC是包含淋巴细胞与单核细胞的混合单核细胞群—可减少由LPS或LTA刺激引起的IL-1 beta水平。  | 
| 分子量 | 384.47 | 
| 分子式 | C24H24N4O | 
| CAS No. | 2097262-60-5 | 
| Smiles | Cc1n[nH]c(c1C)-c1cc(C(=O)N2CC(C2)c2ccc(cc2)C#N)c(C)cc1C | 
| 密度 | 1.26 g/cm3 (Predicted) | 
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | ||||||||||||||||||||||||||||||
| 溶解度信息 | DMSO: 33.33 mg/mL (86.69 mM), Sonication and heating to 80℃ are recommended.   | ||||||||||||||||||||||||||||||
| 体内实验配方 | 10% DMSO+40% PEG300+5% Tween 80+45% Saline: 2 mg/mL (5.2 mM), Sonication is recommended.  请按顺序添加溶剂,在添加下一种溶剂之前,尽可能使溶液澄清。如有必要,可通过加热、超声、涡旋处理进行溶解。工作液建议现配现用。以上配方仅供参考,体内配方并不是绝对的,请根据不同情况进行调整。 | ||||||||||||||||||||||||||||||
溶液配制表  | |||||||||||||||||||||||||||||||
DMSO 
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