首页 工具
登录
抗癌药物库

抗癌药物库

产品编号 L2150 Anti-Cancer Drug Library
  库化合物信息   Excel SDF

尽管在过去的几十年中癌症的研究和治疗取得了巨大的成功,但癌症仍然是人类面临的巨大挑战,给患者身心健康带来巨大的痛苦。癌细胞具有许多显著不同的生物学特征,表现出无限的增殖潜能,维持自身生长信号的持续稳定,逃避应激信号诱导的细胞凋亡,刺激血管生长,为肿瘤提供营养,同时逃避免疫系统防御和诱导局部慢性炎症,发挥其侵袭和转移能力;并且表现出异常的代谢活动,并通过突变和表观遗传机制显著改变全基因组的稳定性。

我们挑选了2900 种具有抗癌活性或潜在抗癌活性的药物,包括上市和临床期药物,可用于具体癌症的阳性对照及不同癌症之间相关性研究,是您抗癌研究的有力工具!

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
我们的产品含有多种规格,如需了解具体的规格以及价格信息,请联系我们咨询订购,对于大额的订购,我们还有额外的优惠!
获取报价
点击图片重新获取验证码
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
获取报价
点击图片重新获取验证码

产品描述

  • 2900个具有抗癌活性小分子的独特集合,生物活性已经临床前实验证实,可用于高通量、高内涵筛选;
  • 所有化合物都具有已知且良好的生物活性、安全性和生物利用度,这些特性可显著加速药物开发和优化,是进行癌症相关研究和药物重定位有效的筛选工具;
  • 作用靶点涉及PI3K、HDAC、mTOR、CDK、JAK 等癌症相关靶点,涉及的研究领域包括肺癌、乳腺癌、白血病、淋巴瘤等15种癌症;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2150)
点击图片重新获取验证码

化合物库组成

Autophagy (442)
Apoptosis (411)
5-HT Receptor (195)
Endogenous Metabolite (183)
Adrenergic Receptor (178)
Antibacterial (147)
COX (135)
Antibiotic (120)
DNA/RNA Synthesis (119)
Dopamine Receptor (118)
Histamine Receptor (104)
Sodium Channel (95)
Calcium Channel (88)
Potassium Channel (88)
VEGFR (80)
EGFR (71)
Parasite (68)
AChR (66)
Reactive Oxygen Species (65)
PI3K (63)
Glucocorticoid Receptor (62)
P450 (59)
GABA Receptor (57)
FLT (55)
Topoisomerase (52)
PPAR (52)
PDGFR (51)
HIV Protease (51)
NF-κB (51)
CDK (50)
Ferroptosis (48)
JAK (47)
c-Kit (47)
FGFR (44)
HDAC (44)
Estrogen/progestogen Receptor (42)
Microtubule Associated (42)
Antifungal (41)
c-Met/HGFR (40)
Dehydrogenase (39)
Influenza Virus (38)
Mitophagy (38)
mTOR (38)
Estrogen Receptor/ERR (35)
Src (35)
Nucleoside Antimetabolite/Analog (34)
iGluR (32)
SARS-CoV (30)
Androgen Receptor (30)
Tyrosine Kinases (29)
Bcr-Abl (29)
Prostaglandin Receptor (28)
PDE (27)
Raf (27)
Serotonin Transporter (24)
Proton pump (23)
Akt (23)
Adenosine Receptor (23)
Norepinephrine (23)
ATPase (23)
DNA Alkylator/Crosslinker (22)
Virus Protease (22)
P-gp (21)
MEK (21)
TRP/TRPV Channel (21)
NMDAR (21)
TNF (21)
PARP (21)
HER (21)
HSV (20)
p38 MAPK (20)
HSP (19)
Aurora Kinase (19)
PKC (19)
ERK (18)
ALK (18)
Opioid Receptor (18)
Epigenetic Reader Domain (18)
ROS (18)
c-RET (18)
AMPK (17)
RAAS (17)
Trk receptor (17)
Phosphatase (16)
BCL (16)
HBV (16)
MMP (15)
HIF/HIF Prolyl-Hydroxylase (15)
GNRH Receptor (15)
TAM Receptor (15)
BTK (15)
Carbonic Anhydrase (15)
Retinoid Receptor (15)
Antifolate (14)
GSK-3 (14)
HCV Protease (14)
Drug Metabolite (14)
STAT (14)
E1/E2/E3 Enzyme (14)
Caspase (14)
DNA Alkylation (14)
Reverse Transcriptase (13)
c-Fms (13)
Mitochondrial Metabolism (13)
Histone Methyltransferase (13)
CXCR (13)
Progesterone Receptor (13)
MRP (12)
TGF-beta/Smad (12)
CFTR (12)
p53 (12)
HMG-CoA Reductase (12)
Lipoxygenase (12)
MAO (12)
DHFR (12)
IL Receptor (12)
Proteasome (12)
DNA-PK (12)
IGF-1R (11)
Transferase (11)
Chk (11)
GluR (11)
Gamma-secretase (11)
Interleukin (11)
FAK (11)
Nrf2 (10)
PKA (10)
HIF (10)
Wnt/beta-catenin (10)
Hedgehog/Smoothened (10)
Antioxidant (10)
CaMK (10)
SGLT (10)
Beta Amyloid (10)
Chloride channel (10)
ROCK (10)
CSF-1R (9)
Monoamine Oxidase (9)
DNA Methyltransferase (9)
Antifection (9)
P2X Receptor (9)
PLK (9)
GPR (9)
AChE (9)
TLR (9)
S1P Receptor (9)
ABC (8)
Sirtuin (8)
Indoleamine 2,3-Dioxygenase (IDO) (8)
Mdm2 (8)
Phospholipase (8)
S6 Kinase (8)
IAP (8)
Smo (8)
JNK (8)
Syk (8)
Neurokinin receptor (8)
DNA (7)
Sigma receptor (7)
Monoamine Transporter (7)
NADPH (7)
Thrombin (7)
LPL Receptor (7)
Guanylate cyclase (7)
P2Y Receptor (7)
ATM/ATR (7)
Endothelin Receptor (7)
Aromatase (7)
Histone Demethylase (7)
ROS Kinase (7)
Ras (7)
Integrin (7)
NO Synthase (6)
CCR (6)
RIP kinase (6)
Antiviral (6)
IκB/IKK (6)
ribosome (6)
Vasopressin Receptor (6)
PAK (6)
cholecystokinin (6)
Kinesin (6)
Isocitrate Dehydrogenase (IDH) (6)
Casein Kinase (6)
Fatty Acid Synthase (6)
Leukotriene Receptor (6)
Pim (5)
Hydroxylase (5)
Glutathione Peroxidase (5)
Tie-2 (5)
Serine Protease (5)
Ephrin Receptor (5)
LTR (5)
IFNAR (5)
FXR (5)
CaSR (5)
NOD (5)
DPP-4 (5)
PGE Synthase (5)
GPCR19 (4)
Oxytocin Receptor (4)
Xanthine Oxidase (4)
Serine/threonin kinase (4)
Melatonin Receptor (4)
Aryl Hydrocarbon Receptor (4)
KSP (4)
Aminopeptidase (4)
Amino Acids and Derivatives (4)
AhR (4)
IDO (4)
Annexin A (4)
Tyrosinase (4)
Rho (3)
OX Receptor (3)
Wee1 (3)
UGT (3)
RSV (3)
PDK (3)
Somatostatin (3)
ROR (3)
STING (3)
Reductase (3)
IRAK (3)
OAT (3)
Cannabinoid Receptor (3)
Hexokinase (3)
Liver X Receptor (3)
Free radical scavengers (3)
DNA gyrase (3)
Melanocortin Receptor (3)
Cysteine Protease (3)
CRM1 (3)
Monocarboxylate transporter (3)
MT Receptor (3)
Na-K-Cl cotransporter (3)
Adenosine deaminase (3)
NAMPT (3)
NOD-like Receptor (NLR) (3)
Beta-Secretase (2)
VDA (2)
Histone Acetyltransferase (2)
Acyltransferase (2)
GST (2)
Glutathione reductase (2)
Glucosidase (2)
GHSR (2)
Gap Junction Protein (2)
DUB (2)
Discoidin Domain Receptor (DDR) (2)
Arginase (2)
TOPK (2)
Decarboxylase (2)
ATP Citrate Lyase (2)
Imidazoline Receptor (2)
c-Myc (2)
Cell wall (2)
Telomerase (2)
CD73 (2)
CAT (2)
BCRP (2)
PYK2 (2)
YAP (2)
p97 (2)
LDL (2)
Porcupine (2)
NEDD8 (2)
Lipid (2)
MAPK (2)
PD-1/PD-L1 (2)
NOS (2)
Protease-activated Receptor (2)
IRE1 (2)
Myosin (1)
Na+/Ca2+ Exchanger (1)
Thioredoxin (1)
N-Acetylglucosaminyltransferase (1)
Thrombopoietin Receptor (1)
PAI-1 (1)
cAMP (1)
Bradykinin Receptor (1)
PAFR (1)
BMI-1 (1)
Immunology/Inflammation related (1)
PAD (1)
transporter (1)
Survivin (1)
BACE (1)
NADPH-oxidase (1)
ASK (1)
Aquaporin (1)
Neprilysin (1)
VDAC (1)
Anion Exchanger (1)
advanced glycation end products (1)
OXPHOS (1)
ACK (1)
CGRP Receptor (1)
CRFR (1)
MTH1 (1)
Glucokinase (1)
Pyroptosis (1)
Hydrogenase (1)
KLF (1)
RAR/RXR  (1)
HCN Channel (1)
Hck (1)
GTPase (1)
LHRH (1)
GRK (1)
NPC1L1 (1)
Glutaminase (1)
Lipase (1)
Glucagon Receptor (1)
Stemness kinase (1)
Platelet aggregation (1)
Galectin (1)
MALT (1)
Factor Xa (1)
FAAH (1)
DYRK (1)
SGK (1)
PI4K (1)
MELK (1)
MLK (1)
MNK (1)
PERK (1)
Complement System (1)
GlyT (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
陶术
生物
TargetMol®中国区唯一合作伙伴
点击进入陶术生物官网陶术生物
联系我们
400-820-0310

上海市静安区江场三路238号8楼