购物车
  • 全部删除
  • TargetMol
    您的购物车当前为空
TargetMol | Compound Library

抗癌药物库现货

Anti-Cancer Drug Library

Rating icon 很棒
产品编号 L2150

尽管在过去的几十年中癌症的研究和治疗取得了巨大的成功,但癌症仍然是人类面临的巨大挑战,给患者身心健康带来巨大的痛苦。癌细胞具有许多显著不同的生物学特征,表现出无限的增殖潜能,维持自身生长信号的持续稳定,逃避应激信号诱导的细胞凋亡,刺激血管生长,为肿瘤提供营养,同时逃避免疫系统防御和诱导局部慢性炎症,发挥其侵袭和转移能力;并且表现出异常的代谢活动,并通过突变和表观遗传机制显著改变全基因组的稳定性。 我们挑选了3230 种具有抗癌活性或潜在抗癌活性的药物,包括上市和临床期药物,可用于具体癌症的阳性对照及不同癌症之间相关性研究,是您抗癌研究的有力工具!

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
资源下载
化合物库相关信息
Excel
SDF
联系我们获取更多批次信息

产品编号 L2150

抗癌药物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 3230个具有抗癌活性小分子的独特集合,生物活性已经临床前实验证实,可用于高通量、高内涵筛选;
  • 所有化合物都具有已知且良好的生物活性、安全性和生物利用度,这些特性可显著加速药物开发和优化,是进行癌症相关研究和药物重定位有效的筛选工具;
  • 作用靶点涉及PI3K、HDAC、mTOR、CDK、JAK 等癌症相关靶点,涉及的研究领域包括肺癌、乳腺癌、白血病、淋巴瘤等15种癌症;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

使用TargetMol产品
发表顶级期刊文献

引用更多关于TargetMol产品的科学文献吧!

查看更多

Library Customization | TargetMol 化合物库定制

Compound Library | TargetMol
您可以通过点击按钮
定制您专属的化合物!
联系专属定制

Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
Endogenous Metabolite
Antibacterial
5-HT Receptor
Adrenergic Receptor
Dopamine Receptor
Antibiotic
DNA/RNA Synthesis
COX
Histamine Receptor
Potassium Channel
Parasite
Sodium Channel
Calcium Channel
VEGFR
EGFR
Reactive Oxygen Species
Cytochromes P450
AChR
PI3K
NF-κB
CDK
Glucocorticoid Receptor
Topoisomerase
HIV Protease
FLT
PDGFR
FGFR
JAK
PPAR
Virus Protease
c-Met/HGFR
GABA Receptor
c-Kit
HDAC
Microtubule Associated
Estrogen Receptor/ERR
Estrogen/progestogen Receptor
Ferroptosis
Antifungal
mTOR
SARS-CoV
Prostaglandin Receptor
Dehydrogenase
Nucleoside Antimetabolite/Analog
Mitophagy
iGluR
Influenza Virus
Akt
Src
Tyrosine Kinases
Androgen Receptor
Bcr-Abl
Adenosine Receptor
TNF
Caspase
Serotonin Transporter
PDE
Bcl-2 Family
Raf
p38 MAPK
HSP
GPCR
PARP
ATPase
Interleukin
Ras
TRP/TRPV Channel
HSV
Epigenetic Reader Domain
ALK
ERK
Opioid Receptor
Norepinephrine
P-gp
Aurora Kinase
HIF/HIF Prolyl-Hydroxylase
PKC
MEK
Drug Metabolite
NMDAR
MMP
HBV
Histone Methyltransferase
AMPK
HER
Proton pump
DNA Alkylator/Crosslinker
c-RET
MDM-2/p53
ROS
STAT
Phosphatase
c-Fms
RAAS
Endothelin Receptor
Trk receptor
HCV Protease
TAM Receptor
Progesterone Receptor
ROS Kinase
Mitochondrial Metabolism
FAK
GSK-3
TGF-beta/Smad
SGLT
Carbonic Anhydrase
E1/E2/E3 Enzyme
LPL Receptor
Reverse Transcriptase
IL Receptor
Chk
Beta Amyloid
Monoamine Oxidase
IGF-1R
CXCR
Retinoid Receptor
p53
PKA
DNA Alkylation
GNRH Receptor
MAO
Lipoxygenase
HIF
S1P Receptor
CFTR
Guanylate cyclase
TLR
Antifolate
P2X Receptor
HMG-CoA Reductase
DHFR
DNA-PK
JNK
ATM/ATR
Vasopressin Receptor
Gamma-secretase
ROCK
Molecular Glues
Anti-infection
Wnt/beta-catenin
Cholinesterase (ChE)
GluR
Kras
Nrf2
ADC Cytotoxin
MRP
Proteasome
Hedgehog/Smoothened
Neurokinin receptor
Transferase
S6 Kinase
Antioxidant
NO Synthase
Isocitrate Dehydrogenase (IDH)
P2Y Receptor
PLK
Syk
Antiviral
IAP
ABC Transporter
Cannabinoid Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Kinesin
CSF-1R
Phospholipase
IDO
DNA Methyltransferase
BTK
Antifection
OX Receptor
Integrin
Smo
IκB/IKK
Ligand for E3 Ligase
Mdm2
MAPK
NADPH
CaMK
DNA
Sirtuin
Casein Kinase
Sigma receptor
Chloride channel
FXR
RIP kinase
PAK
Aromatase
NOD
Serine Protease
Angiotensin-converting Enzyme (ACE)
Pim
Thrombin
Histone Demethylase
Hydroxylase
Glutathione Peroxidase
Leukotriene Receptor
Tie-2
Cholecystokinin Receptor
IRAK
PD-1/PD-L1
GPCR19
NOD-like Receptor (NLR)
Monoamine Transporter
CCR
Serine/threonin kinase
Tyrosinase
IKZF
Fatty Acid Synthase
PGE Synthase
Aminopeptidase
Glucosidase
Photosensitizer
Ephrin Receptor
Oxytocin Receptor
GHSR
Glucagon Receptor
DPP-4
IFNAR
Telomerase
ribosome
Bradykinin Receptor
Xanthine Oxidase
CRM1
PYK2
Glutaminase
UGT
Wee1
Cuproptosis
c-Myc
CaSR
CRFR
GST
Amino Acids and Derivatives
RSV
YAP
Annexin A
Na-K-Cl cotransporter
Neuropeptide Y Receptor
PDK
AhR
PROTACs
LTR
PERK
Melatonin Receptor
Aryl Hydrocarbon Receptor
DNA gyrase
STING
FKBP
CGRP Receptor
Somatostatin
Thrombopoietin Receptor
Discoidin Domain Receptor (DDR)
Protease-activated Receptor
Reductase
Beta-Secretase
Decarboxylase
Adenosine Deaminase
Rho
NAMPT
Melanocortin Receptor
MicroRNA
ROR
Hexokinase
DUB
OAT
MT Receptor
transporter
NEDD8
ATP Citrate Lyase
NOS
Monocarboxylate transporter
KSP
Free radical scavengers
BCRP
p97
TOPK
Acyltransferase
Arginase
Factor Xa
Liver X Receptor
HCN Channel
Histone Acetyltransferase
Gap Junction Protein
Ligands for Target Protein for PROTAC
Galectin
Complement System
Cell wall
Necroptosis
Lipid
LPA Receptor
SGK
VDA
FAAH
Porcupine
CD73
Imidazoline Receptor
Cysteine Protease
IRE1
LDL
OXPHOS
MLK
MIF
Neurotensin Receptor
GlyT
PAD
Survivin
ASK
Methionine Adenosyltransferase (MAT)
Aquaporin
Thyroid hormone receptor(THR)
NPC1L1
Kisspeptin
Myosin
Thioredoxin
Glutathione reductase
Neprilysin
Na+/Ca2+ Exchanger
DYRK
gp120/CD4
GTPase
cAMP
PAI-1
MELK
Platelet aggregation
Lipase
Glucokinase
Immunology/Inflammation related
PAFR
MTH1
MNK
PI4K
KLF
Advanced Glycation End Products
BACE
OCT
Hck
Stemness kinase
GRK
Arp2/3 Complex
ACK1
BMI-1
Hydrogenase
Factor VIIa
N-Acetylglucosaminyltransferase
NR4A
Adiponectin Receptor
Anion Exchanger
PROTAC Linker
Hippo pathway
MALT
PTEN
Cadherin
GluCls
Pyroptosis
RXFP receptor
NADPH-oxidase
Vitamin
PGC-1α

Keywords