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细胞因子抑制剂库

细胞因子抑制剂库

产品编号 L3600 Cytokine Inhibitor Library
  库化合物信息   Excel SDF

细胞因子是与维持免疫平衡相关的小分泌蛋白,与多种自身免疫和炎性疾病的发病机理有关。阻断细胞因子或其受体的生物制剂已经显著改善了这些病症的治疗方法,尽管如此,仍有一些患者对这些药物没有反应或者没有达到理想效果。

细胞因子通常与膜特异受体结合,激活相关信号途径,调控基因表达和细胞功能,例如白细胞介素,干扰素(IFN)和肿瘤坏死因子(TNF)等。转导细胞因子信号的常见途径有:JAK-STA、NF-kB、MAPKPI3K 等,随着研究的深入针对上述途径的小分子抑制剂越来越多,有些已经批准上市,我们精选了 613 个细胞因子相关化合物组成TargetMol 细胞因子抑制剂库,其靶点涉及多种不同功能的细胞因子,适用于高通量、高内涵筛选。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 613个与细胞因子紧密相关的化合物集合,是高通量、高内涵筛选的良好载体;
  • 靶点涵盖不同功能的细胞因子,包括白细胞介素(IL)、集落刺激因子CSF(CSF)、干扰素(IFN)、肿瘤坏死因子(TNF)、转化生长因子-β家族(TGF-β family)、生长因子(GF)、趋化因子(chemokinefamily);
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L3600)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

VEGFR (132)
EGFR (131)
TNF (81)
Apoptosis (80)
PDGFR (79)
FGFR (72)
Autophagy (61)
IL Receptor (60)
c-Kit (54)
TGF-beta/Smad (49)
c-Met/HGFR (47)
FLT (44)
Src (33)
CXCR (31)
NF-κB (30)
CCR (29)
Interleukin (28)
ALK (27)
IGF-1R (27)
HER (26)
Bcr-Abl (22)
c-RET (19)
JAK (17)
COX (16)
Endogenous Metabolite (16)
c-Fms (16)
HIV Protease (15)
Raf (14)
Antibacterial (14)
TAM Receptor (13)
RIP kinase (12)
Potassium Channel (12)
CDK (12)
CSF-1R (11)
Aurora Kinase (9)
p38 MAPK (9)
IFNAR (8)
STAT (8)
Tyrosine Kinases (8)
ERK (8)
Drug Metabolite (7)
FAK (7)
Parasite (7)
Trk receptor (7)
Ferroptosis (6)
NO Synthase (6)
5-HT Receptor (6)
DNA/RNA Synthesis (6)
BTK (6)
Reactive Oxygen Species (6)
Tyrosinase (6)
MEK (5)
JNK (5)
Influenza Virus (5)
Akt (5)
PKC (5)
ROS (5)
IκB/IKK (5)
PDE (5)
Caspase (5)
P450 (4)
PI3K (4)
TLR (4)
PKA (4)
Sodium Channel (4)
S6 Kinase (4)
Chk (4)
MMP (4)
MLK (4)
Ephrin Receptor (4)
NOD (4)
Virus Protease (3)
Mitophagy (3)
AMPK (3)
STING (3)
Anti-infection (3)
Tie-2 (3)
NOS (3)
PPAR (3)
Discoidin Domain Receptor (DDR) (3)
HCV Protease (3)
NOD-like Receptor (NLR) (3)
Calcium Channel (3)
GSK-3 (3)
PLK (2)
Mitochondrial Metabolism (2)
mTOR (2)
P-gp (2)
MAPK (2)
Syk (2)
transporter (2)
PYK2 (2)
IRE1 (2)
Histamine Receptor (2)
GABA Receptor (2)
Hck (2)
Antifungal (2)
HDAC (2)
Chloride channel (2)
Casein Kinase (2)
Adrenergic Receptor (2)
ROCK (1)
c-Myc (1)
ROR (1)
Reverse Transcriptase (1)
CFTR (1)
Dehydrogenase (1)
SARS-CoV (1)
Serine Protease (1)
SGK (1)
SGLT (1)
Sirtuin (1)
DNA Alkylation (1)
cell cycle arrest (1)
LTR (1)
Proton pump (1)
Antibiotic (1)
AChR (1)
ACK (1)
VDA (1)
Adenosine Receptor (1)
TRP/TRPV Channel (1)
Annexin A (1)
Topoisomerase (1)
CaMK (1)
Antifection (1)
Antioxidant (1)
Antiviral (1)
ATPase (1)
BCL (1)
Beta Amyloid (1)
E1/E2/E3 Enzyme (1)
Epigenetic Reader Domain (1)
Prostaglandin Receptor (1)
AChE (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Integrin (1)
NAMPT (1)
NADPH-oxidase (1)
NADPH (1)
Na+/Ca2+ Exchanger (1)
MRP (1)
HSP (1)
MNK (1)
LDL (1)
Leukotriene Receptor (1)
Lipase (1)
Lipoxygenase (1)
Microtubule Associated (1)
iGluR (1)
Histone Acetyltransferase (1)
Progesterone Receptor (1)
Phospholipase (1)
LRRK2 (1)
Estrogen Receptor/ERR (1)
Estrogen/progestogen Receptor (1)
PKM (1)
FAAH (1)
Gap Junction Protein (1)
Glucocorticoid Receptor (1)
HIF/HIF Prolyl-Hydroxylase (1)
PGE Synthase (1)
PDK (1)
Glucokinase (1)
HBV (1)
PARP (1)
PAD (1)
Wnt/beta-catenin (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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